Search results (24 entries covering 8 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
ULK1ULKOther4wnpBBn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1879
ULK1ULKOther4wnpDBn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1880
ULK1ULKOther4wnpBAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1872
ULK1ULKOther9f32AAn-[4-(1h-indazol-5-yl)phenyl]propanamideHuman15545
ULK1ULKOther6qasBBn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10933
ULK1ULKOther9se8AA~{n}4-cyclopropyl-~{n}2-(1,2,3,4-tetrahydroisoquinolin-6-yl)-5-(trifluoromethyl)pyrimidine-2,4-diamineHuman15546
ULK1ULKOther5ci7AAn-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamideHuman5974
ULK1ULKOther6qasBAn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10932
ULK1ULKOther6qasABn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10931
ULK1ULKOther4wnpCBn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1873
ULK1ULKOther6qasAAn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10930
ULK1ULKOther6mnhABn-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamideHuman10980
ULK1ULKOther9se8AB~{n}4-cyclopropyl-~{n}2-(1,2,3,4-tetrahydroisoquinolin-6-yl)-5-(trifluoromethyl)pyrimidine-2,4-diamineHuman15547
ULK1ULKOther4wnpDAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1875
ULK1ULKOther8sv9AA(4p)-4-[(2p)-2-(1,2,5,6-tetrahydropyridin-3-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n-(2,2,2-trifluoroethyl)thiophene-2-carboxamideHuman15222
ULK1ULKOther4wnpCAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1877
ULK1ULKOther4wnoAAn~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1881
ULK1ULKOther9f32ABn-[4-(1h-indazol-5-yl)phenyl]propanamideHuman15548
ULK1ULKOther6mnhAAn-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamideHuman10979
ULK1ULKOther4wnpABn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1874
ULK1ULKOther5ci7ABn-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamideHuman5973
ULK1ULKOther8sv9AB(4p)-4-[(2p)-2-(1,2,5,6-tetrahydropyridin-3-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n-(2,2,2-trifluoroethyl)thiophene-2-carboxamideHuman15223
ULK1ULKOther4wnoABn~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1876
ULK1ULKOther4wnpAAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1878