| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | A | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | 5212 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bl7 | A | | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Human | 5193 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9p | A | B | 4-amino-n-(pyridin-2-yl)benzenesulfonamide | Mouse | 12576 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12071 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | A | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12066 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9b | A | A | - | Mouse | 12577 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | B | 4-methylbenzamide | Mouse | 12578 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12164 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9z | A | A | - | Mouse | 12580 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12163 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p79 | A | | 1-{3-tert-butyl-1-[2-(1,1-dioxidothiomorpholin-4-yl)-2-oxoethyl]-1h-pyrazol-5-yl}-3-naphthalen-2-ylurea | Mouse | 5849 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | B | - | Mouse | 12581 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12036 | |
| Mapk14 (p38a) | MAPK | CMGC | 4tyh | B | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Mouse | 5844 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r94 | A | B | - | Mouse | 12589 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r92 | A | A | (3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamide | Mouse | 12590 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12075 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra0 | A | A | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12592 | |
| Mapk14 (p38a) | MAPK | CMGC | 6soi | A | B | - | Mouse | 11682 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9n | A | A | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12593 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | B | - | Mouse | 12594 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9e | A | A | - | Mouse | 12602 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r90 | A | A | 2,5-diphenyl-4~{h}-pyrazol-3-one | Mouse | 12603 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9w | A | A | ~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamide | Mouse | 12605 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9j | A | A | 3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dione | Mouse | 12609 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r96 | A | A | - | Mouse | 12610 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9k | A | A | 2,3-dihydro-1-benzoxepine-5-carboxylic acid | Mouse | 12611 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5835 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | B | - | Mouse | 12619 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sov | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11677 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12153 | |
| Mapk14 (p38a) | MAPK | CMGC | 6spl | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11687 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r92 | A | B | (3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamide | Mouse | 12620 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8z | A | A | 6-methoxypyridine-3-carbothioamide | Mouse | 12575 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra1 | A | B | 2-phenoxyacetamide | Mouse | 12579 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9c | A | A | - | Mouse | 12591 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | A | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | 12601 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8x | A | B | - | Mouse | 12521 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9j | A | B | 3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dione | Mouse | 12527 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r98 | A | B | - | Mouse | 12606 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12060 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | E | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9981 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5872 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7c | A | | 1-[5-tert-butyl-3-({4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepan-1-yl}carbonyl)thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | Mouse | 5838 | |
| Mapk14 (p38a) | MAPK | CMGC | 2gtm | A | | 8-(2-chlorophenylamino)-2-(2,6-difluorophenylamino)-9-ethyl-9h-purine-1,7-diium | Mouse | 5867 | |
| Mapk14 (p38a) | MAPK | CMGC | 8vmh | A | | (4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamide | Mouse | 16233 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12080 | |
| Mapk14 (p38a) | MAPK | CMGC | 6spl | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11683 | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5112 | |
| Mapk14 (p38a) | MAPK | CMGC | 7z9t | A | | n-(2-cyclobutyl-1h-1,3-benzodiazol-5-yl)benzenesulfonamide | Mouse | 14799 | |
| Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | A | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | 14801 | |
| Mapk14 (p38a) | MAPK | CMGC | 8vmm | A | | (4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Mouse | 16228 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | B | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | 12520 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5839 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | B | - | Human | 11249 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5855 | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | B | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | 6707 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sod | A | A | - | Mouse | 11673 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12065 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loo | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5832 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8y | A | B | thiophene-2-carbothioamide | Mouse | 12524 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r97 | A | B | 4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amine | Mouse | 12525 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12034 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sou | A | B | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | 11672 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5831 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8u | A | B | 3,4-dihydro-2~{h}-chromene-6-carboxamide | Mouse | 12583 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | A | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5196 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 4 | - | Human | 5067 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv7 | A | | 1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylurea | Human | 5223 | |
| MAPK14 (p38a) | MAPK | CMGC | 2baj | A | | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2,3-dichlorophenyl)urea | Human | 5176 | |
| MAPK14 (p38a) | MAPK | CMGC | 3obj | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 4994 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | A | tak-715 | Human | 5033 | |
| Mapk14 (p38a) | MAPK | CMGC | 8efj | A | | (4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamide | Mouse | 14995 | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | A | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | 5062 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aac | A | | n-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamide | Human | 5048 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | B | - | Human | 4996 | |
