Search results (275 entries covering 152 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
MAPK1 (Erk2)MAPKCMGC8pt5AAphosphoaminophosphonic acid-adenylate esterHuman15306
MAPK1 (Erk2)MAPKCMGC8pstAA-Human15311
MAPK1 (Erk2)MAPKCMGC8pt0AAphosphoaminophosphonic acid-adenylate esterHuman15297
MAPK1 (Erk2)MAPKCMGC8aogAB~{n}-(5-methyl-1,2-oxazol-3-yl)propanamideHuman14421
MAPK1 (Erk2)MAPKCMGC8aoaAA~{n}-pyridin-3-ylprop-2-enamideHuman14391
MAPK1 (Erk2)MAPKCMGC8ao6AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14396
MAPK1 (Erk2)MAPKCMGC4iz7AB-Human2577
MAPK1 (Erk2)MAPKCMGC7nr5AB(2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13934
MAPK1 (Erk2)MAPKCMGC1wzyA1-allyl-5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman2618
MAPK1 (Erk2)MAPKCMGC4g6nAB3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHuman2593
MAPK1 (Erk2)MAPKCMGC8u8jA(4m)-4-{(4r)-3-[(2s)-2-methylbutyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(1-methyl-1h-pyrazol-5-yl)pyrimidin-2-amineHuman15224
MAPK1 (Erk2)MAPKCMGC8u8kA(4m)-4-{(4s)-3-[(2-chloropyridin-3-yl)methyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(oxan-4-yl)pyrimidin-2-amineHuman15225
MAPK1 (Erk2)MAPKCMGC5nguA2-[2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneHuman7991
MAPK1 (Erk2)MAPKCMGC5v61AA-Human8265
MAPK1 (Erk2)MAPKCMGC1pmeA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman2583
MAPK1 (Erk2)MAPKCMGC4izaCA-Human2588
MAPK1 (Erk2)MAPKCMGC6nbsAA-Human11510
MAPK1 (Erk2)MAPKCMGC4fv1ABn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHuman2613
MAPK1 (Erk2)MAPKCMGC8ao8AB1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-oneHuman14405
MAPK1 (Erk2)MAPKCMGC8ao8AA1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-oneHuman14410
MAPK1 (Erk2)MAPKCMGC8ao2AA~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman14415
MAPK1 (Erk2)MAPKCMGC4g6nAA3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHuman2609
MAPK1 (Erk2)MAPKCMGC5bveAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6029
MAPK1 (Erk2)MAPKCMGC4qp2B-Human6081
MAPK1 (Erk2)MAPKCMGC5bvdAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-oneHuman6028
MAPK1 (Erk2)MAPKCMGC8aodAB1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-oneHuman14388
MAPK1 (Erk2)MAPKCMGC8ao4AB~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman14399
MAPK1 (Erk2)MAPKCMGC5bujAA4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2560
MAPK1 (Erk2)MAPKCMGC8aocAA~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamideHuman14409
MAPK1 (Erk2)MAPKCMGC2y9qAAphosphoaminophosphonic acid-adenylate esterHuman2626
MAPK1 (Erk2)MAPKCMGC5v62AB5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman8262
MAPK1 (Erk2)MAPKCMGC4g6oA4-{4-[4-(aminomethyl)-3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2565
MAPK1 (Erk2)MAPKCMGC8ao7AA~{n}-[(1-methylindazol-6-yl)methyl]propanamideHuman14389
MAPK1 (Erk2)MAPKCMGC8aoiAB1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-oneHuman14393
MAPK1 (Erk2)MAPKCMGC4fv4AA9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHuman2623
MAPK1 (Erk2)MAPKCMGC5wp1AB5,7-dihydroxy-4h-1-benzopyran-4-oneHuman10440
MAPK1 (Erk2)MAPKCMGC6g9aAA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-oneHuman11408
MAPK1 (Erk2)MAPKCMGC3i5zAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman2579
