| PIK3CG (p110g) | PIK | Atypical | 7mez | A | | - | Human | 13798 | |
| PIK3CG (p110g) | PIK | Atypical | 3t8m | A | | n~2~-{2-chloro-4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-n~2~,n~8~-dimethyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2,8-dicarboxamide | Human | 9186 | |
| PIK3CG (p110g) | PIK | Atypical | 4anx | A | | 5-{3-[(4-{3-[4-(1-methylethyl)phenyl]pyrazin-2-yl}piperazin-1-yl)sulfonyl]phenyl}pyrimidin-2-amine | Human | 9252 | |
| PIK3CG (p110g) | PIK | Atypical | 3ml8 | A | | 8-cyclopentyl-6-[3-(hydroxymethyl)phenyl]-4-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9192 | |
| PIK3CG (p110g) | PIK | Atypical | 3ps6 | A | | 4-amino-n-(6-methoxypyridin-3-yl)-2-methylquinazoline-8-carboxamide | Human | 9170 | |
| PIK3CG (p110g) | PIK | Atypical | 2chw | A | | 2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-one | Human | 9182 | |
| PIK3CG (p110g) | PIK | Atypical | 4aof | A | | n-[6-(5-methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]ethanamide | Human | 9245 | |
| PIK3CG (p110g) | PIK | Atypical | 5kae | A | | 4-azanyl-6-[[(1~{s})-1-(6-fluoranyl-3-phenyl-4-piperazin-1-ylcarbonyl-quinolin-2-yl)ethyl]amino]pyrimidine-5-carbonitrile | Human | 9241 | |
| PIK3CG (p110g) | PIK | Atypical | 5g2n | A | | 2-azanyl-~{n}-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]pyrimidine-5-carboxamide | Human | 9206 | |
| PIK3CG (p110g) | PIK | Atypical | 4kzc | A | | n-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamide | Human | 9224 | |
| PIK3CG (p110g) | PIK | Atypical | 4fhj | A | | 3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-5-yl)imidazo[1,2-a]pyridin-2-amine | Human | 9209 | |
| PIK3CG (p110g) | PIK | Atypical | 5g55 | A | | 6-cyano-4-[[(1r)-1-(4-methylphenyl)ethyl]amino]quinoline-3-carboxamide | Human | 9199 | |
| PIK3CG (p110g) | PIK | Atypical | 4ezk | A | | 2-(1-{[2-(2h-indazol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | 9176 | |
| PIK3CG (p110g) | PIK | Atypical | 4urk | A | | 2-[[(1r)-1-(7-methyl-2-morpholin-4-yl-4-oxidanylidene-pyrido[1,2-a]pyrimidin-9-yl)ethyl]amino]benzoic acid | Human | 9196 | |
| PIK3CG (p110g) | PIK | Atypical | 3qk0 | A | | n-[6-(6-chloro-5-{[(4-fluorophenyl)sulfonyl]amino}pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | 9213 | |
| PIK3CG (p110g) | PIK | Atypical | 4wwo | A | | n-{(1s)-1-[8-chloro-2-(3-fluorophenyl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | 9190 | |
| PIK3CG (p110g) | PIK | Atypical | 4kz0 | A | | methyl 2-(acetylamino)-1,3-benzothiazole-6-carboxylate | Human | 9161 | |
| PIK3CG (p110g) | PIK | Atypical | 4fjz | A | | 1'-[7-fluoro-3-methyl-2-(pyridin-2-yl)quinolin-4-yl]-6'-(morpholin-4-yl)-1',2,2',3,5,6-hexahydrospiro[pyran-4,3'-pyrrolo[3,2-b]pyridine] | Human | 9173 | |
| PIK3CG (p110g) | PIK | Atypical | 6xrl | A | | 2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 12774 | |
| PIK3CG (p110g) | PIK | Atypical | 4fhk | A | | 3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]-n-(1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-2-amine | Human | 9204 | |
| PIK3CG (p110g) | PIK | Atypical | 6c1s | A | | {4-[2-(5,6-dimethoxypyridin-3-yl)-5-oxo-5,7-dihydro-6h-pyrrolo[3,4-b]pyridin-6-yl]-1h-pyrazol-1-yl}acetonitrile | Human | 10037 | |
