| KIT | PDGFR | TK | 6kla | A | B | n-[6-(4-ethylpiperazin-1-yl)-2-methyl-pyrimidin-4-yl]-5-pyridin-4-yl-1,3-thiazol-2-amine | Human | 11823 | |
| KIT | PDGFR | TK | 6mob | A | A | n-{4-chloro-5-[1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl]-2-fluorophenyl}-n'-phenylurea | Human | 11469 | |
| KIT | PDGFR | TK | 8pqe | A | B | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamide | Human | 15117 | |
| KIT | PDGFR | TK | 6xva | B | | ~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamide | Human | 12281 | |
| KIT | PDGFR | TK | 6gqm | B | | ~{n}-[4-[[5-fluoranyl-7-(2-methoxyethoxy)quinazolin-4-yl]amino]phenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10361 | |
| KIT | PDGFR | TK | 6gql | A | | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10362 | |
| KIT | PDGFR | TK | 1t46 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 404 | |
| KIT | PDGFR | TK | 6gqk | A | A | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10355 | |
| KIT | PDGFR | TK | 6hh1 | A | A | ~{n}-(2,3-dimethylphenyl)-5-(4-pyridin-4-yloxyphenyl)-4~{h}-1,2,4-triazol-3-amine | Human | 11629 | |
| KIT | PDGFR | TK | 8pq9 | A | A | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15118 | |
| KIT | PDGFR | TK | 7khk | A | | 4,5-dimethyl-n-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazole-3-carboxamide | Human | 13787 | |
| KIT | PDGFR | TK | 1pkg | A | | adenosine-5'-diphosphate | Human | 397 | |
| KIT | PDGFR | TK | 6gqk | B | B | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10360 | |
| KIT | PDGFR | TK | 7zw8 | A | B | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | 14624 | |
| KIT | PDGFR | TK | 7khg | A | B | 5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amine | Human | 13788 | |
| KIT | PDGFR | TK | 8dfm | A | | - | Human | 14677 | |
| KIT | PDGFR | TK | 8dfp | A | | - | Human | 14678 | |
| KIT | PDGFR | TK | 8pqa | A | A | 6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazine | Human | 15124 | |
| KIT | PDGFR | TK | 8pqb | A | B | (1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15120 | |
| KIT | PDGFR | TK | 8pqg | A | B | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15112 | |
| KIT | PDGFR | TK | 8pqc | A | A | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15122 | |
| KIT | PDGFR | TK | 8pqc | A | B | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15123 | |
| KIT | PDGFR | TK | 8pqe | A | A | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamide | Human | 15119 | |
| KIT | PDGFR | TK | 8s19 | A | B | staurosporine | Human | 15755 | |
| KIT | PDGFR | TK | 8s17 | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 15756 | |
| KIT | PDGFR | TK | 9sxf | A | A | 3-(aminocarbonylamino)-5-(3-fluorophenyl)-~{n}-[(3~{r})-pyrrolidin-3-yl]thiophene-2-carboxamide | Human | 15757 | |
| KIT | PDGFR | TK | 8s1a | A | A | 1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amine | Human | 15758 | |
| KIT | PDGFR | TK | 35ua | A | A | ~{n}-(3,4-dichlorophenyl)-2-[4-([1,2,4]triazolo[1,5-a]pyridin-7-yl)phenyl]ethanamide | Human | 15746 | |
| KIT | PDGFR | TK | 8s13 | A | A | - | Human | 15747 | |
| KIT | PDGFR | TK | 8s19 | A | A | staurosporine | Human | 15748 | |
| KIT | PDGFR | TK | 8s13 | A | B | - | Human | 15749 | |
| KIT | PDGFR | TK | 8s17 | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 15750 | |
| KIT | PDGFR | TK | 35ua | A | B | ~{n}-(3,4-dichlorophenyl)-2-[4-([1,2,4]triazolo[1,5-a]pyridin-7-yl)phenyl]ethanamide | Human | 15751 | |
| KIT | PDGFR | TK | 8s1b | A | A | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | 15752 | |
| KIT | PDGFR | TK | 9sxf | A | B | 3-(aminocarbonylamino)-5-(3-fluorophenyl)-~{n}-[(3~{r})-pyrrolidin-3-yl]thiophene-2-carboxamide | Human | 15753 | |
| KIT | PDGFR | TK | 8s16 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 15754 | |
| KIT | PDGFR | TK | 8pqd | A | A | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamide | Human | 15113 | |
| KIT | PDGFR | TK | 6gqj | A | B | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10354 | |
| KIT | PDGFR | TK | 4u0i | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 405 | |
| KIT | PDGFR | TK | 7khg | A | A | 5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amine | Human | 13786 | |
| KIT | PDGFR | TK | 3g0e | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 401 | |
| KIT | PDGFR | TK | 8pqg | A | A | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15114 | |
| KIT | PDGFR | TK | 6itv | A | A | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11822 | |
