Search results (137 entries covering 87 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
MAP2K1STE7STE7f2xAphosphoaminophosphonic acid-adenylate esterHuman14243
MAP2K1STE7STE2p55A2-[(4-ethynyl-2-fluorophenyl)amino]-3,4-difluoro-n-(2-hydroxyethoxy)benzamideHuman3327
MAP2K1STE7STE6v2wBBphosphoaminophosphonic acid-adenylate esterHuman13017
MAP2K1STE7STE7m0tB5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHuman13512
MAP2K1STE7STE4mneABphosphomethylphosphonic acid adenylate esterHuman3307
MAP2K1STE7STE7m0vBAphosphoaminophosphonic acid-adenylate esterHuman13518
MAP2K1STE7STE4an9Aphosphomethylphosphonic acid adenylate esterHuman3330
MAP2K1STE7STE7b9lBAphosphoaminophosphonic acid-adenylate esterHuman13398
MAP2K1STE7STE6u2gAphosphomethylphosphonic acid adenylate esterHuman11574
MAP2K1STE7STE3vvhAAadenosine-5'-triphosphateHuman3288
MAP2K1STE7STE7b3mBphosphoaminophosphonic acid-adenylate esterHuman13363
MAP2K1STE7STE7pqvAB8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinolineHuman14158
MAP2K1STE7STE7m0yBphosphoaminophosphonic acid-adenylate esterHuman13513
MAP2K1STE7STE6q0jCA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11721
MAP2K1STE7STE3eqgAadenosine-5'-diphosphateHuman3304
MAP2K1STE7STE7mfdBn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHuman14076
MAP2K1STE7STE3e8nAadenosine-5'-triphosphateHuman3323
MAP2K1STE7STE7m0wBphosphoaminophosphonic acid-adenylate esterHuman13515
MAP2K1STE7STE4an3Aadenosine-5'-triphosphateHuman3295
MAP2K1STE7STE7xlpA(1~{r},3~{s})-3-[[6-[2-chloranyl-4-(4-methylpyrimidin-2-yl)oxy-phenyl]-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexan-1-amineHuman14644
MAP2K1STE7STE8chfE-Human15261
MAP2K1STE7STE3eqcAA2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamideHuman3280
MAP2K1STE7STE3dv3ABadenosine-5'-triphosphateHuman3311
MAP2K1STE7STE4arkAadenosine-5'-diphosphateHuman3299
MAP2K1STE7STE4mneHBphosphomethylphosphonic acid adenylate esterHuman3328
MAP2K1STE7STE6q0tCB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11717
MAP2K1STE7STE6q0jCB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11713
MAP2K1STE7STE5yt3Bphosphoaminophosphonic acid-adenylate esterHuman10694
MAP2K1STE7STE6q0tCA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11715
MAP2K1STE7STE4u80Aphosphoaminophosphonic acid-adenylate esterHuman3305
MAP2K1STE7STE4u81A8-[(4-cyclopropyl-2-fluorophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-7-carboxamideHuman3301
MAP2K1STE7STE3os3Aadenosine-5'-triphosphateHuman3281
MAP2K1STE7STE3slsBBphosphoaminophosphonic acid-adenylate esterHuman9484
MAP2K1STE7STE3ornAphosphoaminophosphonic acid-adenylate esterHuman3277
MAP2K1STE7STE7b9lAAphosphoaminophosphonic acid-adenylate esterHuman13402
MAP2K1STE7STE4mneDBphosphomethylphosphonic acid adenylate esterHuman3315
MAP2K1STE7STE9zdqBBphosphoaminophosphonic acid-adenylate esterHuman16178
MAP2K1STE7STE9uw4Bphosphoaminophosphonic acid-adenylate esterHuman16179
MAP2K1STE7STE9rtqCBphosphoaminophosphonic acid-adenylate esterHuman16180
MAP2K1STE7STE9rtsAAadenosine-5'-diphosphateHuman16182
MAP2K1STE7STE13dvC5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman16183
MAP2K1STE7STE9tyiB-Human16181
MAP2K1STE7STE9o0uBAn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHuman16196
MAP2K1STE7STE9tygAadenosine-5'-diphosphateHuman16197
MAP2K1STE7STE7umbBphosphoaminophosphonic acid-adenylate esterHuman14989
MAP2K1STE7STE3eqbABadenosine-5'-triphosphateHuman3310
