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Search results (257 entries covering 80 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
DYRK1ADYRKCMGC6eisCB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10548
DYRK1ADYRKCMGC2vx3CAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3740
DYRK1ADYRKCMGC6eivB~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10536
DYRK1ADYRKCMGC7a52AB3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHuman13750
DYRK1ADYRKCMGC4mq1ABn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3736
DYRK1ADYRKCMGC2vx3CBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3735
DYRK1ADYRKCMGC4yu2BA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3737
DYRK1ADYRKCMGC5a4qAn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6717
DYRK1ADYRKCMGC4yljCA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3777
DYRK1ADYRKCMGC6s17AA~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11369
DYRK1ADYRKCMGC7aj4AA4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHuman13605
DYRK1ADYRKCMGC6uipA4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12027
DYRK1ADYRKCMGC2wo6AAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3758
DYRK1ADYRKCMGC4mq2DAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3757
DYRK1ADYRKCMGC5a4lBBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6735
DYRK1ADYRKCMGC6eipC4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10533
DYRK1ADYRKCMGC6t6aAB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11858
DYRK1ADYRKCMGC6eijB~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10516
DYRK1ADYRKCMGC7ak2A4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13593
DYRK1ADYRKCMGC7a51A4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13753
DYRK1ADYRKCMGC5a4eBBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6726
DYRK1ADYRKCMGC6ln1A1,3,5,8-tetrakis(oxidanyl)xanthen-9-oneHuman13935
DYRK1ADYRKCMGC6yf8B~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13461
DYRK1ADYRKCMGC8c3gABn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15153
DYRK1ADYRKCMGC8c3qABrutinHuman15154
DYRK1ADYRKCMGC8c3gAAn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15155
DYRK1ADYRKCMGC8c3rAAgossypinHuman15156
DYRK1ADYRKCMGC8c3rABgossypinHuman15157
DYRK1ADYRKCMGC8c3qAArutinHuman15158
DYRK1ADYRKCMGC7fhsAB(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14159
DYRK1ADYRKCMGC6qu2CA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12090
DYRK1ADYRKCMGC4azeB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3768
DYRK1ADYRKCMGC2wo6ABn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3764
DYRK1ADYRKCMGC6s11AA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11361
DYRK1ADYRKCMGC3anrB7-methoxy-1-methyl-9h-beta-carbolineHuman3729
DYRK1ADYRKCMGC5a4eDBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6733
DYRK1ADYRKCMGC6a1fAB8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10521
DYRK1ADYRKCMGC6s1jAA3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHuman11365
DYRK1ADYRKCMGC6s11BB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11372
DYRK1ADYRKCMGC6t6aAA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11857
DYRK1ADYRKCMGC6eiqB[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10529
DYRK1ADYRKCMGC6eifD4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10532
DYRK1ADYRKCMGC7a53AB(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHuman13741
DYRK1ADYRKCMGC7a5dAA4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13742
DYRK1ADYRKCMGC6ej4D3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10545
DYRK1ADYRKCMGC4nctApkc412Human3794
DYRK1ADYRKCMGC5a3xAn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6723
DYRK1ADYRKCMGC7zh8AB6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHuman14488
DYRK1ADYRKCMGC6yf8D~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13460
DYRK1ADYRKCMGC4mq1AAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3796
DYRK1ADYRKCMGC5a4tAn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6732
DYRK1ADYRKCMGC7aj8AA4-(1-benzofuran-5-yl)pyridin-2-amineHuman13587
DYRK1ADYRKCMGC7zh8AA6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHuman14489
DYRK1ADYRKCMGC4mq1DBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3763
DYRK1ADYRKCMGC6s1iCB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11373
DYRK1ADYRKCMGC7a4rAB2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHuman13743
DYRK1ADYRKCMGC7aklA4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13589
DYRK1ADYRKCMGC5a4eDAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6714
DYRK1ADYRKCMGC5aikD4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3742
DYRK1ADYRKCMGC7o7kABn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13987
DYRK1ADYRKCMGC5a3xCn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6722
DYRK1ADYRKCMGC6eipA4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10555
DYRK1ADYRKCMGC6eiqD[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10541
DYRK1ADYRKCMGC7ajmAA~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHuman13590
DYRK1ADYRKCMGC6uwyAA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11989
DYRK1ADYRKCMGC7aj5AB4-(1-benzofuran-5-yl)pyridine-2,6-diamineHuman13591
DYRK1ADYRKCMGC6eipD4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10531
DYRK1ADYRKCMGC6t6aDA-Human11862
DYRK1ADYRKCMGC4yljBB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3785
DYRK1ADYRKCMGC6a1gB5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10539
DYRK1ADYRKCMGC5a4lBAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6719
DYRK1ADYRKCMGC4mq2CAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3730
DYRK1ADYRKCMGC4azeC5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3788
DYRK1ADYRKCMGC5aikA4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3732
DYRK1ADYRKCMGC7aj2AB4-(4-methoxyphenyl)pyridin-2-amineHuman13592
DYRK1ADYRKCMGC6eivA~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10540
DYRK1ADYRKCMGC4mq1DAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3744
DYRK1ADYRKCMGC6uwyDA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11988
DYRK1ADYRKCMGC5a4lDBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6730
DYRK1ADYRKCMGC6uwyBB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11982
DYRK1ADYRKCMGC6s1jAB3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHuman11360
DYRK1ADYRKCMGC6t6aCB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11859
DYRK1ADYRKCMGC6qu2DA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12091
DYRK1ADYRKCMGC6uipB4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12025
DYRK1ADYRKCMGC6eirC~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10528
DYRK1ADYRKCMGC7a4oAphosphoaminophosphonic acid-adenylate esterHuman13744
DYRK1ADYRKCMGC6t6aCA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11863
DYRK1ADYRKCMGC4mq1CBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3750
DYRK1ADYRKCMGC2vx3ABn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3762
DYRK1ADYRKCMGC6uwyCA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11984
DYRK1ADYRKCMGC6a1gA5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10530
DYRK1ADYRKCMGC7a5dAB4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13745
DYRK1ADYRKCMGC4yu2CB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3775
DYRK1ADYRKCMGC7ajvA4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamineHuman13594
DYRK1ADYRKCMGC7a55A3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acidHuman13746
DYRK1ADYRKCMGC6eilA[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10546
DYRK1ADYRKCMGC6eiqA[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10554
DYRK1ADYRKCMGC6eilC-Human10552
DYRK1ADYRKCMGC7a5lAA4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHuman13747
DYRK1ADYRKCMGC3anqD(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3795
DYRK1ADYRKCMGC7akaAB4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13595
DYRK1ADYRKCMGC3anrA7-methoxy-1-methyl-9h-beta-carbolineHuman3778
DYRK1ADYRKCMGC6eisAB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10526
DYRK1ADYRKCMGC6eilB[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10557
DYRK1ADYRKCMGC5a54An-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6736
DYRK1ADYRKCMGC6uwyBA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11983
DYRK1ADYRKCMGC5a4lABn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6728
DYRK1ADYRKCMGC5a4eBAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6713
DYRK1ADYRKCMGC6eisCA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10535
DYRK1ADYRKCMGC7akaAA4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13596
DYRK1ADYRKCMGC4ylkAB10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3756
DYRK1ADYRKCMGC3anrD7-methoxy-1-methyl-9h-beta-carbolineHuman3755
DYRK1ADYRKCMGC7ajaAB1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHuman13597
DYRK1ADYRKCMGC6s11BA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11378
DYRK1ADYRKCMGC5a4qCn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6738
DYRK1ADYRKCMGC5a4tCn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6734
DYRK1ADYRKCMGC7ajmAB~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHuman13598
DYRK1ADYRKCMGC6eipB4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10517
DYRK1ADYRKCMGC4nctCpkc412Human3779
DYRK1ADYRKCMGC4mq1BAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3773
DYRK1ADYRKCMGC6s1iDA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11362
DYRK1ADYRKCMGC4yu2CA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3741
DYRK1ADYRKCMGC6ej4A3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10520
DYRK1ADYRKCMGC3anrC7-methoxy-1-methyl-9h-beta-carbolineHuman3783
DYRK1ADYRKCMGC6s1iDB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11379
DYRK1ADYRKCMGC6s17AB~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11375
DYRK1ADYRKCMGC6s1iCA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11366
DYRK1ADYRKCMGC7a52AA3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHuman13748
DYRK1ADYRKCMGC2vx3AAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3776