| KIT | PDGFR | TK | 8pqa | A | B | 6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazine | Human | 15115 | |
| KIT | PDGFR | TK | 6gqj | A | A | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10364 | |
| KIT | PDGFR | TK | 6xvb | A | | ~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12279 | |
| KIT | PDGFR | TK | 1pkg | B | | adenosine-5'-diphosphate | Human | 402 | |
| KIT | PDGFR | TK | 7zw8 | A | A | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | 14622 | |
| KIT | PDGFR | TK | 7khj | A | | 2-phenyl-5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 13789 | |
| KIT | PDGFR | TK | 6gqm | A | | ~{n}-[4-[[5-fluoranyl-7-(2-methoxyethoxy)quinazolin-4-yl]amino]phenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10359 | |
| KIT | PDGFR | TK | 8s16 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 15759 | |
| KIT | PDGFR | TK | 4hvs | A | | 5-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-n-[4-(trifluoromethyl)benzyl]pyridin-2-amine | Human | 403 | |
| KIT | PDGFR | TK | 9sxe | A | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 15760 | |
| KIT | PDGFR | TK | 6itt | A | B | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11824 | |
| KIT | PDGFR | TK | 6xv9 | B | | ~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12283 | |
| KIT | PDGFR | TK | 6kla | A | A | n-[6-(4-ethylpiperazin-1-yl)-2-methyl-pyrimidin-4-yl]-5-pyridin-4-yl-1,3-thiazol-2-amine | Human | 11825 | |
| KIT | PDGFR | TK | 6xva | A | | ~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamide | Human | 12284 | |
| KIT | PDGFR | TK | 6hh1 | A | B | ~{n}-(2,3-dimethylphenyl)-5-(4-pyridin-4-yloxyphenyl)-4~{h}-1,2,4-triazol-3-amine | Human | 11628 | |
| KIT | PDGFR | TK | 6xvb | B | | ~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12280 | |
| KIT | PDGFR | TK | 7zy6 | A | | 5-imidazo[1,2-a]pyridin-3-yl-~{n}-[(1~{r})-1-(6-pyrrolidin-1-ylpyridin-3-yl)ethyl]pyridin-3-amine | Human | 14623 | |
| KIT | PDGFR | TK | 6gql | B | | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10357 | |
| KIT | PDGFR | TK | 8pqf | A | A | methyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamate | Human | 15116 | |
| KIT | PDGFR | TK | 6itt | B | A | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11821 | |
| KIT | PDGFR | TK | 1t45 | A | A | - | Human | 399 | |
| KIT | PDGFR | TK | 6gqj | B | B | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10356 | |
| KIT | PDGFR | TK | 6xv9 | A | | ~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12282 | |
| KIT | PDGFR | TK | 6itt | B | B | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11820 | |
| KIT | PDGFR | TK | 6gqk | A | B | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10353 | |
| KIT | PDGFR | TK | 3g0e | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 398 | |
| KIT | PDGFR | TK | 1t45 | A | B | - | Human | 394 | |
| KIT | PDGFR | TK | 6mob | A | B | n-{4-chloro-5-[1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl]-2-fluorophenyl}-n'-phenylurea | Human | 11470 | |
| KIT | PDGFR | TK | 6gqk | B | A | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10363 | |
| KIT | PDGFR | TK | 8pqb | A | A | (1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15121 | |
| KIT | PDGFR | TK | 1t46 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 393 | |
| KIT | PDGFR | TK | 8pq9 | A | B | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15125 | |
| KIT | PDGFR | TK | 8pqd | A | B | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamide | Human | 15126 | |
| KIT | PDGFR | TK | 6itv | A | B | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11827 | |
| KIT | PDGFR | TK | 8dfq | A | | - | Human | 14679 | |
| KIT | PDGFR | TK | 3g0f | B | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 400 | |
| KIT | PDGFR | TK | 6itt | A | A | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11826 | |
| KIT | PDGFR | TK | 4u0i | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 396 | |
| KIT | PDGFR | TK | 6gqj | B | A | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10358 | |
| KIT | PDGFR | TK | 8pqf | A | B | methyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamate | Human | 15127 | |
| KIT | PDGFR | TK | 3g0f | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 395 | |
| KIT | PDGFR | TK | 8s1b | A | B | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | 15761 | |
| KIT | PDGFR | TK | 8s1a | A | B | 1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amine | Human | 15762 | |
