Search results (609 entries covering 376 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
MAPK14 (p38a)MAPKCMGC3k3iAA(3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinolineHuman5212
MAPK14 (p38a)MAPKCMGC1bl7A4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleHuman5193
Mapk14 (p38a)MAPKCMGC5r9pAB4-amino-n-(pyridin-2-yl)benzenesulfonamideMouse12576
Mapk14 (p38a)MAPKCMGC6y7wAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12071
Mapk14 (p38a)MAPKCMGC6y6vAA5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12066
Mapk14 (p38a)MAPKCMGC5r9bAA-Mouse12577
Mapk14 (p38a)MAPKCMGC5ra7AB4-methylbenzamideMouse12578
Mapk14 (p38a)MAPKCMGC6yk7AB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12164
Mapk14 (p38a)MAPKCMGC5r9zAA-Mouse12580
Mapk14 (p38a)MAPKCMGC6yk7AA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12163
Mapk14 (p38a)MAPKCMGC3p79A1-{3-tert-butyl-1-[2-(1,1-dioxidothiomorpholin-4-yl)-2-oxoethyl]-1h-pyrazol-5-yl}-3-naphthalen-2-ylureaMouse5849
Mapk14 (p38a)MAPKCMGC5ra3AB-Mouse12581
Mapk14 (p38a)MAPKCMGC6y4tAB5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12036
Mapk14 (p38a)MAPKCMGC4tyhBBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideMouse5844
Mapk14 (p38a)MAPKCMGC5r94AB-Mouse12589
Mapk14 (p38a)MAPKCMGC5r92AA(3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamideMouse12590
Mapk14 (p38a)MAPKCMGC6y8hAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12075
Mapk14 (p38a)MAPKCMGC5ra0AA[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12592
Mapk14 (p38a)MAPKCMGC6soiAB-Mouse11682
Mapk14 (p38a)MAPKCMGC5r9nAA[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12593
Mapk14 (p38a)MAPKCMGC5ra4AB-Mouse12594
Mapk14 (p38a)MAPKCMGC5r9eAA-Mouse12602
Mapk14 (p38a)MAPKCMGC5r90AA2,5-diphenyl-4~{h}-pyrazol-3-oneMouse12603
Mapk14 (p38a)MAPKCMGC5r9wAA~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamideMouse12605
Mapk14 (p38a)MAPKCMGC5r9jAA3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dioneMouse12609
Mapk14 (p38a)MAPKCMGC5r96AA-Mouse12610
Mapk14 (p38a)MAPKCMGC5r9kAA2,3-dihydro-1-benzoxepine-5-carboxylic acidMouse12611
Mapk14 (p38a)MAPKCMGC4loqDA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5835
Mapk14 (p38a)MAPKCMGC5ra5AB-Mouse12619
Mapk14 (p38a)MAPKCMGC6sovAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11677
Mapk14 (p38a)MAPKCMGC6ycwAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12153
Mapk14 (p38a)MAPKCMGC6splAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11687
Mapk14 (p38a)MAPKCMGC5r92AB(3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamideMouse12620
Mapk14 (p38a)MAPKCMGC5r8zAA6-methoxypyridine-3-carbothioamideMouse12575
Mapk14 (p38a)MAPKCMGC5ra1AB2-phenoxyacetamideMouse12579
Mapk14 (p38a)MAPKCMGC5r9cAA-Mouse12591
Mapk14 (p38a)MAPKCMGC5ra9AA4-chloranylthieno[3,2-d]pyrimidineMouse12601
Mapk14 (p38a)MAPKCMGC5r8xAB-Mouse12521
Mapk14 (p38a)MAPKCMGC5r9jAB3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dioneMouse12527
Mapk14 (p38a)MAPKCMGC5r98AB-Mouse12606
Mapk14 (p38a)MAPKCMGC6y7xAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12060
Mapk14 (p38a)MAPKCMGC5nzzEAphosphothiophosphoric acid-adenylate esterMouse9981
Mapk14 (p38a)MAPKCMGC4loqAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5872
Mapk14 (p38a)MAPKCMGC3p7cA1-[5-tert-butyl-3-({4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepan-1-yl}carbonyl)thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaMouse5838
Mapk14 (p38a)MAPKCMGC2gtmA8-(2-chlorophenylamino)-2-(2,6-difluorophenylamino)-9-ethyl-9h-purine-1,7-diiumMouse5867
Mapk14 (p38a)MAPKCMGC8vmhA(4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamideMouse16233
Mapk14 (p38a)MAPKCMGC6y80AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12080
Mapk14 (p38a)MAPKCMGC6splAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11683
MAPK14 (p38a)MAPKCMGC3hegAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5112
Mapk14 (p38a)MAPKCMGC7z9tAn-(2-cyclobutyl-1h-1,3-benzodiazol-5-yl)benzenesulfonamideMouse14799
Mapk14 (p38a)MAPKCMGC7z6iAA4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridineMouse14801
Mapk14 (p38a)MAPKCMGC8vmmA(4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideMouse16228
Mapk14 (p38a)MAPKCMGC5ra2AB1-(3-methylpyridin-2-yl)-1,4-diazepaneMouse12520
Mapk14 (p38a)MAPKCMGC4lopBA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5839
MAPK14 (p38a)MAPKCMGC6hwuAB-Human11249
Mapk14 (p38a)MAPKCMGC4lopCB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5855
MAPK14 (p38a)MAPKCMGC4zthAB6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazineHuman6707
Mapk14 (p38a)MAPKCMGC6sodAA-Mouse11673
Mapk14 (p38a)MAPKCMGC6y7wAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12065
Mapk14 (p38a)MAPKCMGC4looAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5832
Mapk14 (p38a)MAPKCMGC5r8yABthiophene-2-carbothioamideMouse12524
Mapk14 (p38a)MAPKCMGC5r97AB4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amineMouse12525
Mapk14 (p38a)MAPKCMGC6y4wAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12034
Mapk14 (p38a)MAPKCMGC6souAB2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanoneMouse11672
Mapk14 (p38a)MAPKCMGC4lopBB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5831
Mapk14 (p38a)MAPKCMGC5r8uAB3,4-dihydro-2~{h}-chromene-6-carboxamideMouse12583
MAPK14 (p38a)MAPKCMGC3fmnAA6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5196
MAPK14 (p38a)MAPKCMGC2lgcA4-Human5067
MAPK14 (p38a)MAPKCMGC3hv7A1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylureaHuman5223
MAPK14 (p38a)MAPKCMGC2bajA1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2,3-dichlorophenyl)ureaHuman5176
MAPK14 (p38a)MAPKCMGC3objA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman4994
MAPK14 (p38a)MAPKCMGC3zsgAAtak-715Human5033
Mapk14 (p38a)MAPKCMGC8efjA(4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamideMouse14995
MAPK14 (p38a)MAPKCMGC2i0hAA2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dioneHuman5062