MAP2K1STE7STE4anbA[3-(aminomethyl)-3-oxidanyl-azetidin-1-yl]-[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]methanoneHuman3302
MAP2K1STE7STE3zlwA(1r)-1-hydroxy-1-methyl-2,3,6,7-tetrahydro-1h,5h-pyrido[3,2,1-ij]quinolin-5-oneHuman3278
MAP2K1STE7STE3vvhCAadenosine-5'-triphosphateHuman3306
MAP2K1STE7STE3dy7Aadenosine-5'-triphosphateHuman3282
MAP2K1STE7STE3mblABadenosine-5'-diphosphateHuman3318
MAP2K1STE7STE8dgsBAphosphothiophosphoric acid-adenylate esterHuman14825
MAP2K1STE7STE8dgtBAphosphothiophosphoric acid-adenylate esterHuman14828
MAP2K1STE7STE8dgsBBphosphothiophosphoric acid-adenylate esterHuman14826
MAP2K1STE7STE8dgtBBphosphothiophosphoric acid-adenylate esterHuman14827
MAP2K1STE7STE9rtqCAphosphoaminophosphonic acid-adenylate esterHuman16173
MAP2K1STE7STE7m0vBBphosphoaminophosphonic acid-adenylate esterHuman13511
MAP2K1STE7STE3zm4A7-chloranyl-6-[(3s)-pyrrolidin-3-yl]oxy-2h-isoquinolin-1-oneHuman3303
MAP2K1STE7STE1s9jAadenosine-5'-triphosphateHuman3316
MAP2K1STE7STE7pqvAA8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinolineHuman14157
MAP2K1STE7STE6pp9BAphosphoaminophosphonic acid-adenylate esterHuman11716
MAP2K1STE7STE6nybBadenosine-5'-diphosphateHuman11719
MAP2K1STE7STE6v2wBAphosphoaminophosphonic acid-adenylate esterHuman13015
MAP2K1STE7STE4mneEBphosphomethylphosphonic acid adenylate esterHuman3286
MAP2K1STE7STE4mneAAphosphomethylphosphonic acid adenylate esterHuman3293
MAP2K1STE7STE6q0jDB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11718
MAP2K1STE7STE5yt3Dphosphoaminophosphonic acid-adenylate esterHuman10695
MAP2K1STE7STE4mneDAphosphomethylphosphonic acid adenylate esterHuman3313
MAP2K1STE7STE3slsBAphosphoaminophosphonic acid-adenylate esterHuman9487
MAP2K1STE7STE7m0xBAphosphoaminophosphonic acid-adenylate esterHuman13514
MAP2K1STE7STE3slsAAphosphoaminophosphonic acid-adenylate esterHuman9486
MAP2K1STE7STE4mneHAphosphomethylphosphonic acid adenylate esterHuman3319
MAP2K1STE7STE7b7rAphosphoaminophosphonic acid-adenylate esterHuman13397
MAP2K1STE7STE6pp9BBphosphoaminophosphonic acid-adenylate esterHuman11720
MAP2K1STE7STE3dv3AAadenosine-5'-triphosphateHuman3322
MAP2K1STE7STE7b94Bphosphoaminophosphonic acid-adenylate esterHuman13364
MAP2K1STE7STE3v04A4-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)-1h-indazole-5-carboxamideHuman3325
MAP2K1STE7STE4lmnAphosphoaminophosphonic acid-adenylate esterHuman3283
MAP2K1STE7STE9o0vBAn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHuman16175
MAP2K1STE7STE9mmrBphosphothiophosphoric acid-adenylate esterHuman16176
MAP2K1STE7STE9twbAadenosine-5'-diphosphateHuman16184
MAP2K1STE7STE9mmsBphosphothiophosphoric acid-adenylate esterHuman16177
MAP2K1STE7STE3eqfAk-252aHuman3317
MAP2K1STE7STE5yt3Aphosphoaminophosphonic acid-adenylate esterHuman10692
MAP2K1STE7STE3eqcAB2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamideHuman3300
MAP2K1STE7STE4mneEAphosphomethylphosphonic acid adenylate esterHuman3314
MAP2K1STE7STE3wigAphosphoaminophosphonic acid-adenylate esterHuman3329
MAP2K1STE7STE9uurAphosphoaminophosphonic acid-adenylate esterHuman16186
MAP2K1STE7STE5hzeAA(3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman7569
MAP2K1STE7STE7b9lBBphosphoaminophosphonic acid-adenylate esterHuman13399
MAP2K1STE7STE3vvhCBadenosine-5'-triphosphateHuman3287
MAP2K1STE7STE3eqbAAadenosine-5'-triphosphateHuman3324
MAP2K1STE7STE3vvhABadenosine-5'-triphosphateHuman3296
MAP2K1STE7STE3pp1ABadenosine-5'-triphosphateHuman3285
