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Search results (159 entries covering 121 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PIK3CA (p110a)PIKAtypical8twyA1-(4-{[2-(4-{(4p)-4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-[(3s)-3-methylmorpholin-4-yl]-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethoxy]methyl}piperidin-1-yl)prop-2-en-1-oneHuman15392
PIK3CA (p110a)PIKAtypical8exoAB1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamideHuman14534
PIK3CA (p110a)PIKAtypical8exlAA2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman14537
PIK3CA (p110a)PIKAtypical8exoAA1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamideHuman14541
PIK3CA (p110a)PIKAtypical8exvAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14542
PIK3CA (p110a)PIKAtypical8gudAA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14535
PIK3CA (p110a)PIKAtypical7pg6AA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14348
PIK3CA (p110a)PIKAtypical7mlkAA4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamideHuman14216
PIK3CA (p110a)PIKAtypical7tz7AA(4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-oneHuman14223
PIK3CA (p110a)PIKAtypical8tsdA-Human15090
PIK3CA (p110a)PIKAtypical8v8hA(2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamideHuman15249
PIK3CA (p110a)PIKAtypical7mynAB-Human13964
PIK3CA (p110a)PIKAtypical8v8iA(2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamideHuman15248
PIK3CA (p110a)PIKAtypical8v8uA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman15250
PIK3CA (p110a)PIKAtypical8v8vA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman15252
PIK3CA (p110a)PIKAtypical8v8jA(2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamideHuman15251
PIK3CA (p110a)PIKAtypical4ovuAB-Human9271
PIK3CA (p110a)PIKAtypical6pysAB(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11576
PIK3CA (p110a)PIKAtypical4ovvA-Human9307
PIK3CA (p110a)PIKAtypical7mlkAB4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamideHuman14217
PIK3CA (p110a)PIKAtypical4ovuAA-Human9291
PIK3CA (p110a)PIKAtypical5sxbA-Human9282
PIK3CA (p110a)PIKAtypical5swoA-Human9303
PIK3CA (p110a)PIKAtypical8tgdABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14970
PIK3CA (p110a)PIKAtypical8tu6A-Human14971
PIK3CA (p110a)PIKAtypical8ilsABn-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14968
PIK3CA (p110a)PIKAtypical8ilvAn-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[3-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14974
PIK3CA (p110a)PIKAtypical8w9bA-Human15273
PIK3CA (p110a)PIKAtypical8w9aA-Human15274
PIK3CA (p110a)PIKAtypical5fi4AB~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamideHuman9309
PIK3CA (p110a)PIKAtypical8ow2AA-Human14765
Pik3ca (p110a)PIKAtypical4a55Apik-108Mouse9403
PIK3CA (p110a)PIKAtypical8tscA-Human15084
PIK3CA (p110a)PIKAtypical8tsbA-Human15085
PIK3CA (p110a)PIKAtypical8tsaA-Human15087
PIK3CA (p110a)PIKAtypical8ts7A-Human15088
PIK3CA (p110a)PIKAtypical8ts9A-Human15089
PIK3CA (p110a)PIKAtypical7myoBA-Human13962
PIK3CA (p110a)PIKAtypical5fi4AA~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamideHuman9302
PIK3CA (p110a)PIKAtypical6oacA4-(difluoromethyl)-5-{4-[(3s)-3-methylmorpholin-4-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}pyridin-2-amineHuman11381
PIK3CA (p110a)PIKAtypical4tuuA-Human9281
PIK3CA (p110a)PIKAtypical5ul1AB3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamideHuman9308
PIK3CA (p110a)PIKAtypical5sxfA-Human9284
PIK3CA (p110a)PIKAtypical8tduABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14969
PIK3CA (p110a)PIKAtypical8ts8A-Human15086
PIK3CA (p110a)PIKAtypical7jiuAB(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13761
PIK3CA (p110a)PIKAtypical5sxeA-Human9280
PIK3CA (p110a)PIKAtypical5xghA3-[(4-fluorophenyl)methylamino]-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenolHuman9864
PIK3CA (p110a)PIKAtypical4wafAAn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9288
PIK3CA (p110a)PIKAtypical5sxkA-Human9296
PIK3CA (p110a)PIKAtypical7k6mAB2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylateHuman13227