MAPK14 (p38a)MAPKCMGC4aacAn-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamideHuman5048
MAPK14 (p38a)MAPKCMGC1r3cAB-Human4996
MAPK14 (p38a)MAPKCMGC3c5uA6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amineHuman5125
MAPK14 (p38a)MAPKCMGC3oc1A1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5019
MAPK14 (p38a)MAPKCMGC3obgA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5211
MAPK14 (p38a)MAPKCMGC5mz3AB~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8681
MAPK14 (p38a)MAPKCMGC5wjjAAn-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamideHuman9514
Mapk14 (p38a)MAPKCMGC4loqCA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5858
Mapk14 (p38a)MAPKCMGC3py3A-Mouse5857
MAPK14 (p38a)MAPKCMGC2fsoX-Human5117
MAPK14 (p38a)MAPKCMGC3qudAA{4-[(2-aminophenyl)amino]phenyl}(phenyl)methanoneHuman5006
Mapk14 (p38a)MAPKCMGC5r9iAAmethyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoateMouse12548
Mapk14 (p38a)MAPKCMGC6y81AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12079
Mapk14 (p38a)MAPKCMGC5r9kAB2,3-dihydro-1-benzoxepine-5-carboxylic acidMouse12549
Mapk14 (p38a)MAPKCMGC6sp9AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11686
Mapk14 (p38a)MAPKCMGC4tyhBAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideMouse5841
Mapk14 (p38a)MAPKCMGC2ewaAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse5870
Mapk14 (p38a)MAPKCMGC2ghlA3-(2-chlorophenyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)ureaMouse5871
MAPK14 (p38a)MAPKCMGC3mh2A-Human4985
Mapk14 (p38a)MAPKCMGC5ra4AA-Mouse12552
Mapk14 (p38a)MAPKCMGC6so4AA-Mouse11627
Mapk14 (p38a)MAPKCMGC5r9iABmethyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoateMouse12551
Mapk14 (p38a)MAPKCMGC7pvuAA-Mouse14747
Mapk14 (p38a)MAPKCMGC7pvuAB-Mouse14748
Mapk14 (p38a)MAPKCMGC7z6iAB4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridineMouse14800
Mapk14 (p38a)MAPKCMGC8acoAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15094
Mapk14 (p38a)MAPKCMGC8acoAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15095
Mapk14 (p38a)MAPKCMGC8acmA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15096
MAPK14 (p38a)MAPKCMGC3fkoA3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazoleHuman5075
MAPK14 (p38a)MAPKCMGC3oefXA-Human5163
MAPK14 (p38a)MAPKCMGC4e5aXB-Human5222
MAPK14 (p38a)MAPKCMGC6qdzAB1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11958
MAPK14 (p38a)MAPKCMGC3zyaAB2-amino-phenylamino-dibenzosuberoneHuman5089
MAPK14 (p38a)MAPKCMGC4ewqAA3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazineHuman5200
MAPK14 (p38a)MAPKCMGC4kiqBethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5013
MAPK14 (p38a)MAPKCMGC3zsiAB5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman4983
MAPK14 (p38a)MAPKCMGC3hp2AB1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-oneHuman5031
MAPK14 (p38a)MAPKCMGC3kq7AAn-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamideHuman5081
MAPK14 (p38a)MAPKCMGC3uvqABn-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamideHuman5214
MAPK14 (p38a)MAPKCMGC5omhA1-(3-chlorophenyl)-3-methyl-4~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11251
MAPK14 (p38a)MAPKCMGC4ehvAA-Human4997
MAPK14 (p38a)MAPKCMGC3mw1A8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxideHuman5072
MAPK14 (p38a)MAPKCMGC1zzlA6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-isopropyl[1,2,4]triazolo[4,3-a]pyridineHuman5249
MAPK14 (p38a)MAPKCMGC3gfeAn-cyclopropyl-3-{[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-4-yl]amino}-4-methylbenzamideHuman4991
MAPK14 (p38a)MAPKCMGC1bmkA4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazoleHuman5235
MAPK14 (p38a)MAPKCMGC3flyA6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5113
MAPK14 (p38a)MAPKCMGC3lffAB(4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acidHuman5120
MAPK14 (p38a)MAPKCMGC3lfeA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5173
MAPK14 (p38a)MAPKCMGC6qdzAA1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11956
MAPK14 (p38a)MAPKCMGC4eh8AA[3-(benzyloxy)phenyl]methanolHuman4978
MAPK14 (p38a)MAPKCMGC2lgcA8-Human5078
MAPK14 (p38a)MAPKCMGC3lfaAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman5018
MAPK14 (p38a)MAPKCMGC2onlB-Human5007
MAPK14 (p38a)MAPKCMGC4aa0ABn-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamideHuman5132
MAPK14 (p38a)MAPKCMGC3mh1A-Human5003
MAPK14 (p38a)MAPKCMGC3mptABn-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamideHuman5246
MAPK14 (p38a)MAPKCMGC5xyyA3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-4h-1,2,4-triazol-3-yl)phenolHuman9513
MAPK14 (p38a)MAPKCMGC3d7zAAn~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamideHuman5247
MAPK14 (p38a)MAPKCMGC3nwwA1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylureaHuman5068
MAPK14 (p38a)MAPKCMGC5wjjABn-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamideHuman9516
MAPK14 (p38a)MAPKCMGC2okrA-Human5136
MAPK14 (p38a)MAPKCMGC3kf7A3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamideHuman5201
MAPK14 (p38a)MAPKCMGC3hucABn-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamideHuman5111
MAPK14 (p38a)MAPKCMGC3gc7AB5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman5256
MAPK14 (p38a)MAPKCMGC6zwpAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman12698
MAPK14 (p38a)MAPKCMGC1oz1AA3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-olHuman5230
MAPK14 (p38a)MAPKCMGC2baqA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5184
MAPK14 (p38a)MAPKCMGC3uvpABn-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamideHuman5155
MAPK14 (p38a)MAPKCMGC3mgyA-Human5171
MAPK14 (p38a)MAPKCMGC3lfbAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)ureaHuman4998
MAPK14 (p38a)MAPKCMGC3nnvAB1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylureaHuman5046
MAPK14 (p38a)MAPKCMGC3zs5AB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4977
MAPK14 (p38a)MAPKCMGC3hv3AA1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5012
MAPK14 (p38a)MAPKCMGC3mvmA4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman4993
