Search results (29 entries covering 22 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PKMYT1 (MYT1)WEEOther8zudA2-azanyl-3-(2,6-dimethyl-3-oxidanyl-phenyl)-5-(2-morpholin-4-ylpyridin-4-yl)benzamideHuman15524
PKMYT1 (MYT1)WEEOther8ztxA2-azanyl-3-(2,6-dimethyl-3-oxidanyl-phenyl)-5-pyridin-4-yl-benzamideHuman15525
PKMYT1 (MYT1)WEEOther9lglA3-azanyl-7-chloranyl-4-(2-methyl-5-oxidanyl-phenyl)-1h-1,5-naphthyridin-2-oneHuman15526
PKMYT1 (MYT1)WEEOther9lidA4-[7-azanyl-8-(7-fluoranyl-1h-indazol-4-yl)-6-oxidanylidene-5h-1,5-naphthyridin-3-yl]-n,n-dimethyl-benzamideHuman15527
PKMYT1 (MYT1)WEEOther8d6fA(1m)-2-amino-1-(5-hydroxy-2-methylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman14297
PKMYT1 (MYT1)WEEOther8d6eAB(1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamideHuman14293
PKMYT1 (MYT1)WEEOther8d6eAA(1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamideHuman14295
PKMYT1 (MYT1)WEEOther8wjyAB[6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanoneHuman15007
PKMYT1 (MYT1)WEEOther5vd3An-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman8343
PKMYT1 (MYT1)WEEOther5vd1AAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman8337
PKMYT1 (MYT1)WEEOther3p1aAB-Human1217
PKMYT1 (MYT1)WEEOther5vcwB(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamideHuman8346
PKMYT1 (MYT1)WEEOther5vcyAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8345
PKMYT1 (MYT1)WEEOther5vcyAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8338
PKMYT1 (MYT1)WEEOther5vczAB4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8336
PKMYT1 (MYT1)WEEOther5vcxAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman8341
PKMYT1 (MYT1)WEEOther8d6cA(1p)-2-amino-6-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman14296
PKMYT1 (MYT1)WEEOther3p1aAA-Human1216
PKMYT1 (MYT1)WEEOther5vcvAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman8339
PKMYT1 (MYT1)WEEOther5vcwA(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamideHuman8335
PKMYT1 (MYT1)WEEOther5vd0A1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman8344
PKMYT1 (MYT1)WEEOther8d6dA(1p)-2-amino-5-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman14294
PKMYT1 (MYT1)WEEOther8wjyAA[6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanoneHuman15008
PKMYT1 (MYT1)WEEOther5vd1ABn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman8340
PKMYT1 (MYT1)WEEOther13lxA(4r)-1-cyclopentyl-4-(3-hydroxyphenyl)-1,4,5,7-tetrahydro-6h-pyrazolo[3,4-b]pyridin-6-oneHuman15528
PKMYT1 (MYT1)WEEOther8zulA2-azanyl-5-[2-[(3~{r})-3-azanylpyrrolidin-1-yl]pyridin-4-yl]-3-(2,6-dimethyl-3-oxidanyl-phenyl)benzamideHuman15529
PKMYT1 (MYT1)WEEOther8zu2A2-azanyl-5-[2-(1,4-diazepan-1-yl)pyridin-4-yl]-3-(2,6-dimethyl-3-oxidanyl-phenyl)benzamideHuman15530
PKMYT1 (MYT1)WEEOther13lwA(4s)-1-cyclopentyl-4-(3-hydroxyphenyl)-1,4,5,7-tetrahydro-6h-pyrazolo[3,4-b]pyridin-6-oneHuman15531
PKMYT1 (MYT1)WEEOther5vczAA4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8342