DYRK1ADYRKCMGC7ajsAA4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13599
DYRK1ADYRKCMGC6eilD[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10551
DYRK1ADYRKCMGC7a4sA7-chlorothieno[3,2-c]pyridin-4-amineHuman13749
DYRK1ADYRKCMGC7aj7A4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamineHuman13600
DYRK1ADYRKCMGC6s1hAA~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman11419
DYRK1ADYRKCMGC6eirB~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10558
DYRK1ADYRKCMGC6eisBB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10537
DYRK1ADYRKCMGC7akeA4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13601
DYRK1ADYRKCMGC5a4qBn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6729
DYRK1ADYRKCMGC6t6aDB-Human11856
DYRK1ADYRKCMGC6eivD~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10527
DYRK1ADYRKCMGC6eisDB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10543
DYRK1ADYRKCMGC6eirA~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10550
DYRK1ADYRKCMGC4yu2AA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3774
DYRK1ADYRKCMGC4yljAA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3782
DYRK1ADYRKCMGC7aj5AA4-(1-benzofuran-5-yl)pyridine-2,6-diamineHuman13602
DYRK1ADYRKCMGC6s1bAA~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11359
DYRK1ADYRKCMGC7aj8AB4-(1-benzofuran-5-yl)pyridin-2-amineHuman13603
DYRK1ADYRKCMGC6uwyCB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11985
DYRK1ADYRKCMGC5aikB4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3759
DYRK1ADYRKCMGC5a4lCAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6721
DYRK1ADYRKCMGC6eisBA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10556
DYRK1ADYRKCMGC7z5nA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14667
DYRK1ADYRKCMGC6uipC4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12026
DYRK1ADYRKCMGC5a3xDn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6718
DYRK1ADYRKCMGC4mq2BAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3792
DYRK1ADYRKCMGC4mq1BBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3770
DYRK1ADYRKCMGC2vx3DBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3790
DYRK1ADYRKCMGC4yljAB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3746
DYRK1ADYRKCMGC2vx3BBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3769
DYRK1ADYRKCMGC6eifA4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10534
DYRK1ADYRKCMGC6s1hAB~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman11420
DYRK1ADYRKCMGC5a4lCBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6711
DYRK1ADYRKCMGC6qu2CB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12087
DYRK1ADYRKCMGC7akbAB4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13604
DYRK1ADYRKCMGC5a54Dn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6710
DYRK1ADYRKCMGC5a4lAAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6731
DYRK1ADYRKCMGC4mq2DBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3734
DYRK1ADYRKCMGC4nctBpkc412Human3743
DYRK1ADYRKCMGC6eijC~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10538
DYRK1ADYRKCMGC6qu2BB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12088
DYRK1ADYRKCMGC7ajyA4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13606
DYRK1ADYRKCMGC5a4tBn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6715
DYRK1ADYRKCMGC4nctDpkc412Human3751
DYRK1ADYRKCMGC4yu2AB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3765
DYRK1ADYRKCMGC5a4eCAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6725
DYRK1ADYRKCMGC7ajsAB4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13607
DYRK1ADYRKCMGC5a4eABn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6740
DYRK1ADYRKCMGC4yljCB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3748
DYRK1ADYRKCMGC6s1iAA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11370
DYRK1ADYRKCMGC5a4eAAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6741
DYRK1ADYRKCMGC6s1iAB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11376
DYRK1ADYRKCMGC5a3xBn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6724
DYRK1ADYRKCMGC7akbAA4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13608
DYRK1ADYRKCMGC6s1iBB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11367
DYRK1ADYRKCMGC7a4wA6-(4-methoxyphenyl)pyrimidine-2,4-diamineHuman13754
DYRK1ADYRKCMGC4mq2BBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3787
DYRK1ADYRKCMGC5aikC4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3754
DYRK1ADYRKCMGC7aj2AA4-(4-methoxyphenyl)pyridin-2-amineHuman13609
DYRK1ADYRKCMGC6t6aBB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11861
DYRK1ADYRKCMGC4yllAB10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3772
DYRK1ADYRKCMGC4yu2DA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3760
DYRK1ADYRKCMGC6a1fAA8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10522
DYRK1ADYRKCMGC6ej4B3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10523
DYRK1ADYRKCMGC5a4lDAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6739
DYRK1ADYRKCMGC7fhsAA(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14160
