Search results (248 entries covering 108 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
GSK3BGSKCMGC8qjiAn-[4-[5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl]pyridin-2-yl]cyclopropanecarboxamideHuman15386
Gsk3b (GSK3B)GSKCMGC8vmgAAadenosine-5'-diphosphateMouse15397
Gsk3b (GSK3B)GSKCMGC8vmgABadenosine-5'-diphosphateMouse15396
Gsk3b (GSK3B)GSKCMGC8vmeAAadenosine-5'-diphosphateMouse15398
Gsk3b (GSK3B)GSKCMGC8vmeABadenosine-5'-diphosphateMouse15399
Gsk3b (GSK3B)GSKCMGC8vmfAAadenosine-5'-diphosphateMouse15400
Gsk3b (GSK3B)GSKCMGC8vmfABadenosine-5'-diphosphateMouse15401
GSK3BGSKCMGC3zrlBB7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman691
GSK3BGSKCMGC6y9sBA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12285
GSK3BGSKCMGC4j1rD(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman736
GSK3BGSKCMGC4j71BB(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman739
GSK3BGSKCMGC4iq6B6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amineHuman750
Gsk3b (GSK3B)GSKCMGC4nu1AAadenosine-5'-diphosphateMouse5699
GSK3BGSKCMGC7oy5AB~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman14119
GSK3BGSKCMGC7oy5AA~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman14118
GSK3BGSKCMGC5t31B(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9564
GSK3BGSKCMGC9hv3A2-oxidanylidene-~{n}-[3-(4-phenylpiperazin-1-yl)propyl]-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamideHuman15794
GSK3BGSKCMGC9x2yAA-Human15795
GSK3BGSKCMGC9hulA~{n}-[3-[4-[2,3-bis(chloranyl)phenyl]piperazin-1-yl]propyl]-2-oxidanylidene-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamideHuman15796
GSK3BGSKCMGC9fr6A3-[[[4-[(3-cyclopropyl-1~{h}-pyrazol-5-yl)amino]thieno[3,2-d]pyrimidin-2-yl]amino]methyl]benzamideHuman15797
GSK3BGSKCMGC9hukA~{n}-[4-[4-[2,3-bis(chloranyl)phenyl]piperazin-1-yl]butyl]-2-oxidanylidene-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamideHuman15800
GSK3BGSKCMGC9fr7A~{n}4-(5-cyclopropyl-1~{h}-pyrazol-3-yl)-~{n}2-(phenylmethyl)furo[3,2-d]pyrimidine-2,4-diamineHuman15801
GSK3BGSKCMGC9x2yAB-Human15802
GSK3BGSKCMGC9fr9A3-[[[4-[(3-cyclobutyl-1~{h}-pyrazol-5-yl)amino]furo[3,2-d]pyrimidin-2-yl]amino]methyl]benzamideHuman15798
GSK3BGSKCMGC9x2qAA-Human15799
GSK3BGSKCMGC9x2xAA-Human15803
GSK3BGSKCMGC9x2vAA-Human15804
GSK3BGSKCMGC9x2uAB-Human15805
GSK3BGSKCMGC9x2vAB-Human15806
GSK3BGSKCMGC9x2wA-Human15807
GSK3BGSKCMGC9x2xAB-Human15808
GSK3BGSKCMGC6tcuAA5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHuman12780
GSK3BGSKCMGC1j1cBadenosine-5'-diphosphateHuman677
GSK3BGSKCMGC6hk3BB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11424
GSK3BGSKCMGC3f7zAA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman743
GSK3BGSKCMGC9hm1An-(4-{5-[(2-aminoethyl)sulfamoyl]thiophen-2-yl}pyridin-2-yl)cyclopropanecarboxamideHuman15792
GSK3BGSKCMGC6hk4BA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11430
GSK3BGSKCMGC1q3dAstaurosporineHuman705
GSK3BGSKCMGC3zrmBA7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman753
GSK3BGSKCMGC3f7zBB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman670
GSK3BGSKCMGC6v6lAA1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-oneHuman11913
GSK3BGSKCMGC3f88BA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman744
GSK3BGSKCMGC1r0eAA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman733
GSK3BGSKCMGC3zrlAC7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman654
GSK3BGSKCMGC1q3dBstaurosporineHuman752
Gsk3b (GSK3B)GSKCMGC5airA-Mouse6863
GSK3BGSKCMGC9x2qAB-Human15789
GSK3BGSKCMGC4acgA2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamideHuman681
GSK3BGSKCMGC9fr5A~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)furo[3,2-d]pyrimidine-2,4-diamineHuman15790
GSK3BGSKCMGC4ptgBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman754
GSK3BGSKCMGC6hk4BB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11427
GSK3BGSKCMGC1gngB-Human700
GSK3BGSKCMGC5f94BA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6372
GSK3BGSKCMGC3sd0B3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHuman673
GSK3BGSKCMGC4ptgAA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman735
GSK3BGSKCMGC8djdAB2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHuman14668
GSK3BGSKCMGC5kpkB(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9731
GSK3BGSKCMGC3pupAruthenium octasporineHuman7207
GSK3BGSKCMGC6y9sAA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12286
GSK3BGSKCMGC8djcAB(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHuman14669
GSK3BGSKCMGC4achA3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamideHuman653