MAPK1 (Erk2)MAPKCMGC8aoeAA~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamideHuman14395
MAPK1 (Erk2)MAPKCMGC6qaqAAthiophen-3-ylmethylazaniumHuman10983
MAPK1 (Erk2)MAPKCMGC4nifBAphosphoaminophosphonic acid-adenylate esterHuman2585
MAPK1 (Erk2)MAPKCMGC4fv5An-[(1s)-2-hydroxy-1-phenylethyl]-4-(5-methyl-2-phenylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHuman2598
MAPK1 (Erk2)MAPKCMGC8ao6AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14397
MAPK1 (Erk2)MAPKCMGC4fv8AA6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHuman2625
MAPK1 (Erk2)MAPKCMGC6dmgAA-Human10811
MAPK1 (Erk2)MAPKCMGC6g9hAB~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamideHuman9958
MAPK1 (Erk2)MAPKCMGC4zznAA2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamideHuman2605
MAPK1 (Erk2)MAPKCMGC6slgAA(6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-oneHuman11815
MAPK1 (Erk2)MAPKCMGC6gjbAB[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman10831
MAPK1 (Erk2)MAPKCMGC8aobAB~{n}-[(1-methylindazol-3-yl)methyl]propanamideHuman14413
MAPK1 (Erk2)MAPKCMGC6rq4AA6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-oneHuman11854
MAPK1 (Erk2)MAPKCMGC7x4uAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14661
MAPK1 (Erk2)MAPKCMGC7x4uAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14660
MAPK1 (Erk2)MAPKCMGC7opmAA1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]ureaHuman14084
MAPK1 (Erk2)MAPKCMGC6g97AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-oneHuman9960
MAPK1 (Erk2)MAPKCMGC4fv3AAethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman2617
MAPK1 (Erk2)MAPKCMGC1tvoA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman2581
MAPK1 (Erk2)MAPKCMGC6qa1AApyridin-2-amineHuman11352
MAPK1 (Erk2)MAPKCMGC5nhoA(6~{s})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7993
MAPK1 (Erk2)MAPKCMGC4h3pDphosphoaminophosphonic acid-adenylate esterHuman2575
MAPK1 (Erk2)MAPKCMGC5bvdAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-oneHuman6030
MAPK1 (Erk2)MAPKCMGC7nr3AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-oneHuman13922
MAPK1 (Erk2)MAPKCMGC7nqwAA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-oneHuman13927
MAPK1 (Erk2)MAPKCMGC7nqqAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamideHuman13928
MAPK1 (Erk2)MAPKCMGC7nr8AB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamideHuman13929
MAPK1 (Erk2)MAPKCMGC7w5oA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14110
MAPK1 (Erk2)MAPKCMGC7auvAB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13930
MAPK1 (Erk2)MAPKCMGC7nr9AB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamideHuman13931
MAPK1 (Erk2)MAPKCMGC4qp7B2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6093
MAPK1 (Erk2)MAPKCMGC6g9aAB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-oneHuman11412
MAPK1 (Erk2)MAPKCMGC4nifEBphosphoaminophosphonic acid-adenylate esterHuman2591
MAPK1 (Erk2)MAPKCMGC7auvAA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13925
MAPK1 (Erk2)MAPKCMGC8pswAB-Human15303
MAPK1 (Erk2)MAPKCMGC8pt3AA-Human15304
MAPK1 (Erk2)MAPKCMGC4qteAB4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamideHuman2564
MAPK1 (Erk2)MAPKCMGC4qp4BAn-cyclohexyl-9h-purin-6-amineHuman6086