MAPK14 (p38a)MAPKCMGC4kinA5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5237
MAPK14 (p38a)MAPKCMGC6zqsA2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-oneHuman12986
MAPK14 (p38a)MAPKCMGC3fmmA6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5186
MAPK14 (p38a)MAPKCMGC4kinD5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5144
MAPK14 (p38a)MAPKCMGC6sfkAA~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamideHuman11617
MAPK14 (p38a)MAPKCMGC3odzX-Human5069
MAPK14 (p38a)MAPKCMGC4fa2AAtrans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanolHuman5150
MAPK14 (p38a)MAPKCMGC3fc1X5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5110
MAPK14 (p38a)MAPKCMGC3e92An-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamideHuman5149
MAPK14 (p38a)MAPKCMGC8yd9AB-Human15696
MAPK14 (p38a)MAPKCMGC3hv4B1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5064
MAPK14 (p38a)MAPKCMGC9r27A4-[4-[[4-chloranyl-3-(trifluoromethyl)phenyl]carbamoylamino]-3-fluoranyl-phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman15697
MAPK14 (p38a)MAPKCMGC1wbnAn-(3-tert-butyl-1h-pyrazol-5-yl)-n'-{4-chloro-3-[(pyridin-3-yloxy)methyl]phenyl}ureaHuman5257
MAPK14 (p38a)MAPKCMGC3rocA3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamideHuman5011
MAPK14 (p38a)MAPKCMGC3gcpAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5194
MAPK14 (p38a)MAPKCMGC3hv6A1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(2-morpholin-4-ylethoxy)phenyl]ureaHuman5101
MAPK14 (p38a)MAPKCMGC2yiwA1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)ureaHuman4988
MAPK14 (p38a)MAPKCMGC4e6cA-Human5015
MAPK14 (p38a)MAPKCMGC1di9A4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazolineHuman5251
MAPK14 (p38a)MAPKCMGC3gcqAB1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5053
MAPK14 (p38a)MAPKCMGC2lgcA5-Human5107
MAPK14 (p38a)MAPKCMGC3l8xAn,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman5041
MAPK14 (p38a)MAPKCMGC8a8mAphosphomethylphosphonic acid adenosyl esterHuman14289
MAPK14 (p38a)MAPKCMGC5etcA-Human6361
MAPK14 (p38a)MAPKCMGC1wfcA-Human4989
MAPK14 (p38a)MAPKCMGC3e93AB4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamideHuman5004
MAPK14 (p38a)MAPKCMGC3gcuBA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5175
MAPK14 (p38a)MAPKCMGC1yqjA6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazineHuman5152
MAPK14 (p38a)MAPKCMGC9cj5ApexmetinibHuman15698
MAPK14 (p38a)MAPKCMGC5o8uA-Human8381
MAPK14 (p38a)MAPKCMGC4e8aA-Human4979
MAPK14 (p38a)MAPKCMGC3mpaA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5026
MAPK14 (p38a)MAPKCMGC6tcaHBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12487
MAPK14 (p38a)MAPKCMGC2npqA-Human5205
MAPK14 (p38a)MAPKCMGC5xyxABn-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amineHuman9517
MAPK14 (p38a)MAPKCMGC3gcuAA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5032
MAPK14 (p38a)MAPKCMGC3hvcA4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridineHuman5054
MAPK14 (p38a)MAPKCMGC4a9yAn-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamideHuman5073
MAPK14 (p38a)MAPKCMGC4r3cAB6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazineHuman5036
MAPK14 (p38a)MAPKCMGC1wbwA3-(1-naphthylmethoxy)pyridin-2-amineHuman5179
MAPK14 (p38a)MAPKCMGC4eh7AA(3-phenoxyphenyl)methanolHuman5208
MAPK14 (p38a)MAPKCMGC3odyX-Human5233
MAPK14 (p38a)MAPKCMGC1wboA2-chlorophenolHuman5039
MAPK14 (p38a)MAPKCMGC8yd9AA-Human15699
MAPK14 (p38a)MAPKCMGC3d83An-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamideHuman5028
MAPK14 (p38a)MAPKCMGC6anlAAtak-715Human9515
MAPK14 (p38a)MAPKCMGC3mvlA4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5060
MAPK14 (p38a)MAPKCMGC2lgcA3-Human5040
MAPK14 (p38a)MAPKCMGC4e5aXA-Human5189
MAPK14 (p38a)MAPKCMGC3iw5An-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamideHuman5076
MAPK14 (p38a)MAPKCMGC4kinC5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5142
MAPK14 (p38a)MAPKCMGC3fskA3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman5008
MAPK14 (p38a)MAPKCMGC1oveAC1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5199
MAPK14 (p38a)MAPKCMGC6zwpAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman12699
MAPK14 (p38a)MAPKCMGC3lhjAn-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamideHuman5234
MAPK14 (p38a)MAPKCMGC4kipB2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamideHuman5180
MAPK14 (p38a)MAPKCMGC3fl4A6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidineHuman5151
MAPK14 (p38a)MAPKCMGC3s4qA3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamideHuman5133
MAPK14 (p38a)MAPKCMGC2zazAB4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehydeHuman5034
MAPK14 (p38a)MAPKCMGC3lfcA(4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acidHuman5160
MAPK14 (p38a)MAPKCMGC2zb1AAn-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamideHuman5038
MAPK14 (p38a)MAPKCMGC4f9yABn,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5017
MAPK14 (p38a)MAPKCMGC3ocgA5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamideHuman4984
MAPK14 (p38a)MAPKCMGC2balA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanoneHuman5260
MAPK14 (p38a)MAPKCMGC5etaB-Human7137
MAPK14 (p38a)MAPKCMGC2fstXB-Human5195
MAPK14 (p38a)MAPKCMGC3hv3AB1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5232
MAPK14 (p38a)MAPKCMGC4aa0AAn-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamideHuman5213
MAPK14 (p38a)MAPKCMGC3flnC6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5090
MAPK14 (p38a)MAPKCMGC3hv5BB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5137
MAPK14 (p38a)MAPKCMGC3gi3An-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamideHuman5226
MAPK14 (p38a)MAPKCMGC6sfiAB~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamideHuman11619
MAPK14 (p38a)MAPKCMGC6tcaFAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12489
MAPK14 (p38a)MAPKCMGC3hp2AA1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-oneHuman5217
MAPK14 (p38a)MAPKCMGC5mtxAA3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamideHuman8382
