| MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15306 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | A | - | Human | 15311 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15297 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | B | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | 14421 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | A | ~{n}-pyridin-3-ylprop-2-enamide | Human | 14391 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14396 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | B | - | Human | 2577 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | B | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13934 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1wzy | A | | 1-allyl-5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 2618 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6n | A | B | 3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazole | Human | 2593 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8u8j | A | | (4m)-4-{(4r)-3-[(2s)-2-methylbutyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(1-methyl-1h-pyrazol-5-yl)pyrimidin-2-amine | Human | 15224 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8u8k | A | | (4m)-4-{(4s)-3-[(2-chloropyridin-3-yl)methyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(oxan-4-yl)pyrimidin-2-amine | Human | 15225 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5ngu | A | | 2-[2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one | Human | 7991 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v61 | A | A | - | Human | 8265 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1pme | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 2583 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | A | - | Human | 2588 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | A | - | Human | 11510 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv1 | A | B | n-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamide | Human | 2613 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | B | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | 14405 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | A | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | 14410 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | 14415 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6n | A | A | 3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazole | Human | 2609 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bve | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6029 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | B | | - | Human | 6081 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvd | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-one | Human | 6028 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | B | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | 14388 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | B | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | 14399 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5buj | A | A | 4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2560 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | A | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | 14409 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2626 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v62 | A | B | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 8262 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6o | A | | 4-{4-[4-(aminomethyl)-3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2565 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | A | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | 14389 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | B | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | 14393 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv4 | A | A | 9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrile | Human | 2623 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5wp1 | A | B | 5,7-dihydroxy-4h-1-benzopyran-4-one | Human | 10440 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | 11408 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3i5z | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamide | Human | 2579 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | A | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | 14395 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | A | thiophen-3-ylmethylazanium | Human | 10983 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 2585 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv5 | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-(5-methyl-2-phenylpyrimidin-4-yl)-1h-pyrrole-2-carboxamide | Human | 2598 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14397 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv8 | A | A | 6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-one | Human | 2625 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | A | - | Human | 10811 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | 9958 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzn | A | A | 2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamide | Human | 2605 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | A | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | 11815 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | B | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 10831 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | B | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | 14413 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | A | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | 11854 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14661 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14660 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | A | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | 14084 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | 9960 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv3 | A | A | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 2617 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1tvo | A | | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 2581 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | A | pyridin-2-amine | Human | 11352 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nho | A | | (6~{s})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7993 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3p | D | | phosphoaminophosphonic acid-adenylate ester | Human | 2575 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvd | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-one | Human | 6030 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13922 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13927 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | 13928 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | 13929 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7w5o | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14110 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13930 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | 13931 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | B | | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6093 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | 11412 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | B | phosphoaminophosphonic acid-adenylate ester | Human | 2591 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13925 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | B | - | Human | 15303 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | A | - | Human | 15304 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | B | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | 2564 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | A | n-cyclohexyl-9h-purin-6-amine | Human | 6086 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv0 | A | A | n-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amine | Human | 2562 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | A | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | 14385 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhp | A | | 5-(2-methoxyethyl)-1-methyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydropyrrolo[3,2-c]pyridin-4-one | Human | 7998 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | B | | n-benzyl-9h-purin-6-amine | Human | 6080 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6oph | A | | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 11509 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | A | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14386 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | A | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | 14387 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3q | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2611 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2ojj | A | | (s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamide | Human | 2612 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | 9970 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | A | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13921 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | A | - | Human | 2569 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | B | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | 11816 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | 9961 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7k | A | | 1h-imidazol-2-amine | Human | 10985 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15298 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | A | - | Human | 11349 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | A | | adenosine-5'-diphosphate | Human | 2554 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qpa | A | | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6077 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | B | - | Human | 2597 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g8x | A | A | 4-chloranyl-1~{h}-indazol-3-amine | Human | 9957 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fux | A | | trans-4-{[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)pyrimidin-2-yl]amino}cyclohexanol | Human | 2568 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | 9972 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | B | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14390 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | 9944 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | B | thiophen-3-ylmethylazanium | Human | 10989 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13923 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g93 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-one | Human | 9959 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | A | n-cyclohexyl-9h-purin-6-amine | Human | 6088 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | 14392 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | A | | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | 6084 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | A | | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6082 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | A | catechol | Human | 6654 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | 9971 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | 14394 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13924 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | B | pyrazole | Human | 11345 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | A | caffeic acid | Human | 2589 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhh | A | | 5-(2-methoxyethyl)-2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7996 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzn | A | B | 2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamide | Human | 2610 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | A | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | 2559 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | A | phosphoaminophosphonic acid-adenylate ester | Human | 2621 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | 13926 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g54 | A | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10937 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e73 | A | | - | Human | 14114 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | D | | adenosine-5'-diphosphate | Human | 2578 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvf | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6031 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lck | A | B | ~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 6836 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | B | - | Human | 15299 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | A | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | 9968 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | 9964 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv1 | A | A | n-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamide | Human | 2594 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | 11413 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fuy | A | A | {4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanone | Human | 2622 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | B | 1-azanylpropylideneazanium | Human | 11348 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | A | | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6087 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | B | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | 14083 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | B | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | 14398 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | B | catechol | Human | 6653 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | 9953 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | A | 1~{h}-1,2,3-triazole | Human | 10988 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | 9966 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | A | | 5h-pyrrolo[2,3-b]pyrazine | Human | 6089 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fmq | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2604 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | B | - | Human | 2627 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | A | 1,2-oxazol-3-amine | Human | 11350 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g91 | A | B | 5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amine | Human | 9956 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opg | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11507 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | 14400 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3tei | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2608 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2ojg | A | | n,n-dimethyl-4-(4-phenyl-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamide | Human | 2603 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g8x | A | B | 4-chloranyl-1~{h}-indazol-3-amine | Human | 9954 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | 11410 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv3 | A | B | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 2580 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | A | | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | 6048 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | C | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14401 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv2 | A | B | 4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2571 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3p | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2624 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | A | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | 14402 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | A | 1~{h}-pyridin-2-one | Human | 11344 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5buj | A | B | 4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2561 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15300 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5ax3 | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 6398 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | B | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | 9946 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | B | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 10810 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | A | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | 14403 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv8 | A | B | 6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-one | Human | 2601 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3i60 | A | | 4-{2-[(2-chlorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-phenylethyl]-1h-pyrrole-2-carboxamide | Human | 2584 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv6 | A | | n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-(2-{[(2s)-1-hydroxybutan-2-yl]amino}-5-methylpyrimidin-4-yl)-1h-pyrrole-2-carboxamide | Human | 2551 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhv | A | | 7-[2-(oxan-4-ylamino)pyrimidin-4-yl]-3,4-dihydro-2~{h}-pyrrolo[1,2-a]pyrazin-1-one | Human | 7995 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | A | 1,1-bis(oxidanylidene)thietan-3-ol | Human | 10987 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv9 | A | A | 3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 2582 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | C | | adenosine-5'-diphosphate | Human | 2595 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g92 | A | A | ~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amine | Human | 11409 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3sa0 | A | B | norathyriol | Human | 2557 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lcj | A | B | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 6834 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v60 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 8263 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g54 | A | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10938 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | B | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | 14404 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15301 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 2602 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | B | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | 14406 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e75 | A | | - | Human | 14115 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | A | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | 9948 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bve | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6026 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | B | ~{n}-pyridin-3-ylpropanamide | Human | 14407 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opi | A | | (3r)-n-[3-(2-cyclopropylpyridin-4-yl)-1h-indazol-5-yl]-3-(methoxymethyl)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]-3,6-dihydropyridin-1(2h)-yl}ethyl)pyrrolidine-3-carboxamide | Human | 11511 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | 9947 