MAP2K1STE7STE3slsABphosphoaminophosphonic acid-adenylate esterHuman9485
MAP2K1STE7STE3vvhBAadenosine-5'-triphosphateHuman3321
MAP2K1STE7STE9uuxAphosphoaminophosphonic acid-adenylate esterHuman16187
MAP2K1STE7STE7b7rBphosphoaminophosphonic acid-adenylate esterHuman13400
MAP2K1STE7STE5eymAB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6969
MAP2K1STE7STE3eqdAphosphothiophosphoric acid-adenylate esterHuman3284
MAP2K1STE7STE5bx0Aethyl 2h-indazole-5-carboxylateHuman6300
MAP2K1STE7STE4u7zA5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHuman3297
MAP2K1STE7STE3zlyA3-amino-1h-indazole-4-carbonitrileHuman3320
MAP2K1STE7STE5hzeAB(3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman7570
MAP2K1STE7STE6q0jDA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11714
MAP2K1STE7STE3w8qAphosphothiophosphoric acid-adenylate esterHuman3298
MAP2K1STE7STE3vvhBBadenosine-5'-triphosphateHuman3289
MAP2K1STE7STE7xncA~{n}-[4-[[6-(3-chloranylpyridin-4-yl)-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexyl]ethanamideHuman14643
MAP2K1STE7STE3eqiAadenosine-5'-diphosphateHuman3308
MAP2K1STE7STE4an2AB[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanoneHuman3326
MAP2K1STE7STE3eqhA(2z)-bis{amino[(2-aminophenyl)sulfanyl]methylidene}butanedinitrileHuman3290
MAP2K1STE7STE3pp1AAadenosine-5'-triphosphateHuman3294
MAP2K1STE7STE7b3mAphosphoaminophosphonic acid-adenylate esterHuman13365
MAP2K1STE7STE3zlsA1h-pyrrolo[2,3-b]pyridine-3-carboxylic acidHuman3279
MAP2K1STE7STE9o0vBBn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHuman16185
MAP2K1STE7STE4an2AA[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanoneHuman3309
MAP2K1STE7STE3v01An-{[(2r)-2,3-dihydroxypropyl]oxy}-3-[(2-fluoro-4-iodophenyl)amino]furo[3,2-c]pyridine-2-carboxamideHuman3291
MAP2K1STE7STE9uw3Aphosphoaminophosphonic acid-adenylate esterHuman16190
MAP2K1STE7STE7m0zBphosphoaminophosphonic acid-adenylate esterHuman13516
MAP2K1STE7STE5eymBA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6968
MAP2K1STE7STE3zlxA7-choro-6-[(3r)-pyrrolidin-3-ylmethoxy]isoquinolin-1(2h)-oneHuman3312
MAP2K1STE7STE7m0uB5-[(4-bromo-2-fluorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHuman13517
MAP2K1STE7STE5yt3Cphosphoaminophosphonic acid-adenylate esterHuman10693
MAP2K1STE7STE9rtsABadenosine-5'-diphosphateHuman16191
MAP2K1STE7STE9o2zBn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHuman16192
MAP2K1STE7STE9rtrAphosphoaminophosphonic acid-adenylate esterHuman16194
MAP2K1STE7STE3mblAAadenosine-5'-diphosphateHuman3292
MAP2K1STE7STE7m0xBBphosphoaminophosphonic acid-adenylate esterHuman13519
MAP2K1STE7STE5eymBB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6967
MAP2K1STE7STE9zdqBAphosphoaminophosphonic acid-adenylate esterHuman16195
MAP2K1STE7STE5eymAA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6966
MAP2K1STE7STE7b9lABphosphoaminophosphonic acid-adenylate esterHuman13401
MAP2K1STE7STE9mmqBphosphothiophosphoric acid-adenylate esterHuman16189
MAP2K1STE7STE9ecuBA4-[2-chloro-3-(methylsulfamamido)phenoxy]-n-cyclopropyl-2-(2-fluoro-4-iodoanilino)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamideHuman16172
MAP2K1STE7STE9ecuBB4-[2-chloro-3-(methylsulfamamido)phenoxy]-n-cyclopropyl-2-(2-fluoro-4-iodoanilino)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamideHuman16174
MAP2K1STE7STE9o0uBBn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHuman16188
MAP2K1STE7STE9tyhBadenosine-5'-diphosphateHuman16193