| PIK3CG (p110g) | PIK | Atypical | 3l13 | A | | [3-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenyl]methanol | Human | 9167 | |
| PIK3CG (p110g) | PIK | Atypical | 5jhb | A | | [1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanol | Human | 9238 | |
| PIK3CG (p110g) | PIK | Atypical | 3p2b | A | B | 3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenol | Human | 9165 | |
| PIK3CG (p110g) | PIK | Atypical | 4anw | A | A | 3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamide | Human | 9174 | |
| PIK3CG (p110g) | PIK | Atypical | 7kke | A | | n-[2-(3,3-dimethylbutoxy)ethyl]-n'-{4-methyl-5-[(pyridin-4-yl)ethynyl]-1,3-thiazol-2-yl}urea | Human | 13433 | |
| PIK3CG (p110g) | PIK | Atypical | 3p2b | A | A | 3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenol | Human | 9169 | |
| PIK3CG (p110g) | PIK | Atypical | 3ml9 | A | | 2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9187 | |
| PIK3CG (p110g) | PIK | Atypical | 3l08 | A | B | 2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide | Human | 9164 | |
| PIK3CG (p110g) | PIK | Atypical | 6aud | A | B | 10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine | Human | 9216 | |
| PIK3CG (p110g) | PIK | Atypical | 4ezj | A | | 2-(1-{[2-(5-fluoro-1h-indol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | 9222 | |
| PIK3CG (p110g) | PIK | Atypical | 3zvv | A | | 5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amine | Human | 9172 | |
| PIK3CG (p110g) | PIK | Atypical | 4dk5 | A | | 4-(2-[(6-methoxypyridin-3-yl)amino]-5-{[4-(methylsulfonyl)piperazin-1-yl]methyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amine | Human | 9232 | |
| PIK3CG (p110g) | PIK | Atypical | 1e8y | A | | - | Human | 9248 | |
| PIK3CG (p110g) | PIK | Atypical | 6fh5 | A | | 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one | Human | 10883 | |
| PIK3CG (p110g) | PIK | Atypical | 4fa6 | A | | 2-amino-8-cyclopentyl-4-methyl-6-(1h-pyrazol-4-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9191 | |
| PIK3CG (p110g) | PIK | Atypical | 1e8z | A | | staurosporine | Human | 9228 | |
| PIK3CG (p110g) | PIK | Atypical | 3ene | A | | 1-methyl-3-naphthalen-2-yl-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9188 | |
| PIK3CG (p110g) | PIK | Atypical | 2chz | A | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9251 | |
| PIK3CG (p110g) | PIK | Atypical | 4fad | A | | 2-amino-6-(5-fluoro-6-methoxypyridin-3-yl)-4-methyl-8-(pyrrolidin-1-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9202 | |
| PIK3CG (p110g) | PIK | Atypical | 3lj3 | A | | (2z)-4,6-dihydroxy-2-{[1-methyl-4-(4-methylpiperazin-1-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methylidene}-1-benzofuran-3(2h)-one | Human | 9214 | |
| PIK3CG (p110g) | PIK | Atypical | 2chx | A | | n-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamide | Human | 9247 | |
| PIK3CG (p110g) | PIK | Atypical | 3csf | A | | - | Human | 9215 | |
| PIK3CG (p110g) | PIK | Atypical | 4f1s | A | | n-(5-{[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(tetrahydro-2h-pyran-4-yl)pyridin-2-yl]amino}-2-chloropyridin-3-yl)methanesulfonamide | Human | 9221 | |
| PIK3CG (p110g) | PIK | Atypical | 3l17 | A | | 4-methyl-5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyrimidin-2-amine | Human | 9185 | |
