Search results (10 entries covering 6 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | A | A | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11691 | ||
| EIF2AK4 (GCN2) | PEK | Other | 8t7t | A | A | - | Human | 15229 | ||
| EIF2AK4 (GCN2) | PEK | Other | 6n3n | A | n-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-2,5-dichloro-3-(hydroxymethyl)benzene-1-sulfonamide | Human | 11690 | |||
| EIF2AK4 (GCN2) | PEK | Other | 7qwk | A | (2~{s})-~{n}-[(1~{s})-1-[4-[(6-pyridin-4-ylquinazolin-2-yl)amino]phenyl]ethyl]piperidine-2-carboxamide | Human | 14209 | |||
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | B | A | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11693 | ||
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | B | B | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11692 | ||
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | A | B | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11694 | ||
| EIF2AK4 (GCN2) | PEK | Other | 7qq6 | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 14116 | |||
| EIF2AK4 (GCN2) | PEK | Other | 8t7t | A | B | - | Human | 15230 | ||
| EIF2AK4 (GCN2) | PEK | Other | 6n3o | A | n-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-5-chloro-2-methoxypyridine-3-sulfonamide | Human | 11695 |