GSK3BGSKCMGC3gb2AB2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHuman734
GSK3BGSKCMGC3zrlBA7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman718
Gsk3b (GSK3B)GSKCMGC5airB-Mouse6864
GSK3BGSKCMGC3zrlBC7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman676
GSK3BGSKCMGC3f88AB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman679
GSK3BGSKCMGC4j71AA(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman642
GSK3BGSKCMGC5hlpBA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6646
GSK3BGSKCMGC1o9uA9-methyl-9h-purin-6-amineHuman708
GSK3BGSKCMGC4acdA3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamideHuman723
GSK3BGSKCMGC1q4lA2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acidHuman714
GSK3BGSKCMGC5hlpAB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6648
GSK3BGSKCMGC4achB3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamideHuman702
GSK3BGSKCMGC9x2uAA-Human15791
GSK3BGSKCMGC7u33AA3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHuman14198
GSK3BGSKCMGC3i4bBn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman629
GSK3BGSKCMGC1j1cAadenosine-5'-diphosphateHuman696
GSK3BGSKCMGC3m1sBBruthenium pyridocarbazoleHuman7208
GSK3BGSKCMGC7z1gA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14662
GSK3BGSKCMGC3f7zBC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman686
GSK3BGSKCMGC1pyxBphosphoaminophosphonic acid-adenylate esterHuman663
GSK3BGSKCMGC3zrkAC2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman697
GSK3BGSKCMGC4pteAAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman716
GSK3BGSKCMGC1r0eAB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman672
GSK3BGSKCMGC3pupBruthenium octasporineHuman7211
GSK3BGSKCMGC5t31A(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9565
GSK3BGSKCMGC5k5nB5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHuman7410
GSK3BGSKCMGC6gjoA(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHuman10974
GSK3BGSKCMGC3l1sB(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHuman713
GSK3BGSKCMGC1q41A(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman628
GSK3BGSKCMGC6v6lAB1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-oneHuman11912
GSK3BGSKCMGC9fr8A~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman15793
GSK3BGSKCMGC4nm0ABadenosine-5'-diphosphateHuman671
GSK3BGSKCMGC4ptcAA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman664
GSK3BGSKCMGC7sxhAB(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14784
GSK3BGSKCMGC3gb2AA2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHuman727
GSK3BGSKCMGC4nm3ABadenosine-5'-diphosphateHuman640
GSK3BGSKCMGC4accB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman669
GSK3BGSKCMGC3zdiA3,6-diamino-4-(2-chlorophenyl)thieno[2,3-b]pyridine-2,5-dicarbonitrileHuman748
GSK3BGSKCMGC4nm5AAadenosine-5'-diphosphateHuman755
GSK3BGSKCMGC5hlnAchir99021Human6649
GSK3BGSKCMGC7b6fAA3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHuman13069
GSK3BGSKCMGC7sxjAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14785
GSK3BGSKCMGC3sayAB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman661
GSK3BGSKCMGC6hk4AA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11429
GSK3BGSKCMGC4j71BA(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman641
GSK3BGSKCMGC6y9rAA~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHuman12287
GSK3BGSKCMGC4pteBAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman722
GSK3BGSKCMGC6hk4AB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11423
GSK3BGSKCMGC5k5nA5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHuman7411
GSK3BGSKCMGC2jldBAruthenium pyridocarbazoleHuman7205
GSK3BGSKCMGC2jldABruthenium pyridocarbazoleHuman7214
GSK3BGSKCMGC6h0uA(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHuman11049
GSK3BGSKCMGC3sayAA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman738
GSK3BGSKCMGC3f88AA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman741
GSK3BGSKCMGC8av1AA2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14706
GSK3BGSKCMGC8auzAA8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14707
GSK3BGSKCMGC3zrlAA7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman712
GSK3BGSKCMGC5hlpAA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6647
GSK3BGSKCMGC5kplBA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9728
GSK3BGSKCMGC8djeAA(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHuman14670
GSK3BGSKCMGC5oy4A~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHuman8621
GSK3BGSKCMGC3zrmBB7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman652
GSK3BGSKCMGC5f95A2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHuman6373
