Search results (42 entries covering 28 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
JAK2-bJakBTK6g3cAB2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10976
JAK2-bJakBTK6brwAA4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman10382
JAK2-bJakBTK6m9hAA4-({4-amino-6-[4-(2-hydroxyethyl)-1h-imidazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman10384
JAK2-bJakBTK6occA2-[4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenyl]-1,3-oxazole-4-carboxylic acidHuman12100
JAK2-bJakBTK6bssAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman10386
JAK2-bJakBTK5uszAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8043
JAK2-bJakBTK5ut0AB1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman8047
JAK2-bJakBTK6m9hAB4-({4-amino-6-[4-(2-hydroxyethyl)-1h-imidazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman10383
JAK2-bJakBTK5ut1AB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman8049
JAK2-bJakBTK5ut2AB2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman8039
JAK2-bJakBTK5ut2AA2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman8040
JAK2-bJakBTK5uszAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8048
JAK2-bJakBTK6g3cAA2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10978
JAK2-bJakBTK6brwAB4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman10377
JAK2-bJakBTK5ut5AAn-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamideHuman8042
JAK2-bJakBTK5i4nABadenosine-5'-triphosphateHuman6524
JAK2-bJakBTK5ut5ABn-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamideHuman8037
JAK2-bJakBTK6oblA[4-({5-amino-3-[(4-cyanophenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acidHuman12101
JAK2-bJakBTK5ut4A8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1h-pyrazol-4-yl)quinoxalineHuman8038
JAK2-bJakBTK5ut0AA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman8041
JAK2-bJakBTK6obfA[4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acidHuman12098
JAK2-bJakBTK5wimA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10385
JAK2-bJakBTK5wijA4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamideHuman10388
JAK2-bJakBTK6oavA5-amino-3-[(4-cyanophenyl)amino]-n-phenyl-1h-1,2,4-triazole-1-carboxamideHuman12099
JAK2-bJakBTK5ut3A5-phenyl-2-ureidothiophene-3-carboxamideHuman8044
JAK2-bJakBTK5ut6AB4-({4-amino-6-[3-(hydroxymethyl)-1h-pyrazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman8045
JAK2-bJakBTK5wikB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman10387
JAK2-bJakBTK4fvqAadenosine-5'-triphosphateHuman1224
JAK2-bJakBTK4fvrAadenosine-5'-triphosphateHuman1223
JAK2-bJakBTK5winA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman10378
JAK2-bJakBTK5wilA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman10379
JAK2-bJakBTK5ut6AA4-({4-amino-6-[3-(hydroxymethyl)-1h-pyrazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman8036
JAK2-bJakBTK5i4nAAadenosine-5'-triphosphateHuman6525
JAK2-bJakBTK6g3cBA2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10977
JAK2-bJakBTK6bs0AA4-(5-aminopyrazin-2-yl)-1h-pyrrolo[2,3-b]pyridin-6-amineHuman10380
JAK2-bJakBTK6bs0AB4-(5-aminopyrazin-2-yl)-1h-pyrrolo[2,3-b]pyridin-6-amineHuman10381
JAK2-bJakBTK5ut1AA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman8046
JAK2-bJakBTK6d2iA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10967
JAK2-bJakBTK6g3cBB2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10975
JAK2-bJakBTK6d2iB1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10966
JAK2-bJakBTK6obbA5-amino-n-phenyl-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carboxamideHuman12097
JAK2-bJakBTK4fvpA-Human1222