Search results (8 entries covering 4 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
| NTRK3 (TRKC) | Trk | TK | 6kzc | A | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Human | 11696 | |||
| NTRK3 (TRKC) | Trk | TK | 3v5q | A | 1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]urea | Human | 102 | |||
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 100 | ||
| NTRK3 (TRKC) | Trk | TK | 3v5q | B | 1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]urea | Human | 97 | |||
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 101 | ||
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 98 | ||
| NTRK3 (TRKC) | Trk | TK | 6kzd | A | 3-[2-[6-(4-aminophenyl)imidazo[1,2-a]pyrazin-3-yl]ethynyl]-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-propan-2-yl-phenyl]benzamide | Human | 11697 | |||
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 99 |