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2oji | A | | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | 2570 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15302 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | B | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | 10986 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvf | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6027 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | B | n-cyclohexyl-9h-purin-6-amine | Human | 6075 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | B | | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6076 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | B | - | Human | 15305 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv2 | A | A | 4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2592 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psy | A | | - | Human | 15308 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | B | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | 14408 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | 9952 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | B | | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | 6079 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv7 | A | A | 4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrile | Human | 2572 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 2566 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lck | A | A | ~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 6835 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3w55 | A | | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 2573 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bue | A | | 1-benzyl-4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2574 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7xc1 | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14665 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhf | A | | 2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-5-(phenylmethyl)-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7997 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fuy | A | B | {4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanone | Human | 2587 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | A | - | Human | 2586 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp9 | A | | 7-(1-propyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6085 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qpa | B | | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6090 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | A | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 10832 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | B | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | 14411 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v61 | A | B | - | Human | 8266 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 2567 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | A | pyrazole | Human | 11353 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | A | 1-[(2~{s})-2-(5-methyl-3-pyridin-4-yl-1~{h}-pyrazol-4-yl)pyrrolidin-1-yl]propan-1-one | Human | 14412 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rfo | A | | - | Human | 12341 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | B | | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | 6049 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | B | - | Human | 2607 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | A | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | 2590 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15307 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15309 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5wp1 | A | A | 5,7-dihydroxy-4h-1-benzopyran-4-one | Human | 10441 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | B | caffeic acid | Human | 2555 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzm | A | | 7-ethylsulfonyl-n-(oxan-4-yl)-6,8-dihydro-5h-pyrido[3,4-d]pyrimidin-2-amine | Human | 2616 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v62 | A | A | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 8264 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | B | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14414 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | A | - | Human | 15310 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | C | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 10809 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | B | pyridin-2-amine | Human | 11346 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | 13932 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv9 | A | B | 3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 2552 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | B | n-cyclohexyl-9h-purin-6-amine | Human | 6083 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | A | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | 14416 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | B | 1,2-oxazol-3-amine | Human | 11347 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5k4i | A | | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 6744 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g93 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-one | Human | 9955 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | B | | 5h-pyrrolo[2,3-b]pyrazine | Human | 6091 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhl | A | | (6~{r})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7992 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6d5y | A | | - | Human | 10939 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv4 | A | B | 9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrile | Human | 2558 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | B | - | Human | 11343 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g92 | A | B | ~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amine | Human | 11411 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | A | | n-benzyl-9h-purin-6-amine | Human | 6092 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | A | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | 14417 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | 9950 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | B | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | 11855 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv7 | A | B | 4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrile | Human | 2614 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | B | - | Human | 11508 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | B | - | Human | 14418 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | B | 1~{h}-1,2,3-triazole | Human | 10982 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | A | | 5-chloro-1,3-benzoxazol-2-amine | Human | 6078 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2556 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | 9949 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | A | - | Human | 2615 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 2576 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | A | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | 14419 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lcj | A | A | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 6833 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhj | A | | 5-(2-methoxyethyl)-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7994 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | B | | adenosine-5'-diphosphate | Human | 2600 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | A | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14420 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3sa0 | A | A | norathyriol | Human | 2596 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | A | 1-azanylpropylideneazanium | Human | 11354 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | A | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | 10984 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bui | A | | 3-(4-fluorophenyl)-5-(pyridin-2-yl)-4,5,6,7-tetrahydro-2h-pyrazolo[4,3-c]pyridine | Human | 2563 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | B | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | 10830 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzo | A | A | n-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 2620 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | B | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | 2553 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | B | 1,1-bis(oxidanylidene)thietan-3-ol | Human | 10981 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g91 | A | A | 5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amine | Human | 9965 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fmq | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2619 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzo | A | B | n-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 2606 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | B | 1~{h}-pyridin-2-one | Human | 11351 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v60 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 8261 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | B | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | 9973 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | A | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | 10829 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | 13933 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv0 | A | B | n-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amine | Human | 2599 | |