| GRK5 (GPRK5) | GRK | AGC | 6pjx | A | A | sangivamycin | Human | 13042 | |
| GRK5 (GPRK5) | GRK | AGC | 9brm | A | | (3z)-3-[(4-{[(2s)-2-hydroxy-2-(oxan-4-yl)ethyl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16142 | |
| GRK5 (GPRK5) | GRK | AGC | 9ckq | A | | - | Human | 16143 | |
| GRK5 (GPRK5) | GRK | AGC | 6pjx | A | B | sangivamycin | Human | 13041 | |
| GRK5 (GPRK5) | GRK | AGC | 4tnb | A | | sangivamycin | Human | 3276 | |
| GRK5 (GPRK5) | GRK | AGC | 9brh | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-({4-[(furan-3-carbonyl)amino]-3,5-dimethyl-1h-pyrrol-2-yl}methylidene)-2-oxo-3,7-dihydro-2h-indole-5-carboxamide | Human | 16144 | |
| GRK5 (GPRK5) | GRK | AGC | 9bre | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-[(4-{[(2s)-2-(furan-2-yl)-2-hydroxyacetyl]amino}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 16145 | |
| GRK5 (GPRK5) | GRK | AGC | 9cks | A | | adenosine-5'-triphosphate | Human | 16146 | |
| GRK5 (GPRK5) | GRK | AGC | 9bri | A | | (3z)-3-[(3,5-dimethyl-4-{[(2s)-5-oxooxolane-2-carbonyl]amino}-1h-pyrrol-2-yl)methylidene]-n-[(1r)-1-(4-fluorophenyl)ethyl]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 16147 | |
| GRK5 (GPRK5) | GRK | AGC | 9brg | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-({4-[(furan-2-carbonyl)amino]-3,5-dimethyl-1h-pyrrol-2-yl}methylidene)-2-oxo-3,7-dihydro-2h-indole-5-carboxamide | Human | 16148 | |
| GRK5 (GPRK5) | GRK | AGC | 9brl | A | | (3z)-3-({3,5-dimethyl-4-[(4-methylpiperidin-4-yl)carbamoyl]-1h-pyrrol-2-yl}methylidene)-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16149 | |
| GRK5 (GPRK5) | GRK | AGC | 9cko | A | A | sangivamycin | Human | 16150 | |
| GRK5 (GPRK5) | GRK | AGC | 9brj | A | | (4s)-n-{5-[(z)-(5-{[(1r)-1-(4-fluorophenyl)ethyl]carbamoyl}-2-oxo-2,7-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrol-3-yl}-2-methylimidazo[1,2-a]pyridine-3-carboxamide | Human | 16151 | |
| GRK5 (GPRK5) | GRK | AGC | 9cko | A | B | sangivamycin | Human | 16152 | |
| GRK5 (GPRK5) | GRK | AGC | 9mx2 | A | | sangivamycin | Human | 16153 | |
| GRK5 (GPRK5) | GRK | AGC | 9bro | A | | (3z)-3-[(4-{[(2s)-1-methoxypropan-2-yl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16154 | |
| GRK5 (GPRK5) | GRK | AGC | 9brf | A | | (3z)-3-{[3,5-dimethyl-4-(2-oxo-2-phenylacetamido)-1h-pyrrol-2-yl]methylidene}-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16155 | |
| GRK5 (GPRK5) | GRK | AGC | 9brn | A | | (3z)-3-[(4-{[2-(dimethylamino)ethyl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16156 | |
| GRK5 (GPRK5) | GRK | AGC | 9brk | A | | tert-butyl (3r)-3-({5-[(z)-(5-{[(1r)-1-(4-fluorophenyl)ethyl]carbamoyl}-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrol-3-yl}carbamoyl)piperazine-1-carboxylate | Human | 16157 | |
| GRK5 (GPRK5) | GRK | AGC | 9brp | A | | (3z)-3-[(4-{[(2r)-2-methoxypropyl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16158 | |
| GRK5 (GPRK5) | GRK | AGC | 8uaq | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-[(4-{[(2s)-2-(furan-2-yl)-2-hydroxyacetyl]amino}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 15092 | |
| GRK5 (GPRK5) | GRK | AGC | 8uap | A | | (3z)-3-{[4-(2-chloroacetamido)-3,5-dimethyl-1h-pyrrol-2-yl]methylidene}-n-[(1r)-1-(4-fluorophenyl)ethyl]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 15093 | |
| GRK5 (GPRK5) | GRK | AGC | 9ckp | A | | sangivamycin | Human | 16141 | |
| GRK5 (GPRK5) | GRK | AGC | 9ckr | A | | adenosine-5'-triphosphate | Human | 16159 | |
| GRK5 (GPRK5) | GRK | AGC | 4tnd | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3275 | |