MAPK14 (p38a)MAPKCMGC3nnxA2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5002
MAPK14 (p38a)MAPKCMGC3ds6Bn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5188
MAPK14 (p38a)MAPKCMGC4l8mAAn-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamideHuman5005
MAPK14 (p38a)MAPKCMGC2bakAn-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamideHuman5114
MAPK14 (p38a)MAPKCMGC2fsmX-Human5044
MAPK14 (p38a)MAPKCMGC9cj2AA-Human15700
MAPK14 (p38a)MAPKCMGC3zshAA2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5216
MAPK14 (p38a)MAPKCMGC3hv5AB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5263
MAPK14 (p38a)MAPKCMGC1oukA4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidineHuman5146
MAPK14 (p38a)MAPKCMGC3hl7A2-{4-[5-(4-chlorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-3-yl]piperidin-1-yl}-2-oxoethanolHuman5236
MAPK14 (p38a)MAPKCMGC6ohdAB3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamideHuman11819
MAPK14 (p38a)MAPKCMGC4kipA2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamideHuman5159
MAPK14 (p38a)MAPKCMGC3ds6Cn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5182
MAPK14 (p38a)MAPKCMGC2lgcA9-Human5127
MAPK14 (p38a)MAPKCMGC3hllAA3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamideHuman5115
MAPK14 (p38a)MAPKCMGC4l8mABn-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamideHuman4992
MAPK14 (p38a)MAPKCMGC3fmlA6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5010
MAPK14 (p38a)MAPKCMGC3fmjA4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amineHuman5129
MAPK14 (p38a)MAPKCMGC6m9lA3-benzyl-6-[(2,4-difluorophenyl)amino]-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-oneHuman11255
MAPK14 (p38a)MAPKCMGC2y8oAB-Human5030
MAPK14 (p38a)MAPKCMGC3fmnAB6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman4995
MAPK14 (p38a)MAPKCMGC3hp5A5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5158
MAPK14 (p38a)MAPKCMGC3hegAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5218
MAPK14 (p38a)MAPKCMGC9cj4AC1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman15706
MAPK14 (p38a)MAPKCMGC4kinB5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5131
MAPK14 (p38a)MAPKCMGC1kv2A1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman5255
MAPK14 (p38a)MAPKCMGC3fmhA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5024
MAPK14 (p38a)MAPKCMGC3flwA6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman5153
MAPK14 (p38a)MAPKCMGC4kiqDethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5016
MAPK14 (p38a)MAPKCMGC4ehvAB-Human4981
MAPK14 (p38a)MAPKCMGC3mh0A-Human5124
MAPK14 (p38a)MAPKCMGC3hecAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman5035
Mapk14 (p38a)MAPKCMGC6ycuAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12152
MAPK14 (p38a)MAPKCMGC5n67AA-Human8523
MAPK14 (p38a)MAPKCMGC1r3cAA-Human5170
Mapk14 (p38a)MAPKCMGC2gtnA2-(2,6-difluorophenoxy)-n-(2-fluorophenyl)-9-isopropyl-9h-purin-8-amineMouse5860
Mapk14 (p38a)MAPKCMGC7be5A5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-methyl-pyrazole-4-carboxamideMouse13407
Mapk14 (p38a)MAPKCMGC5r9fAA-Mouse12526
Mapk14 (p38a)MAPKCMGC5larAA5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse6753
Mapk14 (p38a)MAPKCMGC4lopAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5861
Mapk14 (p38a)MAPKCMGC5nzzHBphosphothiophosphoric acid-adenylate esterMouse9984
Mapk14 (p38a)MAPKCMGC3p5kA1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylureaMouse5854
Mapk14 (p38a)MAPKCMGC4loqCB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5846
Mapk14 (p38a)MAPKCMGC6ycwAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12151
Mapk14 (p38a)MAPKCMGC6sodAB-Mouse11674
Mapk14 (p38a)MAPKCMGC6y4vAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12031
Mapk14 (p38a)MAPKCMGC5r90AB2,5-diphenyl-4~{h}-pyrazol-3-oneMouse12582
Mapk14 (p38a)MAPKCMGC6souAA2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanoneMouse11680
Mapk14 (p38a)MAPKCMGC5nzzFBphosphothiophosphoric acid-adenylate esterMouse9979
Mapk14 (p38a)MAPKCMGC4looAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5851
Mapk14 (p38a)MAPKCMGC4loqBB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5833
Mapk14 (p38a)MAPKCMGC5ra3AA-Mouse12599
MAPK14 (p38a)MAPKCMGC4r3cAA6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazineHuman5198
MAPK14 (p38a)MAPKCMGC3ctqAn-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamideHuman5220
MAPK14 (p38a)MAPKCMGC5tcoA3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-carboxamideHuman8031
MAPK14 (p38a)MAPKCMGC2gfsAB[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5050
MAPK14 (p38a)MAPKCMGC3hv5AA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5203
MAPK14 (p38a)MAPKCMGC3nnvAA1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylureaHuman5037
MAPK14 (p38a)MAPKCMGC3ds6An-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5074
MAPK14 (p38a)MAPKCMGC4dliA-Human5092
MAPK14 (p38a)MAPKCMGC2y8oAA-Human5079
MAPK14 (p38a)MAPKCMGC3oefXB-Human5231
MAPK14 (p38a)MAPKCMGC5tbeA~{n}-[2,4-bis(fluoranyl)-5-[[9-(2-morpholin-4-ylethylcarbamoyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulen-3-yl]amino]phenyl]thiophene-2-carboxamideHuman8032
MAPK14 (p38a)MAPKCMGC3k3jA2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamideHuman5047
MAPK14 (p38a)MAPKCMGC6sfjAC~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11618
MAPK14 (p38a)MAPKCMGC5omgAA3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11246
MAPK14 (p38a)MAPKCMGC3hrbA[3-amino-2-(2-methylphenyl)-1-oxidopyridin-4-yl](2,4-difluorophenyl)methanoneHuman5202
MAPK14 (p38a)MAPKCMGC1w84A3-(2-pyridin-4-ylethyl)-1h-indoleHuman5065
MAPK14 (p38a)MAPKCMGC2gfsAA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5227
MAPK14 (p38a)MAPKCMGC3u8wA3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamideHuman5192
MAPK14 (p38a)MAPKCMGC3hucAAn-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamideHuman5027
MAPK14 (p38a)MAPKCMGC4kiqAethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5141