MAPK1 (Erk2)MAPKCMGC4fv0AAn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHuman2562
MAPK1 (Erk2)MAPKCMGC8aohAA~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamideHuman14385
MAPK1 (Erk2)MAPKCMGC5nhpA5-(2-methoxyethyl)-1-methyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydropyrrolo[3,2-c]pyridin-4-oneHuman7998
MAPK1 (Erk2)MAPKCMGC4qp1Bn-benzyl-9h-purin-6-amineHuman6080
MAPK1 (Erk2)MAPKCMGC6ophA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman11509
MAPK1 (Erk2)MAPKCMGC8ao3AA2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14386
MAPK1 (Erk2)MAPKCMGC8aoiAA1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-oneHuman14387
MAPK1 (Erk2)MAPKCMGC4h3qAphosphoaminophosphonic acid-adenylate esterHuman2611
MAPK1 (Erk2)MAPKCMGC2ojjA(s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHuman2612
MAPK1 (Erk2)MAPKCMGC6g97AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-oneHuman9970
MAPK1 (Erk2)MAPKCMGC7nr5AA(2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13921
MAPK1 (Erk2)MAPKCMGC4iz7CA-Human2569
MAPK1 (Erk2)MAPKCMGC6slgAB(6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-oneHuman11816
MAPK1 (Erk2)MAPKCMGC6ge0AB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamideHuman9961
MAPK1 (Erk2)MAPKCMGC6q7kA1h-imidazol-2-amineHuman10985
MAPK1 (Erk2)MAPKCMGC8psrABphosphoaminophosphonic acid-adenylate esterHuman15298
MAPK1 (Erk2)MAPKCMGC6q7sAA-Human11349
MAPK1 (Erk2)MAPKCMGC4iz5Aadenosine-5'-diphosphateHuman2554
MAPK1 (Erk2)MAPKCMGC4qpaA7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6077
MAPK1 (Erk2)MAPKCMGC4iz7CB-Human2597
MAPK1 (Erk2)MAPKCMGC6g8xAA4-chloranyl-1~{h}-indazol-3-amineHuman9957
MAPK1 (Erk2)MAPKCMGC4fuxAtrans-4-{[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)pyrimidin-2-yl]amino}cyclohexanolHuman2568
MAPK1 (Erk2)MAPKCMGC6g9dAA~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamideHuman9972
MAPK1 (Erk2)MAPKCMGC8ao9AB1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14390
MAPK1 (Erk2)MAPKCMGC6g9mAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamideHuman9944
MAPK1 (Erk2)MAPKCMGC6qaqABthiophen-3-ylmethylazaniumHuman10989
MAPK1 (Erk2)MAPKCMGC7nr3AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-oneHuman13923
MAPK1 (Erk2)MAPKCMGC6g93AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-oneHuman9959
MAPK1 (Erk2)MAPKCMGC4qp4AAn-cyclohexyl-9h-purin-6-amineHuman6088
MAPK1 (Erk2)MAPKCMGC8ao5AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman14392
MAPK1 (Erk2)MAPKCMGC4qp3A(2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-olHuman6084
MAPK1 (Erk2)MAPKCMGC4qp7A2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6082
MAPK1 (Erk2)MAPKCMGC4zxtAAcatecholHuman6654
MAPK1 (Erk2)MAPKCMGC6g9hAA~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamideHuman9971
MAPK1 (Erk2)MAPKCMGC8ao2AB~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman14394
MAPK1 (Erk2)MAPKCMGC7nqwAB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-oneHuman13924
MAPK1 (Erk2)MAPKCMGC6qa3ABpyrazoleHuman11345
MAPK1 (Erk2)MAPKCMGC4n0sAAcaffeic acidHuman2589
MAPK1 (Erk2)MAPKCMGC5nhhA5-(2-methoxyethyl)-2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7996
MAPK1 (Erk2)MAPKCMGC4zznAB2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamideHuman2610