| PIK3CG (p110g) | PIK | Atypical | 5eds | A | | 4-azanyl-6-[[(1~{s})-1-[6-fluoranyl-1-(3-methylsulfonylphenyl)benzimidazol-2-yl]ethyl]amino]pyrimidine-5-carbonitrile | Human | 9208 | |
| PIK3CG (p110g) | PIK | Atypical | 3l08 | A | A | 2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide | Human | 9217 | |
| PIK3CG (p110g) | PIK | Atypical | 4hvb | A | | 1-{1-[(2s)-2-hydroxypropanoyl]piperidin-4-yl}-3-methyl-8-(6-methylpyridin-3-yl)-1,3-dihydro-2h-imidazo[4,5-c][1,5]naphthyridin-2-one | Human | 9225 | |
| PIK3CG (p110g) | PIK | Atypical | 3dbs | A | | 2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidine | Human | 9230 | |
| PIK3CG (p110g) | PIK | Atypical | 6t3b | A | | 2-[(4-methoxy-2-methyl-phenyl)amino]-7-methyl-9-(4-oxidanylcyclohexyl)purin-8-one | Human | 11906 | |
| PIK3CG (p110g) | PIK | Atypical | 3apd | A | | 5-(2-morpholin-4-yl-7-pyridin-3-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamine | Human | 9205 | |
| PIK3CG (p110g) | PIK | Atypical | 4j6i | A | | 2-methyl-1-(4-{2-[1-(2,2,2-trifluoroethyl)-1h-1,2,4-triazol-5-yl]-4,5-dihydro[1]benzoxepino[5,4-d][1,3]thiazol-8-yl}-1h-pyrazol-1-yl)propan-2-ol | Human | 9189 | |
| PIK3CG (p110g) | PIK | Atypical | 3apc | A | | 5-(7-methanesulfonyl-2-morpholin-4-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamine | Human | 9231 | |
| PIK3CG (p110g) | PIK | Atypical | 3tjp | A | | n~6~-(3,4-dimethoxyphenyl)-2-(morpholin-4-yl)-4,5'-bipyrimidine-2',6-diamine | Human | 9234 | |
| PIK3CG (p110g) | PIK | Atypical | 7jwz | A | | 2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 13410 | |
| PIK3CG (p110g) | PIK | Atypical | 7jwe | A | | gedatolisib | Human | 13412 | |
| PIK3CG (p110g) | PIK | Atypical | 3nzu | A | | 6-(2h-indazol-4-yl)-1-methyl-n-[3-(methylsulfonyl)propyl]-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9177 | |
| PIK3CG (p110g) | PIK | Atypical | 6aud | A | A | 10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine | Human | 9239 | |
| PIK3CG (p110g) | PIK | Atypical | 3tl5 | A | | (2s)-1-(4-{[2-(2-aminopyrimidin-5-yl)-7-methyl-4-(morpholin-4-yl)thieno[3,2-d]pyrimidin-6-yl]methyl}piperazin-1-yl)-2-hydroxypropan-1-one | Human | 9160 | |
| PIK3CG (p110g) | PIK | Atypical | 3prz | A | | 4-amino-2-methyl-n-(1h-pyrazol-3-yl)quinazoline-8-carboxamide | Human | 9210 | |
| PIK3CG (p110g) | PIK | Atypical | 3ibe | A | | 1-(4-{4-morpholin-4-yl-1-[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-6-yl}phenyl)-3-pyridin-4-ylurea | Human | 9171 | |
| PIK3CG (p110g) | PIK | Atypical | 4wwp | A | | n-{(1s)-1-[8-chloro-2-(2-methylpyridin-3-yl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | 9200 | |
| PIK3CG (p110g) | PIK | Atypical | 2a5u | A | | (5e)-5-(quinoxalin-6-ylmethylene)-1,3-thiazolidine-2,4-dione | Human | 9183 | |
| PIK3CG (p110g) | PIK | Atypical | 3oaw | A | | 2-amino-4-methyl-8-(1-methylethyl)-6-(1h-pyrazol-4-yl)pteridin-7(8h)-one | Human | 9240 | |
| PIK3CG (p110g) | PIK | Atypical | 3dpd | A | | 5,5-dimethyl-2-morpholin-4-yl-5,6-dihydro-1,3-benzothiazol-7(4h)-one | Human | 9159 | |
| PIK3CG (p110g) | PIK | Atypical | 4fjy | A | | 4-[3,3-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1h-indol-1-yl]-7-fluoro-3-methyl-2-(pyridin-3-yl)quinoline | Human | 9249 | |
| PIK3CG (p110g) | PIK | Atypical | 5t23 | A | | 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{s})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine | Human | 9157 | |