| MAPK14 (p38a) | MAPK | CMGC | 3c5u | A | | 6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amine | Human | 5125 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oc1 | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5019 | |
| MAPK14 (p38a) | MAPK | CMGC | 3obg | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5211 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | B | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8681 | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | A | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | 9514 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5858 | |
| Mapk14 (p38a) | MAPK | CMGC | 3py3 | A | | - | Mouse | 5857 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fso | X | | - | Human | 5117 | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | A | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | 5006 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9i | A | A | methyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoate | Mouse | 12548 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12079 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9k | A | B | 2,3-dihydro-1-benzoxepine-5-carboxylic acid | Mouse | 12549 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11686 | |
| Mapk14 (p38a) | MAPK | CMGC | 4tyh | B | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Mouse | 5841 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 5870 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ghl | A | | 3-(2-chlorophenyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | 5871 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh2 | A | | - | Human | 4985 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | A | - | Mouse | 12552 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | A | - | Mouse | 11627 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9i | A | B | methyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoate | Mouse | 12551 | |
| Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | A | - | Mouse | 14747 | |
| Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | B | - | Mouse | 14748 | |
| Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | B | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | 14800 | |
| Mapk14 (p38a) | MAPK | CMGC | 8aco | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 15094 | |
| Mapk14 (p38a) | MAPK | CMGC | 8aco | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 15095 | |
| Mapk14 (p38a) | MAPK | CMGC | 8acm | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 15096 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fko | A | | 3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazole | Human | 5075 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | A | - | Human | 5163 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | B | - | Human | 5222 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | B | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11958 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | B | 2-amino-phenylamino-dibenzosuberone | Human | 5089 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | A | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | 5200 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | B | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5013 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | B | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 4983 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | B | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | 5031 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | A | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | 5081 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | B | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | 5214 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omh | A | | 1-(3-chlorophenyl)-3-methyl-4~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11251 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | A | - | Human | 4997 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mw1 | A | | 8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxide | Human | 5072 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zzl | A | | 6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-isopropyl[1,2,4]triazolo[4,3-a]pyridine | Human | 5249 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gfe | A | | n-cyclopropyl-3-{[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-4-yl]amino}-4-methylbenzamide | Human | 4991 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bmk | A | | 4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazole | Human | 5235 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fly | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5113 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | B | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5120 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfe | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5173 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | A | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11956 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | A | [3-(benzyloxy)phenyl]methanol | Human | 4978 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 8 | - | Human | 5078 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfa | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 5018 | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | B | | - | Human | 5007 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | B | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | 5132 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh1 | A | | - | Human | 5003 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | B | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | 5246 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyy | A | | 3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-4h-1,2,4-triazol-3-yl)phenol | Human | 9513 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | A | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | 5247 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nww | A | | 1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylurea | Human | 5068 | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | B | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | 9516 | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | A | | - | Human | 5136 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kf7 | A | | 3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamide | Human | 5201 | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | B | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | 5111 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | B | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 5256 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 12698 | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | A | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | 5230 | |
| MAPK14 (p38a) | MAPK | CMGC | 2baq | A | | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5184 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | B | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | 5155 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mgy | A | | - | Human | 5171 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | 4998 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | B | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | 5046 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 4977 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | A | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5012 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | A | | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 4993 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | A | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5237 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zqs | A | | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | 12986 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmm | A | | 6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5186 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | D | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5144 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | 11617 | |
