Search results (20 entries covering 7 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
GAKNAKOther4y8dBB2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman342
GAKNAKOther4c57BB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human348
GAKNAKOther4c57AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human340
GAKNAKOther4c57BA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human334
GAKNAKOther4c59AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human346
GAKNAKOther5y80AAgefitinibHuman10329
GAKNAKOther4y8dAA2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman344
GAKNAKOther4c59AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human337
GAKNAKOther5y7zAgefitinibHuman10332
GAKNAKOther4c57AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human341
GAKNAKOther4o38BA-Human338
GAKNAKOther5y7zBgefitinibHuman10331
GAKNAKOther4o38AB-Human335
GAKNAKOther4c58AB9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman333
GAKNAKOther4y8dBA2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman347
GAKNAKOther4o38AA-Human345
GAKNAKOther5y80ABgefitinibHuman10330
GAKNAKOther4c58AA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman336
GAKNAKOther4o38BB-Human343
GAKNAKOther4y8dAB2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman339