| INSR | InsR | TK | 1irk | A | A | - | Human | 596 | |
| INSR | InsR | TK | 4ibm | B | B | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 599 | |
| INSR | InsR | TK | 5e1s | A | B | (5r)-n-(1-{2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl}-1h-pyrazol-3-yl)-5,8-dimethyl-9-phenyl-6,8-dihydro-5h-pyrazolo[3,4-h]quinazolin-2-amine | Human | 6147 | |
| Insr (INSR) | InsR | TK | 8eyx | A | | - | Mouse | 14496 | |
| Insr (INSR) | InsR | TK | 8eyy | A | | - | Mouse | 14497 | |
| INSR | InsR | TK | 8u4b | A | | - | Human | 15258 | |
| INSR | InsR | TK | 8x2m | A | | - | Human | 16058 | |
| INSR | InsR | TK | 8dwn | A | | - | Human | 14975 | |
| Insr (INSR) | InsR | TK | 8dtl | B | | - | Mouse | 14362 | |
| INSR | InsR | TK | 4ibm | A | A | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 589 | |
| INSR | InsR | TK | 7bw7 | C | | - | Human | 13505 | |
| INSR | InsR | TK | 1p14 | A | | - | Human | 593 | |
| INSR | InsR | TK | 1gag | A | | - | Human | 586 | |
| INSR | InsR | TK | 4ibm | B | A | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 604 | |
| INSR | InsR | TK | 7bw8 | A | | - | Human | 13502 | |
| INSR | InsR | TK | 8xkm | A | | - | Human | 16054 | |
| INSR | InsR | TK | 5e1s | A | A | (5r)-n-(1-{2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl}-1h-pyrazol-3-yl)-5,8-dimethyl-9-phenyl-6,8-dihydro-5h-pyrazolo[3,4-h]quinazolin-2-amine | Human | 6146 | |
| INSR | InsR | TK | 3ekn | A | B | 2-fluoro-6-{[2-({2-methoxy-4-[4-(1-methylethyl)piperazin-1-yl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 594 | |
| INSR | InsR | TK | 8xkr | E | | - | Human | 16055 | |
| INSR | InsR | TK | 7bw8 | C | | - | Human | 13503 | |
| INSR | InsR | TK | 2auh | A | | - | Human | 584 | |
| INSR | InsR | TK | 3bu3 | A | | - | Human | 591 | |
| INSR | InsR | TK | 9dni | C | | - | Human | 16056 | |
| INSR | InsR | TK | 3eta | B | B | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 600 | |
| INSR | InsR | TK | 6pxw | A | | - | Human | 11593 | |
| INSR | InsR | TK | 3ekk | A | A | 2-[(2-{[1-(n,n-dimethylglycyl)-5-methoxy-1h-indol-6-yl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-6-fluoro-n-methylbenzamide | Human | 578 | |
| INSR | InsR | TK | 5hhw | A | B | 7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2~{r})-oxan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6522 | |
| INSR | InsR | TK | 4ibm | A | B | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 598 | |
| INSR | InsR | TK | 7pg4 | A | | - | Human | 14100 | |
| INSR | InsR | TK | 1ir3 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 602 | |
| INSR | InsR | TK | 7pg0 | A | | - | Human | 14097 | |
| INSR | InsR | TK | 8yys | C | | - | Human | 16050 | |
| INSR | InsR | TK | 9puv | A | | - | Human | 16051 | |
| INSR | InsR | TK | 8x06 | A | | - | Human | 16052 | |
| INSR | InsR | TK | 9dn6 | C | | - | Human | 16053 | |
| INSR | InsR | TK | 4xlv | A | | phosphomethylphosphonic acid adenylate ester | Human | 577 | |
| INSR | InsR | TK | 1rqq | A | | thiophosphoric acid o-((adenosyl-phospho)phospho)-s-acetamidyl-diester | Human | 7407 | |
| INSR | InsR | TK | 3ekn | A | A | 2-fluoro-6-{[2-({2-methoxy-4-[4-(1-methylethyl)piperazin-1-yl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 597 | |
| INSR | InsR | TK | 1rqq | B | | thiophosphoric acid o-((adenosyl-phospho)phospho)-s-acetamidyl-diester | Human | 7406 | |
| INSR | InsR | TK | 7pg2 | A | | - | Human | 14098 | |
| INSR | InsR | TK | 3bu6 | A | | - | Human | 601 | |
| INSR | InsR | TK | 3eta | A | A | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 590 | |
| INSR | InsR | TK | 3bu5 | A | | adenosine-5'-triphosphate | Human | 595 | |
| INSR | InsR | TK | 6pxw | B | | - | Human | 11591 | |
| INSR | InsR | TK | 7bw7 | A | | - | Human | 13504 | |
| INSR | InsR | TK | 8ysz | B | | - | Human | 16057 | |
| INSR | InsR | TK | 6pxv | C | | - | Human | 11590 | |
| INSR | InsR | TK | 6pxv | A | | - | Human | 11592 | |
| INSR | InsR | TK | 3ekk | A | B | 2-[(2-{[1-(n,n-dimethylglycyl)-5-methoxy-1h-indol-6-yl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-6-fluoro-n-methylbenzamide | Human | 581 | |
| INSR | InsR | TK | 2b4s | D | | - | Human | 583 | |
| INSR | InsR | TK | 3eta | A | B | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 579 | |
| INSR | InsR | TK | 2z8c | A | | [4-({5-(aminocarbonyl)-4-[(3-methylphenyl)amino]pyrimidin-2-yl}amino)phenyl]acetic acid | Human | 587 | |
| INSR | InsR | TK | 3eta | B | A | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 588 | |
| INSR | InsR | TK | 2b4s | B | | - | Human | 585 | |
| INSR | InsR | TK | 1i44 | A | | phosphomethylphosphonic acid adenylate ester | Human | 582 | |
| INSR | InsR | TK | 7pg3 | A | | - | Human | 14099 | |
| INSR | InsR | TK | 5hhw | A | A | 7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2~{r})-oxan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6523 | |
| INSR | InsR | TK | 1irk | A | B | - | Human | 603 | |
| Insr (INSR) | InsR | TK | 7sl7 | A | | - | Mouse | 14169 | |
| Insr (INSR) | InsR | TK | 7stj | A | | - | Mouse | 14170 | |
| Insr (INSR) | InsR | TK | 7sl6 | A | | - | Mouse | 14171 | |
| Insr (INSR) | InsR | TK | 7sl4 | A | | - | Mouse | 14172 | |