| PIK3CG (p110g) | PIK | Atypical | 4ps3 | A | | 1-[6-(5-methoxypyridin-3-yl)-1,3-benzothiazol-2-yl]-3-[2-(1-propyl-1h-imidazol-4-yl)ethyl]urea | Human | 9193 | |
| PIK3CG (p110g) | PIK | Atypical | 3apf | A | | 3-[7-(1h-benzimidazol-5-yl)-2-(morpholin-4-yl)-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl]phenol | Human | 9250 | |
| PIK3CG (p110g) | PIK | Atypical | 6t3c | A | | 7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-one | Human | 11907 | |
| PIK3CG (p110g) | PIK | Atypical | 3zw3 | A | | n-{6-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]imidazo[1,2-a]pyridin-2-yl}acetamide | Human | 9207 | |
| PIK3CG (p110g) | PIK | Atypical | 3qjz | A | | n-{6-[2-(methylsulfanyl)pyrimidin-4-yl]-1,3-benzothiazol-2-yl}acetamide | Human | 9181 | |
| PIK3CG (p110g) | PIK | Atypical | 4gb9 | A | | 2-[1-({2-[2-(dimethylamino)-1h-benzimidazol-1-yl]-9-methyl-6-(morpholin-4-yl)-9h-purin-8-yl}methyl)piperidin-4-yl]propan-2-ol | Human | 9218 | |
| PIK3CG (p110g) | PIK | Atypical | 4xz4 | A | | n-[5-(6-methoxypyrazin-2-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide | Human | 9194 | |
| PIK3CG (p110g) | PIK | Atypical | 3sd5 | A | | 5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amine | Human | 9243 | |
| PIK3CG (p110g) | PIK | Atypical | 2v4l | A | | 3-[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]phenol | Human | 9237 | |
| PIK3CG (p110g) | PIK | Atypical | 3mjw | A | | (2z)-4,6-dihydroxy-2-[(8-methoxy-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)methylidene]-1-benzofuran-3(2h)-one | Human | 9229 | |
| PIK3CG (p110g) | PIK | Atypical | 4hle | A | | 2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepine-8-carboxamide | Human | 9219 | |
| PIK3CG (p110g) | PIK | Atypical | 3cst | A | | methylated ruthenium pyridocarbazole | Human | 9220 | |
| PIK3CG (p110g) | PIK | Atypical | 3nzs | A | | 6-(1,1-dioxidothiomorpholin-4-yl)-n-(3-methoxyphenyl)-1-methyl-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9179 | |
| PIK3CG (p110g) | PIK | Atypical | 4anu | A | | 3-amino-n-methyl-6-[3-(1h-tetrazol-5-yl)phenyl]pyrazine-2-carboxamide | Human | 9162 | |
| PIK3CG (p110g) | PIK | Atypical | 5jha | A | | [1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)pyrimidin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanol | Human | 9246 | |
| PIK3CG (p110g) | PIK | Atypical | 3pre | A | | 2-amino-8-(trans-4-methoxycyclohexyl)-4-methyl-6-(1h-pyrazol-3-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9198 | |
| PIK3CG (p110g) | PIK | Atypical | 7z61 | A | | 9-[(3~{r},4~{r})-4-fluoranylpyrrolidin-3-yl]-7-methyl-2-[(7-methylquinolin-6-yl)amino]purin-8-one | Human | 14286 | |
| PIK3CG (p110g) | PIK | Atypical | 4anv | A | A | 2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazine | Human | 9195 | |
| PIK3CG (p110g) | PIK | Atypical | 2a4z | A | | (5e)-5-[(2,2-difluoro-1,3-benzodioxol-5-yl)methylene]-1,3-thiazolidine-2,4-dione | Human | 9180 | |
| PIK3CG (p110g) | PIK | Atypical | 4wwn | A | | n-{(1s)-1-[7-fluoro-2-(pyridin-2-yl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | 9226 | |
| PIK3CG (p110g) | PIK | Atypical | 7jx0 | A | | n~3~-{[5-(4-acetylphenyl)-4-methyl-1,3-thiazol-2-yl]carbamoyl}-n-tert-butyl-beta-alaninamide | Human | 13411 | |
| PIK3CG (p110g) | PIK | Atypical | 5oq4 | A | B | 5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 9203 | |
| PIK3CG (p110g) | PIK | Atypical | 4flh | A | | 4-(2-[(5-fluoro-6-methoxypyridin-3-yl)amino]-5-{(1r)-1-[4-(methylsulfonyl)piperazin-1-yl]ethyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amine | Human | 9212 | |
| PIK3CG (p110g) | PIK | Atypical | 1he8 | A | | - | Human | 9201 | |
| PIK3CG (p110g) | PIK | Atypical | 4anv | A | B | 2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazine | Human | 9166 | |
| PIK3CG (p110g) | PIK | Atypical | 3qaq | A | | [(4-{2-[(3-hydroxyphenyl)amino]-1h-benzimidazol-1-yl}-1,3,5-triazin-2-yl)amino]acetonitrile | Human | 9211 | |
| PIK3CG (p110g) | PIK | Atypical | 4anw | A | B | 3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamide | Human | 9175 | |
| PIK3CG (p110g) | PIK | Atypical | 3l16 | A | | 5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyridin-2-amine | Human | 9233 | |
| PIK3CG (p110g) | PIK | Atypical | 3r7r | A | | 8-(acetylamino)-n-(2-chlorophenyl)-n-methyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2-carboxamide | Human | 9168 | |
| PIK3CG (p110g) | PIK | Atypical | 3r7q | A | | n-(2-chlorophenyl)-n-methyl-4h-thieno[3,2-c]chromene-2-carboxamide | Human | 9227 | |
| PIK3CG (p110g) | PIK | Atypical | 6xrm | A | | 5-[2-amino-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-2-[(1s)-1-cyclopropylethyl]-7-(trifluoromethyl)-2,3-dihydro-1h-isoindol-1-one | Human | 12775 | |
| PIK3CG (p110g) | PIK | Atypical | 4ezl | A | | 2-(1-{[2-(2-aminopyrimidin-5-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | 9235 | |
| PIK3CG (p110g) | PIK | Atypical | 4xx5 | A | | n-[5-(5-methoxypyridin-3-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide | Human | 9236 | |
| PIK3CG (p110g) | PIK | Atypical | 4ps7 | A | | n-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | 9163 | |
| PIK3CG (p110g) | PIK | Atypical | 3s2a | A | | n-{2-chloro-5-[4-(morpholin-4-yl)quinolin-6-yl]pyridin-3-yl}-4-fluorobenzenesulfonamide | Human | 9158 | |
| PIK3CG (p110g) | PIK | Atypical | 4ps8 | A | | n-[6-(5,6-dimethoxypyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | 9184 | |
| PIK3CG (p110g) | PIK | Atypical | 3l54 | A | | 6-(1h-pyrazolo[3,4-b]pyridin-5-yl)-4-pyridin-4-ylquinoline | Human | 9197 | |
| PIK3CG (p110g) | PIK | Atypical | 3qar | A | | 1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-3-yl)-1h-benzimidazol-2-amine | Human | 9178 | |
| PIK3CG (p110g) | PIK | Atypical | 4g11 | A | | 2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]-n-phenylacetamide | Human | 9223 | |
| PIK3CG (p110g) | PIK | Atypical | 6gq7 | A | | 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one | Human | 10009 | |
| PIK3CG (p110g) | PIK | Atypical | 5oq4 | A | A | 5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 9244 | |
| PIK3CG (p110g) | PIK | Atypical | 6xrn | A | | 2-amino-5-{2-[(1s)-1-cyclopropylethyl]-7-methyl-1-oxo-2,3-dihydro-1h-isoindol-5-yl}-n-(trans-3-hydroxycyclobutyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 13954 | |
| PIK3CG (p110g) | PIK | Atypical | 4ful | A | | 4-({4-[3-(piperidin-1-ylcarbonyl)phenyl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 9242 | |
| PIK3CG (p110g) | PIK | Atypical | 8dp0 | A | | - | Human | 14838 | |