GSK3BGSKCMGC2jldAAruthenium pyridocarbazoleHuman7213
GSK3BGSKCMGC4afjBA5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman678
GSK3BGSKCMGC3zrmAC7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman724
GSK3BGSKCMGC4b7tA(5z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-methyl-2-(propan-2-ylamino)imidazol-4-oneHuman732
GSK3BGSKCMGC3zrkAA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman675
GSK3BGSKCMGC1uv5A6-bromoindirubin-3'-oximeHuman759
GSK3BGSKCMGC4j71AB(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman690
GSK3BGSKCMGC1q5kAn-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaHuman680
GSK3BGSKCMGC8auzAB8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14708
GSK3BGSKCMGC5kpmB(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9734
GSK3BGSKCMGC3zrlAB7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman725
GSK3BGSKCMGC6hk3BA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11422
GSK3BGSKCMGC7u31AA5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHuman14199
GSK3BGSKCMGC6hk7A3-azanyl-~{n}-(2-methoxyethyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11428
GSK3BGSKCMGC4ptcBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman747
GSK3BGSKCMGC4pteABn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman717
GSK3BGSKCMGC3zrkBA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman637
GSK3BGSKCMGC1r0eBA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman687
GSK3BGSKCMGC1h8fA-Human745
GSK3BGSKCMGC6y9sBB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12288
GSK3BGSKCMGC5f94BB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6371
GSK3BGSKCMGC4ptgBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman740
GSK3BGSKCMGC3l1sA(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHuman757
GSK3BGSKCMGC7u33AB3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHuman14200
GSK3BGSKCMGC5f94AB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6369
GSK3BGSKCMGC6y9rAB~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHuman12289
GSK3BGSKCMGC4afjAA5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman632
GSK3BGSKCMGC3f7zAC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman685
GSK3BGSKCMGC4acdB3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamideHuman692
GSK3BGSKCMGC3zrmAA7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman751
GSK3BGSKCMGC4afjAC5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman742
GSK3BGSKCMGC1q41B(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman658
GSK3BGSKCMGC1j1bBphosphoaminophosphonic acid-adenylate esterHuman657
GSK3BGSKCMGC1gngA-Human665
GSK3BGSKCMGC6hk3AA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11425
GSK3BGSKCMGC4j1rC(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman688
GSK3BGSKCMGC4afjBC5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman711
GSK3BGSKCMGC4ditAn-(pyridin-3-yl)-2-(thiophen-3-yl)-3h-imidazo[4,5-b]pyridine-7-carboxamideHuman689
GSK3BGSKCMGC7u31AB5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHuman14201
GSK3BGSKCMGC3m1sBAruthenium pyridocarbazoleHuman7210
GSK3BGSKCMGC4afjAB5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman683
GSK3BGSKCMGC1h8fB-Human666
GSK3BGSKCMGC4acgB2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamideHuman721
GSK3BGSKCMGC4ptcBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman758
GSK3BGSKCMGC4nm7ABadenosine-5'-diphosphateHuman684
GSK3BGSKCMGC3zrmAB7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman648
GSK3BGSKCMGC1q3wA9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-oneHuman635
GSK3BGSKCMGC5f94AA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6374
GSK3BGSKCMGC4nm5ABadenosine-5'-diphosphateHuman694
GSK3BGSKCMGC5hlpBB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6645
GSK3BGSKCMGC3sayBB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman710
GSK3BGSKCMGC8av1AB2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14709
GSK3BGSKCMGC1q5kBn-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaHuman651
GSK3BGSKCMGC3zrkBC2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman731
GSK3BGSKCMGC5kpkA(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9735
GSK3BGSKCMGC6hk3AB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11426
GSK3BGSKCMGC5oy4B~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHuman8622
GSK3BGSKCMGC2ow3Abis-(indole)maleimide pyridinophaneHuman698
GSK3BGSKCMGC1pyxAphosphoaminophosphonic acid-adenylate esterHuman645
GSK3BGSKCMGC5kplAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9730
GSK3BGSKCMGC3sd0A3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHuman720