MAPK14 (p38a)MAPKCMGC1wbtA3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamideHuman5082
MAPK14 (p38a)MAPKCMGC3k3iAB(3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinolineHuman5022
MAPK14 (p38a)MAPKCMGC3nnwAB2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5138
MAPK14 (p38a)MAPKCMGC5mtxAB3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamideHuman8379
MAPK14 (p38a)MAPKCMGC6sfiAA~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamideHuman11613
MAPK14 (p38a)MAPKCMGC6sfoAB5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman11621
MAPK14 (p38a)MAPKCMGC1w83An-[4-chloro-3-(pyridin-3-yloxymethyl)-phenyl]-3-fluoro-Human4986
MAPK14 (p38a)MAPKCMGC5mtyA~{n}-[2,4-bis(fluoranyl)-5-[[14-(2-hydroxyethylcarbamoyl)-2-oxidanylidene-6-tricyclo[9.4.0.0^{3,8}]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]amino]phenyl]thiophene-2-carboxamideHuman8383
MAPK14 (p38a)MAPKCMGC5o8vA-Human8380
MAPK14 (p38a)MAPKCMGC3lfbAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)ureaHuman5001
MAPK14 (p38a)MAPKCMGC5etfAA-Human7134
MAPK14 (p38a)MAPKCMGC3fsfA3-(2,6-dichlorophenyl)-7-({4-[(diethylamino)methoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman5097
MAPK14 (p38a)MAPKCMGC3fmkA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5209
MAPK14 (p38a)MAPKCMGC3uvqAAn-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamideHuman5183
MAPK14 (p38a)MAPKCMGC4eh9A-Human4982
MAPK14 (p38a)MAPKCMGC1bl6A4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazoleHuman5243
MAPK14 (p38a)MAPKCMGC6tcaDAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12486
MAPK14 (p38a)MAPKCMGC6sfkAB~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamideHuman11620
MAPK14 (p38a)MAPKCMGC3iphAB6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamideHuman5156
MAPK14 (p38a)MAPKCMGC3pg3AA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5122
MAPK14 (p38a)MAPKCMGC3flsA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5119
MAPK14 (p38a)MAPKCMGC3queA2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-oneHuman5095
MAPK14 (p38a)MAPKCMGC6hwtAB3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamideHuman11254
MAPK14 (p38a)MAPKCMGC3nnuAB2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamideHuman5059
MAPK14 (p38a)MAPKCMGC4kiqCethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5215
MAPK14 (p38a)MAPKCMGC3mh3A-Human5109
MAPK14 (p38a)MAPKCMGC3zsgABtak-715Human5098
MAPK14 (p38a)MAPKCMGC6sfjAB~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11616
MAPK14 (p38a)MAPKCMGC6qyxA-Human12127
MAPK14 (p38a)MAPKCMGC3flzA8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5204
MAPK14 (p38a)MAPKCMGC3hubA2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5029
MAPK14 (p38a)MAPKCMGC6hwvAA-Human11253
MAPK14 (p38a)MAPKCMGC2lgcA2-Human5093
MAPK14 (p38a)MAPKCMGC3newAA-Human5025
MAPK14 (p38a)MAPKCMGC3qudAB{4-[(2-aminophenyl)amino]phenyl}(phenyl)methanoneHuman5262
MAPK14 (p38a)MAPKCMGC3gc7AA5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman5061
MAPK14 (p38a)MAPKCMGC4eh3AnaringeninHuman5042
MAPK14 (p38a)MAPKCMGC3uvrAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}ureaHuman6880
MAPK14 (p38a)MAPKCMGC6hwuAA-Human11247
MAPK14 (p38a)MAPKCMGC5mz3AA~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8680
MAPK14 (p38a)MAPKCMGC4eh2A3-phenylquinazolin-4(3h)-oneHuman5244
MAPK14 (p38a)MAPKCMGC2fslX-Human5264
MAPK14 (p38a)MAPKCMGC2onlA-Human5177
MAPK14 (p38a)MAPKCMGC3ha8ABn~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamideHuman5187
MAPK14 (p38a)MAPKCMGC3mvmB4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5210
MAPK14 (p38a)MAPKCMGC3itzA4-chloro-n-cyclopropyl-3-{[1-(2,6-difluorophenyl)-1h-pyrazolo[3,4-d]pyridazin-4-yl]amino}benzamideHuman5135
MAPK14 (p38a)MAPKCMGC3kq7ABn-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamideHuman5057
MAPK14 (p38a)MAPKCMGC6qe1A1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{r})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11957
MAPK14 (p38a)MAPKCMGC3uvpAAn-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamideHuman5070
MAPK14 (p38a)MAPKCMGC3newAB-Human5248
MAPK14 (p38a)MAPKCMGC3hv4A1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5121
MAPK14 (p38a)MAPKCMGC3bx5An-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamideHuman5000
MAPK14 (p38a)MAPKCMGC3nnwAA2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5139
MAPK14 (p38a)MAPKCMGC2fstXA-Human5080
MAPK14 (p38a)MAPKCMGC6tcaBBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12488
MAPK14 (p38a)MAPKCMGC1kv1A1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5252
MAPK14 (p38a)MAPKCMGC2i0hAB2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dioneHuman5009
MAPK14 (p38a)MAPKCMGC3pg3AB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5096
MAPK14 (p38a)MAPKCMGC4aa4An-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamideHuman5045
MAPK14 (p38a)MAPKCMGC1wbsA3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamideHuman5258
MAPK14 (p38a)MAPKCMGC1m7qA1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-oneHuman5128
MAPK14 (p38a)MAPKCMGC4e6aA-Human5238
MAPK14 (p38a)MAPKCMGC3bv3A5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5207
MAPK14 (p38a)MAPKCMGC6tcaFBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12490
MAPK14 (p38a)MAPKCMGC3hecAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman5166
MAPK14 (p38a)MAPKCMGC3lffAA(4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acidHuman5140
MAPK14 (p38a)MAPKCMGC5etiA-Human6362
MAPK14 (p38a)MAPKCMGC6tcaBAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12491
MAPK14 (p38a)MAPKCMGC1w82An-[(3z)-5-tert-butyl-2-phenyl-1,2-dihydro-3h-pyrazol-3-ylidene]-n'-(4-chlorophenyl)ureaHuman5165
MAPK14 (p38a)MAPKCMGC4geoA-Human5190
MAPK14 (p38a)MAPKCMGC6tcaDBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12492
MAPK14 (p38a)MAPKCMGC3gcsAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5077
MAPK14 (p38a)MAPKCMGC3iw7A2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridineHuman5084