| MAPK14 (p38a) | MAPK | CMGC | 3odz | X | | - | Human | 5069 | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | A | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | 5150 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fc1 | X | | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5110 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e92 | A | | n-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamide | Human | 5149 | |
| MAPK14 (p38a) | MAPK | CMGC | 8yd9 | A | B | - | Human | 15696 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | B | | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5064 | |
| MAPK14 (p38a) | MAPK | CMGC | 9r27 | A | | 4-[4-[[4-chloranyl-3-(trifluoromethyl)phenyl]carbamoylamino]-3-fluoranyl-phenoxy]-~{n}-methyl-pyridine-2-carboxamide | Human | 15697 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbn | A | | n-(3-tert-butyl-1h-pyrazol-5-yl)-n'-{4-chloro-3-[(pyridin-3-yloxy)methyl]phenyl}urea | Human | 5257 | |
| MAPK14 (p38a) | MAPK | CMGC | 3roc | A | | 3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamide | Human | 5011 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5194 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv6 | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(2-morpholin-4-ylethoxy)phenyl]urea | Human | 5101 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yiw | A | | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | 4988 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6c | A | | - | Human | 5015 | |
| MAPK14 (p38a) | MAPK | CMGC | 1di9 | A | | 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline | Human | 5251 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | B | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5053 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 5 | - | Human | 5107 | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8x | A | | n,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 5041 | |
| MAPK14 (p38a) | MAPK | CMGC | 8a8m | A | | phosphomethylphosphonic acid adenosyl ester | Human | 14289 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etc | A | | - | Human | 6361 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wfc | A | | - | Human | 4989 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | B | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | 5004 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5175 | |
| MAPK14 (p38a) | MAPK | CMGC | 1yqj | A | | 6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazine | Human | 5152 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj5 | A | | pexmetinib | Human | 15698 | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8u | A | | - | Human | 8381 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e8a | A | | - | Human | 4979 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpa | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5026 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12487 | |
| MAPK14 (p38a) | MAPK | CMGC | 2npq | A | | - | Human | 5205 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | B | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | 9517 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5032 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hvc | A | | 4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridine | Human | 5054 | |
| MAPK14 (p38a) | MAPK | CMGC | 4a9y | A | | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | 5073 | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | B | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | 5036 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbw | A | | 3-(1-naphthylmethoxy)pyridin-2-amine | Human | 5179 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | A | (3-phenoxyphenyl)methanol | Human | 5208 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ody | X | | - | Human | 5233 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbo | A | | 2-chlorophenol | Human | 5039 | |
| MAPK14 (p38a) | MAPK | CMGC | 8yd9 | A | A | - | Human | 15699 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d83 | A | | n-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamide | Human | 5028 | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | A | tak-715 | Human | 9515 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | A | | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5060 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 3 | - | Human | 5040 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | A | - | Human | 5189 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw5 | A | | n-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamide | Human | 5076 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | C | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5142 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsk | A | | 3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 5008 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | C | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5199 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 12699 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lhj | A | | n-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamide | Human | 5234 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | B | | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | 5180 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fl4 | A | | 6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidine | Human | 5151 | |
| MAPK14 (p38a) | MAPK | CMGC | 3s4q | A | | 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamide | Human | 5133 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | B | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | 5034 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfc | A | | (4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5160 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | A | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | 5038 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | B | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5017 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ocg | A | | 5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamide | Human | 4984 | |
| MAPK14 (p38a) | MAPK | CMGC | 2bal | A | | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanone | Human | 5260 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | B | | - | Human | 7137 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | B | - | Human | 5195 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | B | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5232 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | A | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | 5213 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fln | C | | 6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5090 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5137 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gi3 | A | | n-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamide | Human | 5226 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | B | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | 11619 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12489 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | A | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | 5217 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | A | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | 8382 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnx | A | | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5002 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | B | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5188 | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | A | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | 5005 | |