PIK3CA (p110a)PIKAtypical7r9yAn-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-n-methyl-1-(prop-2-enoyl)piperidine-4-carboxamideHuman14179
PIK3CA (p110a)PIKAtypical3hhmA(1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetateHuman9275
PIK3CA (p110a)PIKAtypical5sxjA-Human9301
PIK3CA (p110a)PIKAtypical5dxtA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman9299
PIK3CA (p110a)PIKAtypical9xw5AB-Human16019
PIK3CA (p110a)PIKAtypical5xgjA3-(4-morpholin-4-ylfuro[3,2-d]pyrimidin-2-yl)-5-[(phenylmethyl)amino]phenolHuman9863
PIK3CA (p110a)PIKAtypical8ow2AB-Human14764
PIK3CA (p110a)PIKAtypical9b4sA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman16024
PIK3CA (p110a)PIKAtypical8dcpAA-Human14380
PIK3CA (p110a)PIKAtypical5swtA-Human9273
PIK3CA (p110a)PIKAtypical4zopAA(2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamideHuman9298
PIK3CA (p110a)PIKAtypical5xgiA3-azanyl-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenolHuman9865
PIK3CA (p110a)PIKAtypical5swpA-Human9293
PIK3CA (p110a)PIKAtypical5sxdA-Human9304
PIK3CA (p110a)PIKAtypical9xw7AB-Human16025
PIK3CA (p110a)PIKAtypical5dxhAmethyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamateHuman9310
PIK3CA (p110a)PIKAtypical4zopAB(2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamideHuman9312
PIK3CA (p110a)PIKAtypical8sbcAB(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridineHuman14842
PIK3CA (p110a)PIKAtypical7myoBB-Human13965
PIK3CA (p110a)PIKAtypical7pg6AB(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14349
PIK3CA (p110a)PIKAtypical4yknAA3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acidHuman9283
PIK3CA (p110a)PIKAtypical6nctA-Human11221
PIK3CA (p110a)PIKAtypical8ilrABn-[(2s)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14973
PIK3CA (p110a)PIKAtypical9nidA-Human16026
PIK3CA (p110a)PIKAtypical9nlcA-Human16027
PIK3CA (p110a)PIKAtypical9xw8AA-Human16028
PIK3CA (p110a)PIKAtypical9xw5AA-Human16029
PIK3CA (p110a)PIKAtypical9lwsA-Human16011
PIK3CA (p110a)PIKAtypical6gviAA3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman11656
PIK3CA (p110a)PIKAtypical9ni8A-Human16007
PIK3CA (p110a)PIKAtypical5itdA5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrileHuman9313
PIK3CA (p110a)PIKAtypical8tduAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14967
PIK3CA (p110a)PIKAtypical5sx9A-Human9305
PIK3CA (p110a)PIKAtypical8sbjAA(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridineHuman14839
PIK3CA (p110a)PIKAtypical9cmvA-Human16008
PIK3CA (p110a)PIKAtypical6gviAB3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman11654
PIK3CA (p110a)PIKAtypical4l1bA-Human9292
PIK3CA (p110a)PIKAtypical8bfuA-Human14613
PIK3CA (p110a)PIKAtypical8dd8A-Human14375
PIK3CA (p110a)PIKAtypical9lwrAA-Human16009
PIK3CA (p110a)PIKAtypical7k6nABtert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylateHuman13224
PIK3CA (p110a)PIKAtypical6gvfAB5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11658
PIK3CA (p110a)PIKAtypical6gvfAA5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11659
PIK3CA (p110a)PIKAtypical7mynAA-Human13963
PIK3CA (p110a)PIKAtypical8am0A(2r)-2-[[2-[(4s)-4-[bis(fluoranyl)methyl]-2-oxidanylidene-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl]amino]propanamideHuman15083
PIK3CA (p110a)PIKAtypical5swgA-Human9306
PIK3CA (p110a)PIKAtypical7r9vAn-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-1-(prop-2-enoyl)piperidine-4-carboxamideHuman14178
PIK3CA (p110a)PIKAtypical5swrA-Human9279
PIK3CA (p110a)PIKAtypical9ni7A-Human16010
PIK3CA (p110a)PIKAtypical7k71A2-(morpholin-4-yl)[4,5'-bipyrimidin]-2'-amineHuman13219
PIK3CA (p110a)PIKAtypical7pg5AA-Human14346
PIK3CA (p110a)PIKAtypical8dcpAB-Human14376
PIK3CA (p110a)PIKAtypical5ul1AA3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamideHuman9316
PIK3CA (p110a)PIKAtypical7k6oAB(3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamideHuman13206
PIK3CA (p110a)PIKAtypical7pg5AB-Human14347
PIK3CA (p110a)PIKAtypical8sbjAB(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridineHuman14840
