Search results (17 entries covering 13 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PDGFRA (PDGFRa)PDGFRTK8pqiAA(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15109
PDGFRA (PDGFRa)PDGFRTK8pqjAA-Human15106
PDGFRA (PDGFRa)PDGFRTK6joiA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHuman12102
PDGFRA (PDGFRa)PDGFRTK8pqiAB(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15104
PDGFRA (PDGFRa)PDGFRTK8pqjAB-Human15105
PDGFRA (PDGFRa)PDGFRTK5grnABn-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamideHuman9478
PDGFRA (PDGFRa)PDGFRTK8pqkAA-Human15110
PDGFRA (PDGFRa)PDGFRTK6jokAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman12105
PDGFRA (PDGFRa)PDGFRTK5k5xA-Human6962
PDGFRA (PDGFRa)PDGFRTK9sxgA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman15731
PDGFRA (PDGFRa)PDGFRTK6a32A-Human11327
PDGFRA (PDGFRa)PDGFRTK8xrrArh140Human15730
PDGFRA (PDGFRa)PDGFRTK8pqhA(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15107
PDGFRA (PDGFRa)PDGFRTK8pqkAB-Human15108
PDGFRA (PDGFRa)PDGFRTK6jojA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHuman12104
PDGFRA (PDGFRa)PDGFRTK5grnAAn-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamideHuman9479
PDGFRA (PDGFRa)PDGFRTK6jolA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman12103