| MAPK14 (p38a) | MAPK | CMGC | 2bak | A | | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | 5114 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsm | X | | - | Human | 5044 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj2 | A | A | - | Human | 15700 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | A | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5216 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5263 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouk | A | | 4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidine | Human | 5146 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hl7 | A | | 2-{4-[5-(4-chlorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-3-yl]piperidin-1-yl}-2-oxoethanol | Human | 5236 | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | B | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | 11819 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | A | | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | 5159 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | C | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5182 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 9 | - | Human | 5127 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | A | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | 5115 | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | B | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | 4992 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fml | A | | 6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5010 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmj | A | | 4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amine | Human | 5129 | |
| MAPK14 (p38a) | MAPK | CMGC | 6m9l | A | | 3-benzyl-6-[(2,4-difluorophenyl)amino]-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Human | 11255 | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | B | - | Human | 5030 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | B | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 4995 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp5 | A | | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5158 | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5218 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj4 | A | C | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15706 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | B | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5131 | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv2 | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 5255 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmh | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5024 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flw | A | | 6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5153 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | D | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5016 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | B | - | Human | 4981 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh0 | A | | - | Human | 5124 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 5035 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12152 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | A | - | Human | 8523 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | A | - | Human | 5170 | |
| Mapk14 (p38a) | MAPK | CMGC | 2gtn | A | | 2-(2,6-difluorophenoxy)-n-(2-fluorophenyl)-9-isopropyl-9h-purin-8-amine | Mouse | 5860 | |
| Mapk14 (p38a) | MAPK | CMGC | 7be5 | A | | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-methyl-pyrazole-4-carboxamide | Mouse | 13407 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9f | A | A | - | Mouse | 12526 | |
| Mapk14 (p38a) | MAPK | CMGC | 5lar | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 6753 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5861 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | H | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9984 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p5k | A | | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | 5854 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5846 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12151 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sod | A | B | - | Mouse | 11674 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12031 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r90 | A | B | 2,5-diphenyl-4~{h}-pyrazol-3-one | Mouse | 12582 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sou | A | A | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | 11680 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | F | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9979 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loo | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5851 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5833 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | A | - | Mouse | 12599 | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | A | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | 5198 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ctq | A | | n-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamide | Human | 5220 | |
| MAPK14 (p38a) | MAPK | CMGC | 5tco | A | | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-carboxamide | Human | 8031 | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | B | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5050 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5203 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | A | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | 5037 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | A | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5074 | |
| MAPK14 (p38a) | MAPK | CMGC | 4dli | A | | - | Human | 5092 | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | A | - | Human | 5079 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | B | - | Human | 5231 | |
| MAPK14 (p38a) | MAPK | CMGC | 5tbe | A | | ~{n}-[2,4-bis(fluoranyl)-5-[[9-(2-morpholin-4-ylethylcarbamoyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulen-3-yl]amino]phenyl]thiophene-2-carboxamide | Human | 8032 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3j | A | | 2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamide | Human | 5047 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | C | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11618 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | A | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11246 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hrb | A | | [3-amino-2-(2-methylphenyl)-1-oxidopyridin-4-yl](2,4-difluorophenyl)methanone | Human | 5202 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w84 | A | | 3-(2-pyridin-4-ylethyl)-1h-indole | Human | 5065 | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | A | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5227 | |