PIK3CA (p110a)PIKAtypical5sxaA-Human9285
PIK3CA (p110a)PIKAtypical9b4tA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman16012
PIK3CA (p110a)PIKAtypical7jiuAA(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13760
PIK3CA (p110a)PIKAtypical4wafABn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9272
PIK3CA (p110a)PIKAtypical6gvhAA5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11657
PIK3CA (p110a)PIKAtypical8exlAB2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman14536
PIK3CA (p110a)PIKAtypical5ubrA1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-oneHuman9289
PIK3CA (p110a)PIKAtypical7k6mAA2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylateHuman13225
PIK3CA (p110a)PIKAtypical4jpsAA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman9317
PIK3CA (p110a)PIKAtypical8dcxA-Human14377
PIK3CA (p110a)PIKAtypical9ni5A-Human16013
PIK3CA (p110a)PIKAtypical9xw7AA-Human16014
PIK3CA (p110a)PIKAtypical7k6nAAtert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylateHuman13226
PIK3CA (p110a)PIKAtypical3zimA1-[4-[[2-(1h-indazol-4-yl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidin-6-yl]methyl]piperazin-1-yl]-6-methyl-hept-5-ene-1,4-dioneHuman9294
PIK3CA (p110a)PIKAtypical5sw8A-Human9274
PIK3CA (p110a)PIKAtypical4tv3A2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman9278
PIK3CA (p110a)PIKAtypical5uk8AA(r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholineHuman9295
PIK3CA (p110a)PIKAtypical5ukjAn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9277
PIK3CA (p110a)PIKAtypical7k6oAA(3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamideHuman13207
PIK3CA (p110a)PIKAtypical2rd0A-Human9287
PIK3CA (p110a)PIKAtypical4l23A3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenolHuman9290
PIK3CA (p110a)PIKAtypical6pysAA(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11575
PIK3CA (p110a)PIKAtypical4l2yA3-amino-5-[4-(morpholin-4-yl)pyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl]phenolHuman9276
PIK3CA (p110a)PIKAtypical6gvgA5-(6-azanyl-4-methyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11655
PIK3CA (p110a)PIKAtypical7tz7AB(4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-oneHuman14222
PIK3CA (p110a)PIKAtypical3hizA-Human9311
PIK3CA (p110a)PIKAtypical9nieA-Human16015
PIK3CA (p110a)PIKAtypical4jpsAB(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman9314
PIK3CA (p110a)PIKAtypical8exvABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14538
PIK3CA (p110a)PIKAtypical9lwqA-Human16016
PIK3CA (p110a)PIKAtypical9yf2An~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman16017
PIK3CA (p110a)PIKAtypical9ni3A-Human16018
PIK3CA (p110a)PIKAtypical5sxiA-Human9270
PIK3CA (p110a)PIKAtypical4yknAB3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acidHuman9315
PIK3CA (p110a)PIKAtypical8exuAA(2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamideHuman14539
PIK3CA (p110a)PIKAtypical8guaA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14540
PIK3CA (p110a)PIKAtypical9lwrAB-Human16020
PIK3CA (p110a)PIKAtypical5dxhDmethyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamateHuman9300
PIK3CA (p110a)PIKAtypical5sx8A-Human9269
PIK3CA (p110a)PIKAtypical8sbcAA(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridineHuman14841
PIK3CA (p110a)PIKAtypical9nifA-Human16021
PIK3CA (p110a)PIKAtypical8tgdAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14972
PIK3CA (p110a)PIKAtypical8dd4AA-Human14378
PIK3CA (p110a)PIKAtypical9c15A-Human16022
PIK3CA (p110a)PIKAtypical8dd4AB-Human14379
PIK3CA (p110a)PIKAtypical9xw8AB-Human16023
PIK3CA (p110a)PIKAtypical6gvhAB5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11653
PIK3CA (p110a)PIKAtypical5sxcA-Human9297
PIK3CA (p110a)PIKAtypical9ni4A-Human16030
PIK3CA (p110a)PIKAtypical8gubA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14543
PIK3CA (p110a)PIKAtypical8exuAB(2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamideHuman14544
PIK3CA (p110a)PIKAtypical5uk8AB(r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholineHuman9286
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