MAPK14 (p38a)MAPKCMGC3d7zABn~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamideHuman5108
MAPK14 (p38a)MAPKCMGC6sfoAA5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman11615
MAPK14 (p38a)MAPKCMGC2zazAA4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehydeHuman4980
MAPK14 (p38a)MAPKCMGC1r39A-Human5116
MAPK14 (p38a)MAPKCMGC5omgAB3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11245
MAPK14 (p38a)MAPKCMGC1a9uA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5229
MAPK14 (p38a)MAPKCMGC3flqA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5168
MAPK14 (p38a)MAPKCMGC3uvrAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}ureaHuman6879
MAPK14 (p38a)MAPKCMGC3o8tA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5167
MAPK14 (p38a)MAPKCMGC3o8pA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5071
MAPK14 (p38a)MAPKCMGC2yisA1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}ureaHuman5240
MAPK14 (p38a)MAPKCMGC3iw6ABethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylateHuman5154
MAPK14 (p38a)MAPKCMGC2qd9A1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanoneHuman5197
MAPK14 (p38a)MAPKCMGC3mvlB4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5091
MAPK14 (p38a)MAPKCMGC1oveAA1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5178
MAPK14 (p38a)MAPKCMGC3iphAA6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamideHuman4999
MAPK14 (p38a)MAPKCMGC6hwtAA3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamideHuman11248
MAPK14 (p38a)MAPKCMGC3l8sA3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamideHuman5055
MAPK14 (p38a)MAPKCMGC4f9wABn,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5106
MAPK14 (p38a)MAPKCMGC6tcaHAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12493
MAPK14 (p38a)MAPKCMGC3fi4A(2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-olHuman5051
MAPK14 (p38a)MAPKCMGC3o8uA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5250
MAPK14 (p38a)MAPKCMGC3s3iA3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamideHuman5169
MAPK14 (p38a)MAPKCMGC3dt1An-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamideHuman5086
MAPK14 (p38a)MAPKCMGC3lfdA1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5102
MAPK14 (p38a)MAPKCMGC3gcvAB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5174
MAPK14 (p38a)MAPKCMGC1ouyA1-(2,6-dichlorophenyl)-6-[(2,4-difluorophenyl)sulfanyl]-7-(1,2,3,6-tetrahydro-4-pyridinyl)-3,4-dihydropyrido[3,2-d]pyrimidin-2(1h)-oneHuman7258
MAPK14 (p38a)MAPKCMGC2zb1ABn-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamideHuman5103
MAPK14 (p38a)MAPKCMGC5etaA-Human7136
MAPK14 (p38a)MAPKCMGC2yixA1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)ureaHuman5143
MAPK14 (p38a)MAPKCMGC3zs5AA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4987
MAPK14 (p38a)MAPKCMGC8x3mAA-Human15701
MAPK14 (p38a)MAPKCMGC3rinAn-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamideHuman5239
MAPK14 (p38a)MAPKCMGC1wbvA3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamideHuman5148
MAPK14 (p38a)MAPKCMGC4f9yAAn,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5225
MAPK14 (p38a)MAPKCMGC2zb0ABn-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamideHuman5147
MAPK14 (p38a)MAPKCMGC3nnuAA2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamideHuman5094
MAPK14 (p38a)MAPKCMGC3zyaAA2-amino-phenylamino-dibenzosuberoneHuman5105
MAPK14 (p38a)MAPKCMGC4eh7AB(3-phenoxyphenyl)methanolHuman5020
MAPK14 (p38a)MAPKCMGC3iw6AAethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylateHuman4990
MAPK14 (p38a)MAPKCMGC1w7hA3-(benzyloxy)pyridin-2-amineHuman5023
MAPK14 (p38a)MAPKCMGC2okrD-Human5100
MAPK14 (p38a)MAPKCMGC9cj2AB-Human15702
MAPK14 (p38a)MAPKCMGC4aa5An-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamideHuman5206
MAPK14 (p38a)MAPKCMGC4fa2ABtrans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanolHuman5145
MAPK14 (p38a)MAPKCMGC6hwvAB-Human11250
MAPK14 (p38a)MAPKCMGC5n66A1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman8524
MAPK14 (p38a)MAPKCMGC2lgcA1-Human5021
MAPK14 (p38a)MAPKCMGC3gcuAB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5162
MAPK14 (p38a)MAPKCMGC6m95A(4-benzylpiperidin-1-yl)[2-methoxy-4-(methylsulfanyl)phenyl]methanoneHuman11252
MAPK14 (p38a)MAPKCMGC4eh8AB[3-(benzyloxy)phenyl]methanolHuman5014
MAPK14 (p38a)MAPKCMGC2lgcA10-Human5063
MAPK14 (p38a)MAPKCMGC2zb0AAn-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamideHuman5099
MAPK14 (p38a)MAPKCMGC6anlABtak-715Human9518
MAPK14 (p38a)MAPKCMGC3ds6Dn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5123
MAPK14 (p38a)MAPKCMGC5ml5A3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{h}-imidazol-5-yl]pyridin-2-yl]propanamideHuman7544
MAPK14 (p38a)MAPKCMGC2rg6A4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5228
MAPK14 (p38a)MAPKCMGC9cj4AA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman15703
MAPK14 (p38a)MAPKCMGC3ha8AAn~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamideHuman5253
MAPK14 (p38a)MAPKCMGC2lgcA6-Human5219
MAPK14 (p38a)MAPKCMGC3e93AA4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamideHuman5241
MAPK14 (p38a)MAPKCMGC9cj4AB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman15704
MAPK14 (p38a)MAPKCMGC3gcsAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5052
MAPK14 (p38a)MAPKCMGC4eh6An-phenylpyridine-3-carboxamideHuman5083
MAPK14 (p38a)MAPKCMGC3bv2A5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5191
MAPK14 (p38a)MAPKCMGC8x3mAB-Human15705
MAPK14 (p38a)MAPKCMGC3hllAB3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamideHuman5104
MAPK14 (p38a)MAPKCMGC3mptAAn-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamideHuman5224
MAPK14 (p38a)MAPKCMGC4e5bA-Human5221
MAPK14 (p38a)MAPKCMGC2lgcA7-Human5161
MAPK14 (p38a)MAPKCMGC5xyxAAn-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amineHuman9519
MAPK14 (p38a)MAPKCMGC4f9wAAn,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5130