| MAPK14 (p38a) | MAPK | CMGC | 3u8w | A | | 3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamide | Human | 5192 | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | A | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | 5027 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | A | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5141 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbt | A | | 3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamide | Human | 5082 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | B | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | 5022 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | B | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5138 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | B | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | 8379 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | A | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | 11613 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | B | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 11621 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w83 | A | | n-[4-chloro-3-(pyridin-3-yloxymethyl)-phenyl]-3-fluoro- | Human | 4986 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mty | A | | ~{n}-[2,4-bis(fluoranyl)-5-[[14-(2-hydroxyethylcarbamoyl)-2-oxidanylidene-6-tricyclo[9.4.0.0^{3,8}]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]amino]phenyl]thiophene-2-carboxamide | Human | 8383 | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8v | A | | - | Human | 8380 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | 5001 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | A | - | Human | 7134 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsf | A | | 3-(2,6-dichlorophenyl)-7-({4-[(diethylamino)methoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 5097 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmk | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5209 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | A | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | 5183 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh9 | A | | - | Human | 4982 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bl6 | A | | 4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazole | Human | 5243 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12486 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | 11620 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | B | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | 5156 | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5122 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fls | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5119 | |
| MAPK14 (p38a) | MAPK | CMGC | 3que | A | | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | 5095 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | B | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | 11254 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | B | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | 5059 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | C | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5215 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh3 | A | | - | Human | 5109 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | B | tak-715 | Human | 5098 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11616 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qyx | A | | - | Human | 12127 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flz | A | | 8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5204 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hub | A | | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5029 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | A | - | Human | 11253 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 2 | - | Human | 5093 | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | A | - | Human | 5025 | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | B | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | 5262 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | A | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 5061 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh3 | A | | naringenin | Human | 5042 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | 6880 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | A | - | Human | 11247 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | A | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8680 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh2 | A | | 3-phenylquinazolin-4(3h)-one | Human | 5244 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsl | X | | - | Human | 5264 | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | A | | - | Human | 5177 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | B | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | 5187 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | B | | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5210 | |
| MAPK14 (p38a) | MAPK | CMGC | 3itz | A | | 4-chloro-n-cyclopropyl-3-{[1-(2,6-difluorophenyl)-1h-pyrazolo[3,4-d]pyridazin-4-yl]amino}benzamide | Human | 5135 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | B | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | 5057 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qe1 | A | | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{r})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11957 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | A | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | 5070 | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | B | - | Human | 5248 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | A | | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5121 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bx5 | A | | n-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamide | Human | 5000 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | A | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5139 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | A | - | Human | 5080 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12488 | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv1 | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5252 | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | B | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | 5009 | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5096 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa4 | A | | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamide | Human | 5045 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbs | A | | 3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamide | Human | 5258 | |
| MAPK14 (p38a) | MAPK | CMGC | 1m7q | A | | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-one | Human | 5128 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6a | A | | - | Human | 5238 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv3 | A | | 5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5207 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12490 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 5166 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | A | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5140 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eti | A | | - | Human | 6362 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12491 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w82 | A | | n-[(3z)-5-tert-butyl-2-phenyl-1,2-dihydro-3h-pyrazol-3-ylidene]-n'-(4-chlorophenyl)urea | Human | 5165 | |
| MAPK14 (p38a) | MAPK | CMGC | 4geo | A | | - | Human | 5190 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12492 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5077 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw7 | A | | 2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridine | Human | 5084 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | B | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | 5108 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | A | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 11615 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | A | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | 4980 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r39 | A | | - | Human | 5116 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | B | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11245 | |