MAPK1 (Erk2)MAPKCMGC4o6eAAn-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamideHuman2559
MAPK1 (Erk2)MAPKCMGC4nifEAphosphoaminophosphonic acid-adenylate esterHuman2621
MAPK1 (Erk2)MAPKCMGC7nqqAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamideHuman13926
MAPK1 (Erk2)MAPKCMGC6g54ABn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10937
MAPK1 (Erk2)MAPKCMGC7e73A-Human14114
MAPK1 (Erk2)MAPKCMGC4iz5Dadenosine-5'-diphosphateHuman2578
MAPK1 (Erk2)MAPKCMGC5bvfAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6031
MAPK1 (Erk2)MAPKCMGC5lckAB~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamideHuman6836
MAPK1 (Erk2)MAPKCMGC8pstAB-Human15299
MAPK1 (Erk2)MAPKCMGC6gdmAA(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamideHuman9968
MAPK1 (Erk2)MAPKCMGC6g9mAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamideHuman9964
MAPK1 (Erk2)MAPKCMGC4fv1AAn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHuman2594
MAPK1 (Erk2)MAPKCMGC6g9nAB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamideHuman11413
MAPK1 (Erk2)MAPKCMGC4fuyAA{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHuman2622
MAPK1 (Erk2)MAPKCMGC6qahAB1-azanylpropylideneazaniumHuman11348
MAPK1 (Erk2)MAPKCMGC4qp8A2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6087
MAPK1 (Erk2)MAPKCMGC7opmAB1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]ureaHuman14083
MAPK1 (Erk2)MAPKCMGC8ao7AB~{n}-[(1-methylindazol-6-yl)methyl]propanamideHuman14398
MAPK1 (Erk2)MAPKCMGC4zxtABcatecholHuman6653
MAPK1 (Erk2)MAPKCMGC6g9dAB~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamideHuman9953
MAPK1 (Erk2)MAPKCMGC6qagAA1~{h}-1,2,3-triazoleHuman10988
MAPK1 (Erk2)MAPKCMGC6g9kAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamideHuman9966
MAPK1 (Erk2)MAPKCMGC4qp6A5h-pyrrolo[2,3-b]pyrazineHuman6089
MAPK1 (Erk2)MAPKCMGC4fmqAAphosphoaminophosphonic acid-adenylate esterHuman2604
MAPK1 (Erk2)MAPKCMGC4izaCB-Human2627
MAPK1 (Erk2)MAPKCMGC6q7tAA1,2-oxazol-3-amineHuman11350
MAPK1 (Erk2)MAPKCMGC6g91AB5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amineHuman9956
MAPK1 (Erk2)MAPKCMGC6opgAphosphoaminophosphonic acid-adenylate esterHuman11507
MAPK1 (Erk2)MAPKCMGC8ao5AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman14400
MAPK1 (Erk2)MAPKCMGC3teiAphosphoaminophosphonic acid-adenylate esterHuman2608
MAPK1 (Erk2)MAPKCMGC2ojgAn,n-dimethyl-4-(4-phenyl-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHuman2603
MAPK1 (Erk2)MAPKCMGC6g8xAB4-chloranyl-1~{h}-indazol-3-amineHuman9954
MAPK1 (Erk2)MAPKCMGC6g9nAA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamideHuman11410
MAPK1 (Erk2)MAPKCMGC4fv3ABethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman2580
MAPK1 (Erk2)MAPKCMGC4xj0A1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-oneHuman6048
MAPK1 (Erk2)MAPKCMGC8ao9AC1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14401
MAPK1 (Erk2)MAPKCMGC4fv2AB4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2571
MAPK1 (Erk2)MAPKCMGC4h3pAphosphoaminophosphonic acid-adenylate esterHuman2624
MAPK1 (Erk2)MAPKCMGC8aobAA~{n}-[(1-methylindazol-3-yl)methyl]propanamideHuman14402
MAPK1 (Erk2)MAPKCMGC6qa4AA1~{h}-pyridin-2-oneHuman11344
MAPK1 (Erk2)MAPKCMGC5bujAB4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2561