MAPK14 (p38a)MAPKCMGC1zz2An-[3-(4-fluorophenoxy)phenyl]-4-[(2-hydroxybenzyl)amino]piperidine-1-sulfonamideHuman5164
MAPK14 (p38a)MAPKCMGC3gcuBB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5126
MAPK14 (p38a)MAPKCMGC3iw8A1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)ureaHuman5181
MAPK14 (p38a)MAPKCMGC4ewqAB3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazineHuman5245
MAPK14 (p38a)MAPKCMGC4eh4Aphenyl(piperidin-1-yl)methanoneHuman5043
MAPK14 (p38a)MAPKCMGC5etfAB-Human7135
MAPK14 (p38a)MAPKCMGC3fklAn-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamideHuman5172
MAPK14 (p38a)MAPKCMGC4eh5Abenzyl pyridine-3-carboxylateHuman5185
MAPK14 (p38a)MAPKCMGC5n67AB-Human8521
MAPK14 (p38a)MAPKCMGC4zthAA6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazineHuman6706
MAPK14 (p38a)MAPKCMGC1zyjA4-phenoxy-n-(pyridin-2-ylmethyl)benzamideHuman5058
MAPK14 (p38a)MAPKCMGC3fknA3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidineHuman5049
MAPK14 (p38a)MAPKCMGC6sfjAA~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11614
MAPK14 (p38a)MAPKCMGC1oveAB1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5087
MAPK14 (p38a)MAPKCMGC2rg5An-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5254
MAPK14 (p38a)MAPKCMGC5n65A2-phenyl-~{n}4-(2-thiophen-2-ylethyl)quinazoline-4,7-diamineHuman8525
MAPK14 (p38a)MAPKCMGC4dljA2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamineHuman5242
MAPK14 (p38a)MAPKCMGC5n63A-Human8526
MAPK14 (p38a)MAPKCMGC3gcpAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5157
MAPK14 (p38a)MAPKCMGC3hv5BA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5085
MAPK14 (p38a)MAPKCMGC1oz1AB3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-olHuman5261
MAPK14 (p38a)MAPKCMGC3zshAB2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5118
MAPK14 (p38a)MAPKCMGC6ohdAA3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamideHuman11818
MAPK14 (p38a)MAPKCMGC3gcvAA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5088
MAPK14 (p38a)MAPKCMGC5n64A-Human8527
MAPK14 (p38a)MAPKCMGC3gcqAA1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5066
MAPK14 (p38a)MAPKCMGC3od6X-Human5134
MAPK14 (p38a)MAPKCMGC5n68A-Human8522
MAPK14 (p38a)MAPKCMGC3zsiAA5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5056
Mapk14 (p38a)MAPKCMGC3p7aA1-[5-tert-butyl-2-(1,1-dioxidothiomorpholin-4-yl)thiophen-3-yl]-3-naphthalen-1-ylureaMouse5853
Mapk14 (p38a)MAPKCMGC5r9pAA4-amino-n-(pyridin-2-yl)benzenesulfonamideMouse12518
Mapk14 (p38a)MAPKCMGC5nzzHAphosphothiophosphoric acid-adenylate esterMouse9978
Mapk14 (p38a)MAPKCMGC5o90A4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse9525
Mapk14 (p38a)MAPKCMGC4ka3A-Mouse5852
Mapk14 (p38a)MAPKCMGC5nzzGBphosphothiophosphoric acid-adenylate esterMouse9982
Mapk14 (p38a)MAPKCMGC5uojA-Mouse7466
Mapk14 (p38a)MAPKCMGC5r9rAA4-acetyl-n-ethylpiperazine-1-carboxamideMouse12519
Mapk14 (p38a)MAPKCMGC5r9cAB-Mouse12522
Mapk14 (p38a)MAPKCMGC7bdoAB~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamideMouse13405
Mapk14 (p38a)MAPKCMGC5r9lAB(3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-olMouse12523
Mapk14 (p38a)MAPKCMGC7be4A5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse13406
Mapk14 (p38a)MAPKCMGC5r9vAB-Mouse12528
Mapk14 (p38a)MAPKCMGC5r97AA4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amineMouse12529
Mapk14 (p38a)MAPKCMGC6sotAA-Mouse11689
Mapk14 (p38a)MAPKCMGC5r9vAA-Mouse12530
Mapk14 (p38a)MAPKCMGC5nzzEBphosphothiophosphoric acid-adenylate esterMouse9980
Mapk14 (p38a)MAPKCMGC5r9sAA-Mouse12531
Mapk14 (p38a)MAPKCMGC5r94AA-Mouse12532
Mapk14 (p38a)MAPKCMGC4loqAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5836
Mapk14 (p38a)MAPKCMGC4lopCA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5847
Mapk14 (p38a)MAPKCMGC5r99AB3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12533
Mapk14 (p38a)MAPKCMGC3p4kA-Mouse5842
Mapk14 (p38a)MAPKCMGC6yjcAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12437
Mapk14 (p38a)MAPKCMGC5r8wAB-Mouse12534
Mapk14 (p38a)MAPKCMGC2puuA5-tert-butyl-2-(4-methylphenyl)-3-{[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]-1-naphthyl}amino)carbonyl]amino}-1h-pyrazol-2-iumMouse6866
Mapk14 (p38a)MAPKCMGC5r8wAA-Mouse12535
Mapk14 (p38a)MAPKCMGC1yw2A2-(ethoxymethyl)-4-(4-fluorophenyl)-3-[2-(2-hydroxyphenoxy)pyrimidin-4-yl]isoxazol-5(2h)-oneMouse5869
Mapk14 (p38a)MAPKCMGC6y7zAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12070
Mapk14 (p38a)MAPKCMGC5nzzGAphosphothiophosphoric acid-adenylate esterMouse9977
Mapk14 (p38a)MAPKCMGC6y81AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12073
Mapk14 (p38a)MAPKCMGC5r9rAB4-acetyl-n-ethylpiperazine-1-carboxamideMouse12536
Mapk14 (p38a)MAPKCMGC1lewA-Mouse5864
Mapk14 (p38a)MAPKCMGC4loqBA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5834
Mapk14 (p38a)MAPKCMGC6y4xAA5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12039
Mapk14 (p38a)MAPKCMGC5r9yAA3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12537
Mapk14 (p38a)MAPKCMGC5r9tAB-Mouse12538
Mapk14 (p38a)MAPKCMGC6y7yAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12076
Mapk14 (p38a)MAPKCMGC6y7xAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12072
Mapk14 (p38a)MAPKCMGC5r91AB-Mouse12539
Mapk14 (p38a)MAPKCMGC5r9bAB-Mouse12540
Mapk14 (p38a)MAPKCMGC6y4xAB5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12032
Mapk14 (p38a)MAPKCMGC5r9uAA[4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanoneMouse12541
Mapk14 (p38a)MAPKCMGC5r9wAB~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamideMouse12542
Mapk14 (p38a)MAPKCMGC5r9xAB-Mouse12543
Mapk14 (p38a)MAPKCMGC5r8zAB6-methoxypyridine-3-carbothioamideMouse12544
Mapk14 (p38a)MAPKCMGC5r93AB-Mouse12545
Mapk14 (p38a)MAPKCMGC5r9uAB[4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanoneMouse12546
Mapk14 (p38a)MAPKCMGC5r9gAA-Mouse12547
Mapk14 (p38a)MAPKCMGC6soiAA-Mouse11676
Mapk14 (p38a)MAPKCMGC6y7zAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12082
Mapk14 (p38a)MAPKCMGC2ozaB-Mouse5862
Mapk14 (p38a)MAPKCMGC6so2AB-Mouse11679