| MAPK14 (p38a) | MAPK | CMGC | 1a9u | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5229 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flq | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5168 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | 6879 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8t | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5167 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8p | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5071 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yis | A | | 1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}urea | Human | 5240 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | B | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | 5154 | |
| MAPK14 (p38a) | MAPK | CMGC | 2qd9 | A | | 1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanone | Human | 5197 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | B | | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5091 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | A | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5178 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | A | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | 4999 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | A | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | 11248 | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8s | A | | 3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamide | Human | 5055 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | B | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5106 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12493 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fi4 | A | | (2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol | Human | 5051 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8u | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5250 | |
| MAPK14 (p38a) | MAPK | CMGC | 3s3i | A | | 3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamide | Human | 5169 | |
| MAPK14 (p38a) | MAPK | CMGC | 3dt1 | A | | n-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamide | Human | 5086 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfd | A | | 1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5102 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5174 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouy | A | | 1-(2,6-dichlorophenyl)-6-[(2,4-difluorophenyl)sulfanyl]-7-(1,2,3,6-tetrahydro-4-pyridinyl)-3,4-dihydropyrido[3,2-d]pyrimidin-2(1h)-one | Human | 7258 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | B | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | 5103 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | A | | - | Human | 7136 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yix | A | | 1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | 5143 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 4987 | |
| MAPK14 (p38a) | MAPK | CMGC | 8x3m | A | A | - | Human | 15701 | |
| MAPK14 (p38a) | MAPK | CMGC | 3rin | A | | n-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamide | Human | 5239 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbv | A | | 3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamide | Human | 5148 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | A | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5225 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | B | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | 5147 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | A | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | 5094 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | A | 2-amino-phenylamino-dibenzosuberone | Human | 5105 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | B | (3-phenoxyphenyl)methanol | Human | 5020 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | A | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | 4990 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w7h | A | | 3-(benzyloxy)pyridin-2-amine | Human | 5023 | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | D | | - | Human | 5100 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj2 | A | B | - | Human | 15702 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa5 | A | | n-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamide | Human | 5206 | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | B | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | 5145 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | B | - | Human | 11250 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n66 | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 8524 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 1 | - | Human | 5021 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5162 | |
| MAPK14 (p38a) | MAPK | CMGC | 6m95 | A | | (4-benzylpiperidin-1-yl)[2-methoxy-4-(methylsulfanyl)phenyl]methanone | Human | 11252 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | B | [3-(benzyloxy)phenyl]methanol | Human | 5014 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 10 | - | Human | 5063 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | A | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | 5099 | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | B | tak-715 | Human | 9518 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | D | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5123 | |
| MAPK14 (p38a) | MAPK | CMGC | 5ml5 | A | | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{h}-imidazol-5-yl]pyridin-2-yl]propanamide | Human | 7544 | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg6 | A | | 4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5228 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj4 | A | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15703 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | A | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | 5253 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 6 | - | Human | 5219 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | A | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | 5241 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj4 | A | B | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15704 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5052 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh6 | A | | n-phenylpyridine-3-carboxamide | Human | 5083 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv2 | A | | 5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5191 | |