MAPK1 (Erk2)MAPKCMGC8psrAAphosphoaminophosphonic acid-adenylate esterHuman15300
MAPK1 (Erk2)MAPKCMGC5ax3A(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman6398
MAPK1 (Erk2)MAPKCMGC6gdmAB(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamideHuman9946
MAPK1 (Erk2)MAPKCMGC6dmgABethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman10810
MAPK1 (Erk2)MAPKCMGC8aogAA~{n}-(5-methyl-1,2-oxazol-3-yl)propanamideHuman14403
MAPK1 (Erk2)MAPKCMGC4fv8AB6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHuman2601
MAPK1 (Erk2)MAPKCMGC3i60A4-{2-[(2-chlorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-phenylethyl]-1h-pyrrole-2-carboxamideHuman2584
MAPK1 (Erk2)MAPKCMGC4fv6An-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-(2-{[(2s)-1-hydroxybutan-2-yl]amino}-5-methylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHuman2551
MAPK1 (Erk2)MAPKCMGC5nhvA7-[2-(oxan-4-ylamino)pyrimidin-4-yl]-3,4-dihydro-2~{h}-pyrrolo[1,2-a]pyrazin-1-oneHuman7995
MAPK1 (Erk2)MAPKCMGC6qalAA1,1-bis(oxidanylidene)thietan-3-olHuman10987
MAPK1 (Erk2)MAPKCMGC4fv9AA3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman2582
MAPK1 (Erk2)MAPKCMGC4iz5Cadenosine-5'-diphosphateHuman2595
MAPK1 (Erk2)MAPKCMGC6g92AA~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amineHuman11409
MAPK1 (Erk2)MAPKCMGC3sa0ABnorathyriolHuman2557
MAPK1 (Erk2)MAPKCMGC5lcjAB[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman6834
MAPK1 (Erk2)MAPKCMGC5v60ABphosphomethylphosphonic acid adenylate esterHuman8263
MAPK1 (Erk2)MAPKCMGC6g54AAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10938
MAPK1 (Erk2)MAPKCMGC8aohAB~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamideHuman14404
MAPK1 (Erk2)MAPKCMGC8pt5ABphosphoaminophosphonic acid-adenylate esterHuman15301
MAPK1 (Erk2)MAPKCMGC4qtaAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman2602
MAPK1 (Erk2)MAPKCMGC8aocAB~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamideHuman14406
MAPK1 (Erk2)MAPKCMGC7e75A-Human14115
MAPK1 (Erk2)MAPKCMGC6gdqAA4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamideHuman9948
MAPK1 (Erk2)MAPKCMGC5bveAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6026
MAPK1 (Erk2)MAPKCMGC8aoaAB~{n}-pyridin-3-ylpropanamideHuman14407
MAPK1 (Erk2)MAPKCMGC6opiA(3r)-n-[3-(2-cyclopropylpyridin-4-yl)-1h-indazol-5-yl]-3-(methoxymethyl)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]-3,6-dihydropyridin-1(2h)-yl}ethyl)pyrrolidine-3-carboxamideHuman11511
MAPK1 (Erk2)MAPKCMGC6g9kAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamideHuman9947
MAPK1 (Erk2)MAPKCMGC2ojiAn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHuman2570
MAPK1 (Erk2)MAPKCMGC8pt1AAphosphoaminophosphonic acid-adenylate esterHuman15302
MAPK1 (Erk2)MAPKCMGC6qawAB[1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazaniumHuman10986
MAPK1 (Erk2)MAPKCMGC5bvfAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6027
MAPK1 (Erk2)MAPKCMGC4qp4ABn-cyclohexyl-9h-purin-6-amineHuman6075
MAPK1 (Erk2)MAPKCMGC4qp8B2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6076
MAPK1 (Erk2)MAPKCMGC8pt3AB-Human15305
MAPK1 (Erk2)MAPKCMGC4fv2AA4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2592
MAPK1 (Erk2)MAPKCMGC8psyA-Human15308