Mapk14 (p38a)MAPKCMGC6so1AB-Mouse11675
Mapk14 (p38a)MAPKCMGC6y4uAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12038
Mapk14 (p38a)MAPKCMGC5r9dAAbenzyl hydroxycarbamateMouse12550
Mapk14 (p38a)MAPKCMGC6sovAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11685
Mapk14 (p38a)MAPKCMGC3p7bA1-{5-tert-butyl-3-[(5-oxo-1,4-diazepan-1-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylureaMouse5856
Mapk14 (p38a)MAPKCMGC5r8vAA-Mouse12553
Mapk14 (p38a)MAPKCMGC5r9dABbenzyl hydroxycarbamateMouse12554
Mapk14 (p38a)MAPKCMGC5r8uAA3,4-dihydro-2~{h}-chromene-6-carboxamideMouse12555
Mapk14 (p38a)MAPKCMGC5r8vAB-Mouse12556
Mapk14 (p38a)MAPKCMGC6y4tAA5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12030
Mapk14 (p38a)MAPKCMGC8yp8A-Mouse16229
Mapk14 (p38a)MAPKCMGC2ewaAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse5859
Mapk14 (p38a)MAPKCMGC5r9qAA1-phenylmethoxyureaMouse12557
Mapk14 (p38a)MAPKCMGC6y80AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12081
Mapk14 (p38a)MAPKCMGC6zwrAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12708
Mapk14 (p38a)MAPKCMGC6y7yAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12063
Mapk14 (p38a)MAPKCMGC8vt6A(4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamideMouse16230
Mapk14 (p38a)MAPKCMGC1lezA-Mouse5863
Mapk14 (p38a)MAPKCMGC5nzzFAphosphothiophosphoric acid-adenylate esterMouse9983
Mapk14 (p38a)MAPKCMGC8vwmA(4p)-4-{6-[(azetidin-1-yl)methyl]-5-(2-chloro-6-fluoroanilino)-1h-indazol-1-yl}-n-methylthiophene-2-carboxamideMouse16231
Mapk14 (p38a)MAPKCMGC6sp9AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11684
Mapk14 (p38a)MAPKCMGC5ra5AA-Mouse12558
Mapk14 (p38a)MAPKCMGC5r96AB-Mouse12559
Mapk14 (p38a)MAPKCMGC5r91AA-Mouse12560
Mapk14 (p38a)MAPKCMGC5r9sAB-Mouse12561
Mapk14 (p38a)MAPKCMGC5r9lAA(3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-olMouse12562
Mapk14 (p38a)MAPKCMGC3p78A1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-2-ylureaMouse5866
Mapk14 (p38a)MAPKCMGC5larAB5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse6752
Mapk14 (p38a)MAPKCMGC5r98AA-Mouse12563
Mapk14 (p38a)MAPKCMGC5r9eAB-Mouse12564
Mapk14 (p38a)MAPKCMGC5r9aAA-Mouse12565
Mapk14 (p38a)MAPKCMGC6zwrAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12709
Mapk14 (p38a)MAPKCMGC5r9xAA-Mouse12566
Mapk14 (p38a)MAPKCMGC6y8hAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12078
Mapk14 (p38a)MAPKCMGC5ra7AA4-methylbenzamideMouse12567
Mapk14 (p38a)MAPKCMGC2ghmA3-(2-chlorobenzyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)ureaMouse5845
Mapk14 (p38a)MAPKCMGC5ra2AA1-(3-methylpyridin-2-yl)-1,4-diazepaneMouse12568
Mapk14 (p38a)MAPKCMGC6y82AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12061
Mapk14 (p38a)MAPKCMGC5r9fAB-Mouse12569
Mapk14 (p38a)MAPKCMGC5r9mAB-Mouse12570
Mapk14 (p38a)MAPKCMGC6y85AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12068
Mapk14 (p38a)MAPKCMGC5r93AA-Mouse12571
Mapk14 (p38a)MAPKCMGC6sotAB-Mouse11688
Mapk14 (p38a)MAPKCMGC5r99AA3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12572
Mapk14 (p38a)MAPKCMGC5r8xAA-Mouse12573
Mapk14 (p38a)MAPKCMGC4loqDB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5843
Mapk14 (p38a)MAPKCMGC5r9mAA-Mouse12574
Mapk14 (p38a)MAPKCMGC4lopDB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5837
Mapk14 (p38a)MAPKCMGC5r8yAAthiophene-2-carbothioamideMouse12584
Mapk14 (p38a)MAPKCMGC3tg1A-Mouse5850
Mapk14 (p38a)MAPKCMGC4lopAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5848
Mapk14 (p38a)MAPKCMGC5ra8AA5-(trifluoromethyl)-1,2-benzoxazol-3-amineMouse12585
Mapk14 (p38a)MAPKCMGC5r95AA-Mouse12586
Mapk14 (p38a)MAPKCMGC5r9hAB-Mouse12587
Mapk14 (p38a)MAPKCMGC6y4wAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12033
Mapk14 (p38a)MAPKCMGC6y85AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12069
Mapk14 (p38a)MAPKCMGC5r9oAA-Mouse12588
Mapk14 (p38a)MAPKCMGC6y82AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12077
Mapk14 (p38a)MAPKCMGC6y4uAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12035
Mapk14 (p38a)MAPKCMGC6yjcAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12438
Mapk14 (p38a)MAPKCMGC6ycuAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12154
Mapk14 (p38a)MAPKCMGC5r9gAB-Mouse12595
Mapk14 (p38a)MAPKCMGC7bdqA~{n}-[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]-4-[[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]benzamideMouse13408
Mapk14 (p38a)MAPKCMGC5r9nAB[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12596
Mapk14 (p38a)MAPKCMGC5r95AB-Mouse12597
Mapk14 (p38a)MAPKCMGC6y6vAB5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12067
Mapk14 (p38a)MAPKCMGC5ra6AB1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thioureaMouse12598
Mapk14 (p38a)MAPKCMGC6so1AA-Mouse11681
Mapk14 (p38a)MAPKCMGC5ra1AA2-phenoxyacetamideMouse12600
Mapk14 (p38a)MAPKCMGC6so2AA-Mouse11678
Mapk14 (p38a)MAPKCMGC5r9aAB-Mouse12604
Mapk14 (p38a)MAPKCMGC5ra9AB4-chloranylthieno[3,2-d]pyrimidineMouse12607
Mapk14 (p38a)MAPKCMGC5ra8AB5-(trifluoromethyl)-1,2-benzoxazol-3-amineMouse12608
Mapk14 (p38a)MAPKCMGC1ywrA4-(4-fluorophenyl)-1-methyl-5-(2-{[(1s)-1-phenylethyl]amino}pyrimidin-4-yl)-2-piperidin-4-yl-1,2-dihydro-3h-pyrazol-3-oneMouse5840
Mapk14 (p38a)MAPKCMGC5r9qAB1-phenylmethoxyureaMouse12612
Mapk14 (p38a)MAPKCMGC7bdoAA~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamideMouse13409
Mapk14 (p38a)MAPKCMGC6so4AB-Mouse11626
Mapk14 (p38a)MAPKCMGC4lopDA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5865
Mapk14 (p38a)MAPKCMGC5r9zAB-Mouse12613
Mapk14 (p38a)MAPKCMGC5ra6AA1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thioureaMouse12614
Mapk14 (p38a)MAPKCMGC8ypfA-Mouse16232
Mapk14 (p38a)MAPKCMGC5r9hAA-Mouse12615
Mapk14 (p38a)MAPKCMGC5r9oAB-Mouse12616
Mapk14 (p38a)MAPKCMGC5ra0AB[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12617
Mapk14 (p38a)MAPKCMGC5r9tAA-Mouse12618
Mapk14 (p38a)MAPKCMGC6y4vAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12037
Mapk14 (p38a)MAPKCMGC5r9yAB3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12621