| MAPK14 (p38a) | MAPK | CMGC | 8x3m | A | B | - | Human | 15705 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | B | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | 5104 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | A | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | 5224 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5b | A | | - | Human | 5221 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 7 | - | Human | 5161 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | A | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | 9519 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | A | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5130 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zz2 | A | | n-[3-(4-fluorophenoxy)phenyl]-4-[(2-hydroxybenzyl)amino]piperidine-1-sulfonamide | Human | 5164 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5126 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw8 | A | | 1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)urea | Human | 5181 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | B | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | 5245 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh4 | A | | phenyl(piperidin-1-yl)methanone | Human | 5043 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | B | - | Human | 7135 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkl | A | | n-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamide | Human | 5172 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh5 | A | | benzyl pyridine-3-carboxylate | Human | 5185 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | B | - | Human | 8521 | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | A | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | 6706 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zyj | A | | 4-phenoxy-n-(pyridin-2-ylmethyl)benzamide | Human | 5058 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkn | A | | 3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidine | Human | 5049 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11614 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | B | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5087 | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg5 | A | | n-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5254 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n65 | A | | 2-phenyl-~{n}4-(2-thiophen-2-ylethyl)quinazoline-4,7-diamine | Human | 8525 | |
| MAPK14 (p38a) | MAPK | CMGC | 4dlj | A | | 2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamine | Human | 5242 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n63 | A | | - | Human | 8526 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5157 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5085 | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | B | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | 5261 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | B | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5118 | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | A | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | 11818 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5088 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n64 | A | | - | Human | 8527 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | A | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5066 | |
| MAPK14 (p38a) | MAPK | CMGC | 3od6 | X | | - | Human | 5134 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n68 | A | | - | Human | 8522 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | A | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5056 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7a | A | | 1-[5-tert-butyl-2-(1,1-dioxidothiomorpholin-4-yl)thiophen-3-yl]-3-naphthalen-1-ylurea | Mouse | 5853 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9p | A | A | 4-amino-n-(pyridin-2-yl)benzenesulfonamide | Mouse | 12518 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | H | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9978 | |
| Mapk14 (p38a) | MAPK | CMGC | 5o90 | A | | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 9525 | |
| Mapk14 (p38a) | MAPK | CMGC | 4ka3 | A | | - | Mouse | 5852 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | G | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9982 | |
| Mapk14 (p38a) | MAPK | CMGC | 5uoj | A | | - | Mouse | 7466 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9r | A | A | 4-acetyl-n-ethylpiperazine-1-carboxamide | Mouse | 12519 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9c | A | B | - | Mouse | 12522 | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | B | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | 13405 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9l | A | B | (3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-ol | Mouse | 12523 | |
| Mapk14 (p38a) | MAPK | CMGC | 7be4 | A | | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 13406 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9v | A | B | - | Mouse | 12528 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r97 | A | A | 4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amine | Mouse | 12529 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sot | A | A | - | Mouse | 11689 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9v | A | A | - | Mouse | 12530 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | E | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9980 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9s | A | A | - | Mouse | 12531 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r94 | A | A | - | Mouse | 12532 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5836 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5847 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r99 | A | B | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12533 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p4k | A | | - | Mouse | 5842 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12437 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8w | A | B | - | Mouse | 12534 | |
| Mapk14 (p38a) | MAPK | CMGC | 2puu | A | | 5-tert-butyl-2-(4-methylphenyl)-3-{[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]-1-naphthyl}amino)carbonyl]amino}-1h-pyrazol-2-ium | Mouse | 6866 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8w | A | A | - | Mouse | 12535 | |
| Mapk14 (p38a) | MAPK | CMGC | 1yw2 | A | | 2-(ethoxymethyl)-4-(4-fluorophenyl)-3-[2-(2-hydroxyphenoxy)pyrimidin-4-yl]isoxazol-5(2h)-one | Mouse | 5869 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12070 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | G | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9977 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12073 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9r | A | B | 4-acetyl-n-ethylpiperazine-1-carboxamide | Mouse | 12536 | |
| Mapk14 (p38a) | MAPK | CMGC | 1lew | A | | - | Mouse | 5864 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5834 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12039 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9y | A | A | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12537 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9t | A | B | - | Mouse | 12538 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12076 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12072 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r91 | A | B | - | Mouse | 12539 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9b | A | B | - | Mouse | 12540 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12032 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9u | A | A | [4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanone | Mouse | 12541 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9w | A | B | ~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamide | Mouse | 12542 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9x | A | B | - | Mouse | 12543 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8z | A | B | 6-methoxypyridine-3-carbothioamide | Mouse | 12544 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r93 | A | B | - | Mouse | 12545 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9u | A | B | [4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanone | Mouse | 12546 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9g | A | A | - | Mouse | 12547 | |
| Mapk14 (p38a) | MAPK | CMGC | 6soi | A | A | - | Mouse | 11676 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12082 | |