DYRK1ADYRKCMGC6s11AB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11364
DYRK1ADYRKCMGC6qu2AA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12085
DYRK1ADYRKCMGC3anqC(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3791
DYRK1ADYRKCMGC4mq2CBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3780
DYRK1ADYRKCMGC4azeA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3761
DYRK1ADYRKCMGC6s1bAB~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11377
DYRK1ADYRKCMGC4yllAC10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3731
DYRK1ADYRKCMGC6eiqC[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10524
DYRK1ADYRKCMGC5a4tDn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6712
DYRK1ADYRKCMGC7a53AA(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHuman13755
DYRK1ADYRKCMGC4yu2DB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3733
DYRK1ADYRKCMGC4mq1CAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3781
DYRK1ADYRKCMGC6s1iBA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11371
DYRK1ADYRKCMGC6ej4C3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10519
DYRK1ADYRKCMGC2wo6BAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3749
DYRK1ADYRKCMGC7a5bA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman13756
DYRK1ADYRKCMGC5a54Cn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6720
DYRK1ADYRKCMGC6uwyAB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11987
DYRK1ADYRKCMGC4mq2AAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3752
DYRK1ADYRKCMGC6yf8A~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13462
DYRK1ADYRKCMGC7o7kAAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13988
DYRK1ADYRKCMGC3anqB(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3745
DYRK1ADYRKCMGC6eifC4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10525
DYRK1ADYRKCMGC6eijA~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10518
DYRK1ADYRKCMGC6yf8C~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13463
DYRK1ADYRKCMGC4yljDA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3784
DYRK1ADYRKCMGC5a4eCBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6727
DYRK1ADYRKCMGC6s14AB~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11421
DYRK1ADYRKCMGC6eivC~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10542
DYRK1ADYRKCMGC3anqA(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3767
DYRK1ADYRKCMGC2vx3BAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3766
DYRK1ADYRKCMGC4yljBA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3753
DYRK1ADYRKCMGC7ajaAA1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHuman13610
DYRK1ADYRKCMGC4ylkAA10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3789
DYRK1ADYRKCMGC4yljDB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3793
DYRK1ADYRKCMGC7fhtAA(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14161
DYRK1ADYRKCMGC6eifB4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10544
DYRK1ADYRKCMGC6s14AA~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11418
DYRK1ADYRKCMGC6uwyDB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11986
DYRK1ADYRKCMGC4yu2BB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3738
DYRK1ADYRKCMGC6eisDA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10547
DYRK1ADYRKCMGC6t6aBA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11860
DYRK1ADYRKCMGC6qu2DB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12089
DYRK1ADYRKCMGC5a54Bn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6716
DYRK1ADYRKCMGC2wo6BBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3739
DYRK1ADYRKCMGC7ajwAB4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13611
DYRK1ADYRKCMGC7ajwAA4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13612
DYRK1ADYRKCMGC7fhtAB(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14162
DYRK1ADYRKCMGC6eijD~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10559
DYRK1ADYRKCMGC7a5nA5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman13757
DYRK1ADYRKCMGC6qu2BA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12086
DYRK1ADYRKCMGC7a5lAB4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHuman13758
DYRK1ADYRKCMGC7aj4AB4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHuman13588
DYRK1ADYRKCMGC6eisAA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10553
DYRK1ADYRKCMGC2vx3DAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3786
DYRK1ADYRKCMGC6eirD~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10549
DYRK1ADYRKCMGC6qu2AB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12092
DYRK1ADYRKCMGC4yllAA10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3747
DYRK1ADYRKCMGC4mq2ABmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3771
DYRK1ADYRKCMGC7a4rAA2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHuman13751
DYRK1ADYRKCMGC5a4qDn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6737
DYRK1ADYRKCMGC7a4zA3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amineHuman13752
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