MAPK1 (Erk2)MAPKCMGC8aofAB~{n}-(2-methylpyrimidin-5-yl)propanamideHuman14408
MAPK1 (Erk2)MAPKCMGC6g9jAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamideHuman9952
MAPK1 (Erk2)MAPKCMGC4qp3B(2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-olHuman6079
MAPK1 (Erk2)MAPKCMGC4fv7AA4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHuman2572
MAPK1 (Erk2)MAPKCMGC4nifBBphosphoaminophosphonic acid-adenylate esterHuman2566
MAPK1 (Erk2)MAPKCMGC5lckAA~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamideHuman6835
MAPK1 (Erk2)MAPKCMGC3w55A(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman2573
MAPK1 (Erk2)MAPKCMGC5bueA1-benzyl-4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2574
MAPK1 (Erk2)MAPKCMGC7xc1A(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14665
MAPK1 (Erk2)MAPKCMGC5nhfA2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-5-(phenylmethyl)-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7997
MAPK1 (Erk2)MAPKCMGC4fuyAB{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHuman2587
MAPK1 (Erk2)MAPKCMGC4izaAA-Human2586
MAPK1 (Erk2)MAPKCMGC4qp9A7-(1-propyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6085
MAPK1 (Erk2)MAPKCMGC4qpaB7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6090
MAPK1 (Erk2)MAPKCMGC6gjbAA[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman10832
MAPK1 (Erk2)MAPKCMGC8aoeAB~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamideHuman14411
MAPK1 (Erk2)MAPKCMGC5v61AB-Human8266
MAPK1 (Erk2)MAPKCMGC2y9qACphosphoaminophosphonic acid-adenylate esterHuman2567
MAPK1 (Erk2)MAPKCMGC6qa3AApyrazoleHuman11353
MAPK1 (Erk2)MAPKCMGC8aojAA1-[(2~{s})-2-(5-methyl-3-pyridin-4-yl-1~{h}-pyrazol-4-yl)pyrrolidin-1-yl]propan-1-oneHuman14412
MAPK1 (Erk2)MAPKCMGC6rfoA-Human12341
MAPK1 (Erk2)MAPKCMGC4xj0B1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-oneHuman6049
MAPK1 (Erk2)MAPKCMGC4izaAB-Human2607
MAPK1 (Erk2)MAPKCMGC4qteAA4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamideHuman2590
MAPK1 (Erk2)MAPKCMGC8pt0ABphosphoaminophosphonic acid-adenylate esterHuman15307
MAPK1 (Erk2)MAPKCMGC8pt1ABphosphoaminophosphonic acid-adenylate esterHuman15309
MAPK1 (Erk2)MAPKCMGC5wp1AA5,7-dihydroxy-4h-1-benzopyran-4-oneHuman10441
MAPK1 (Erk2)MAPKCMGC4n0sABcaffeic acidHuman2555
MAPK1 (Erk2)MAPKCMGC4zzmA7-ethylsulfonyl-n-(oxan-4-yl)-6,8-dihydro-5h-pyrido[3,4-d]pyrimidin-2-amineHuman2616
MAPK1 (Erk2)MAPKCMGC5v62AA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman8264
MAPK1 (Erk2)MAPKCMGC8ao3AB2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14414
MAPK1 (Erk2)MAPKCMGC8pswAA-Human15310
MAPK1 (Erk2)MAPKCMGC6dmgACethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman10809
MAPK1 (Erk2)MAPKCMGC6qa1ABpyridin-2-amineHuman11346
MAPK1 (Erk2)MAPKCMGC7nr9AA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamideHuman13932
MAPK1 (Erk2)MAPKCMGC4fv9AB3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman2552
MAPK1 (Erk2)MAPKCMGC4qp4BBn-cyclohexyl-9h-purin-6-amineHuman6083
MAPK1 (Erk2)MAPKCMGC8ao4AA~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman14416
MAPK1 (Erk2)MAPKCMGC6q7tAB1,2-oxazol-3-amineHuman11347
MAPK1 (Erk2)MAPKCMGC5k4iA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6744
MAPK1 (Erk2)MAPKCMGC6g93AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-oneHuman9955