| Mapk14 (p38a) | MAPK | CMGC | 2oza | B | | - | Mouse | 5862 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | B | - | Mouse | 11679 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | B | - | Mouse | 11675 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12038 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9d | A | A | benzyl hydroxycarbamate | Mouse | 12550 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sov | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11685 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7b | A | | 1-{5-tert-butyl-3-[(5-oxo-1,4-diazepan-1-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | 5856 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8v | A | A | - | Mouse | 12553 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9d | A | B | benzyl hydroxycarbamate | Mouse | 12554 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8u | A | A | 3,4-dihydro-2~{h}-chromene-6-carboxamide | Mouse | 12555 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8v | A | B | - | Mouse | 12556 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12030 | |
| Mapk14 (p38a) | MAPK | CMGC | 8yp8 | A | | - | Mouse | 16229 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 5859 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9q | A | A | 1-phenylmethoxyurea | Mouse | 12557 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12081 | |
| Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12708 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12063 | |
| Mapk14 (p38a) | MAPK | CMGC | 8vt6 | A | | (4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamide | Mouse | 16230 | |
| Mapk14 (p38a) | MAPK | CMGC | 1lez | A | | - | Mouse | 5863 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | F | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9983 | |
| Mapk14 (p38a) | MAPK | CMGC | 8vwm | A | | (4p)-4-{6-[(azetidin-1-yl)methyl]-5-(2-chloro-6-fluoroanilino)-1h-indazol-1-yl}-n-methylthiophene-2-carboxamide | Mouse | 16231 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11684 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | A | - | Mouse | 12558 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r96 | A | B | - | Mouse | 12559 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r91 | A | A | - | Mouse | 12560 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9s | A | B | - | Mouse | 12561 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9l | A | A | (3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-ol | Mouse | 12562 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p78 | A | | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-2-ylurea | Mouse | 5866 | |
| Mapk14 (p38a) | MAPK | CMGC | 5lar | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 6752 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r98 | A | A | - | Mouse | 12563 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9e | A | B | - | Mouse | 12564 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9a | A | A | - | Mouse | 12565 | |
| Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12709 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9x | A | A | - | Mouse | 12566 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12078 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | A | 4-methylbenzamide | Mouse | 12567 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ghm | A | | 3-(2-chlorobenzyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | 5845 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | A | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | 12568 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12061 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9f | A | B | - | Mouse | 12569 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9m | A | B | - | Mouse | 12570 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12068 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r93 | A | A | - | Mouse | 12571 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sot | A | B | - | Mouse | 11688 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r99 | A | A | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12572 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8x | A | A | - | Mouse | 12573 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5843 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9m | A | A | - | Mouse | 12574 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5837 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8y | A | A | thiophene-2-carbothioamide | Mouse | 12584 | |
| Mapk14 (p38a) | MAPK | CMGC | 3tg1 | A | | - | Mouse | 5850 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5848 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | A | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | 12585 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r95 | A | A | - | Mouse | 12586 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9h | A | B | - | Mouse | 12587 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12033 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12069 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9o | A | A | - | Mouse | 12588 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12077 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12035 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12438 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12154 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9g | A | B | - | Mouse | 12595 | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdq | A | | ~{n}-[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]-4-[[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]benzamide | Mouse | 13408 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9n | A | B | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12596 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r95 | A | B | - | Mouse | 12597 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | B | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12067 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | B | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | 12598 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | A | - | Mouse | 11681 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra1 | A | A | 2-phenoxyacetamide | Mouse | 12600 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | A | - | Mouse | 11678 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9a | A | B | - | Mouse | 12604 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | B | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | 12607 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | B | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | 12608 | |
| Mapk14 (p38a) | MAPK | CMGC | 1ywr | A | | 4-(4-fluorophenyl)-1-methyl-5-(2-{[(1s)-1-phenylethyl]amino}pyrimidin-4-yl)-2-piperidin-4-yl-1,2-dihydro-3h-pyrazol-3-one | Mouse | 5840 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9q | A | B | 1-phenylmethoxyurea | Mouse | 12612 | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | A | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | 13409 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | B | - | Mouse | 11626 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5865 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9z | A | B | - | Mouse | 12613 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | A | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | 12614 | |
| Mapk14 (p38a) | MAPK | CMGC | 8ypf | A | | - | Mouse | 16232 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9h | A | A | - | Mouse | 12615 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9o | A | B | - | Mouse | 12616 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra0 | A | B | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12617 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9t | A | A | - | Mouse | 12618 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12037 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9y | A | B | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12621 | |