GSK3BGSKCMGC1q3wB9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-oneHuman693
GSK3BGSKCMGC3f7zAB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman647
GSK3BGSKCMGC3f7zBA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman749
GSK3BGSKCMGC6gjoB(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHuman10973
GSK3BGSKCMGC4ptgAB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman634
GSK3BGSKCMGC3du8B(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman737
GSK3BGSKCMGC1i09B-Human638
GSK3BGSKCMGC6b8jABchir99021Human8659
GSK3BGSKCMGC4iq6A6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amineHuman728
GSK3BGSKCMGC7u2zAB(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14202
GSK3BGSKCMGC4nm0AAadenosine-5'-diphosphateHuman715
GSK3BGSKCMGC4j1rB(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman656
GSK3BGSKCMGC3du8A(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman701
GSK3BGSKCMGC7u2zAA(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14203
GSK3BGSKCMGC5hlnBchir99021Human6650
GSK3BGSKCMGC4pteBBn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman667
GSK3BGSKCMGC2ow3Bbis-(indole)maleimide pyridinophaneHuman649
GSK3BGSKCMGC1q4lB2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acidHuman655
GSK3BGSKCMGC8djeAB(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHuman14671
GSK3BGSKCMGC3sayBA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman682
GSK3BGSKCMGC1j1bAphosphoaminophosphonic acid-adenylate esterHuman707
GSK3BGSKCMGC6gn1A~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHuman9997
GSK3BGSKCMGC4nm7AAadenosine-5'-diphosphateHuman695
GSK3BGSKCMGC5kplBB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9733
GSK3BGSKCMGC4j1rA(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman709
GSK3BGSKCMGC2o5kA2-(2,4-dichloro-phenyl)-7-hydroxy-1h-benzoimidazole-4-carboxylic acid [2-(4-methanesulfonylamino-phenyl)-ethyl]-amideHuman633
GSK3BGSKCMGC7sxjAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14786
GSK3BGSKCMGC6y9sAB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12290
GSK3BGSKCMGC3q3bA4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman660
GSK3BGSKCMGC6b8jAAchir99021Human8658
GSK3BGSKCMGC7z1fA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14663
GSK3BGSKCMGC3zrmBC7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman706
GSK3BGSKCMGC6tcuAB5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHuman12781
GSK3BGSKCMGC7u36A(3s)-1-[(2-fluorophenoxy)acetyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14204
GSK3BGSKCMGC5kplAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9729
GSK3BGSKCMGC5f95B2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHuman6370
GSK3BGSKCMGC7sxhAA(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14787
GSK3BGSKCMGC8ff8A2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamideHuman14763
GSK3BGSKCMGC3zrkBB2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman662
GSK3BGSKCMGC3zrkAB2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman644
GSK3BGSKCMGC3f88BB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman756
GSK3BGSKCMGC7b6fAB3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHuman13070
GSK3BGSKCMGC4accA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman704
GSK3BGSKCMGC6gn1B~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHuman9996
GSK3BGSKCMGC2jldBBruthenium pyridocarbazoleHuman7209
GSK3BGSKCMGC8djcAA(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHuman14672
GSK3BGSKCMGC3q3bB4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman674
GSK3BGSKCMGC3m1sAAruthenium pyridocarbazoleHuman7212
GSK3BGSKCMGC3i4bAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman646
GSK3BGSKCMGC4nm3AAadenosine-5'-diphosphateHuman730
GSK3BGSKCMGC3m1sABruthenium pyridocarbazoleHuman7206
GSK3BGSKCMGC4ptcAB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman659
GSK3BGSKCMGC1i09A-Human630
GSK3BGSKCMGC5kpmA(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9732
GSK3BGSKCMGC1r0eBB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman639
GSK3BGSKCMGC8djdAA2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHuman14673
GSK3BGSKCMGC6h0uB(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHuman11050
GSK3BGSKCMGC4afjBB5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman726
Gsk3b (GSK3B)GSKCMGC6ae3D-Mouse10604
Gsk3b (GSK3B)GSKCMGC6ae3B2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-oneMouse10606
Gsk3b (GSK3B)GSKCMGC6ae3A2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-oneMouse10607
Gsk3b (GSK3B)GSKCMGC4nu1ABadenosine-5'-diphosphateMouse5700
Gsk3b (GSK3B)GSKCMGC6ae3C-Mouse10605