MAPK1 (Erk2)MAPKCMGC4qp6B5h-pyrrolo[2,3-b]pyrazineHuman6091
MAPK1 (Erk2)MAPKCMGC5nhlA(6~{r})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7992
MAPK1 (Erk2)MAPKCMGC6d5yA-Human10939
MAPK1 (Erk2)MAPKCMGC4fv4AB9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHuman2558
MAPK1 (Erk2)MAPKCMGC6q7sAB-Human11343
MAPK1 (Erk2)MAPKCMGC6g92AB~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amineHuman11411
MAPK1 (Erk2)MAPKCMGC4qp1An-benzyl-9h-purin-6-amineHuman6092
MAPK1 (Erk2)MAPKCMGC8aodAA1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-oneHuman14417
MAPK1 (Erk2)MAPKCMGC6ge0AA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamideHuman9950
MAPK1 (Erk2)MAPKCMGC6rq4AB6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-oneHuman11855
MAPK1 (Erk2)MAPKCMGC4fv7AB4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHuman2614
MAPK1 (Erk2)MAPKCMGC6nbsAB-Human11508
MAPK1 (Erk2)MAPKCMGC8aojAB-Human14418
MAPK1 (Erk2)MAPKCMGC6qagAB1~{h}-1,2,3-triazoleHuman10982
MAPK1 (Erk2)MAPKCMGC4qp2A5-chloro-1,3-benzoxazol-2-amineHuman6078
MAPK1 (Erk2)MAPKCMGC2y9qABphosphoaminophosphonic acid-adenylate esterHuman2556
MAPK1 (Erk2)MAPKCMGC6g9jAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamideHuman9949
MAPK1 (Erk2)MAPKCMGC4iz7AA-Human2615
MAPK1 (Erk2)MAPKCMGC4qtaAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman2576
MAPK1 (Erk2)MAPKCMGC8aofAA~{n}-(2-methylpyrimidin-5-yl)propanamideHuman14419
MAPK1 (Erk2)MAPKCMGC5lcjAA[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman6833
MAPK1 (Erk2)MAPKCMGC5nhjA5-(2-methoxyethyl)-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7994
MAPK1 (Erk2)MAPKCMGC4iz5Badenosine-5'-diphosphateHuman2600
MAPK1 (Erk2)MAPKCMGC8ao9AA1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14420
MAPK1 (Erk2)MAPKCMGC3sa0AAnorathyriolHuman2596
MAPK1 (Erk2)MAPKCMGC6qahAA1-azanylpropylideneazaniumHuman11354
MAPK1 (Erk2)MAPKCMGC6qawAA[1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazaniumHuman10984
MAPK1 (Erk2)MAPKCMGC5buiA3-(4-fluorophenyl)-5-(pyridin-2-yl)-4,5,6,7-tetrahydro-2h-pyrazolo[4,3-c]pyridineHuman2563
MAPK1 (Erk2)MAPKCMGC6gjdABcyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamateHuman10830
MAPK1 (Erk2)MAPKCMGC4zzoAAn-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamideHuman2620
MAPK1 (Erk2)MAPKCMGC4o6eABn-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamideHuman2553
MAPK1 (Erk2)MAPKCMGC6qalAB1,1-bis(oxidanylidene)thietan-3-olHuman10981
MAPK1 (Erk2)MAPKCMGC6g91AA5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amineHuman9965
MAPK1 (Erk2)MAPKCMGC4fmqABphosphoaminophosphonic acid-adenylate esterHuman2619
MAPK1 (Erk2)MAPKCMGC4zzoABn-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamideHuman2606
MAPK1 (Erk2)MAPKCMGC6qa4AB1~{h}-pyridin-2-oneHuman11351
MAPK1 (Erk2)MAPKCMGC5v60AAphosphomethylphosphonic acid adenylate esterHuman8261
MAPK1 (Erk2)MAPKCMGC6gdqAB4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamideHuman9973
MAPK1 (Erk2)MAPKCMGC6gjdAAcyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamateHuman10829
MAPK1 (Erk2)MAPKCMGC7nr8AA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamideHuman13933
MAPK1 (Erk2)MAPKCMGC4fv0ABn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHuman2599