Search results (72 entries covering 46 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PAK4STE20STE4l67A-Human1376
PAK4STE20STE4njdAAn-(1h-indazol-5-yl)-n'-[2-(1h-indol-3-yl)ethyl]-6-methoxy-1,3,5-triazine-2,4-diamineHuman1382
PAK4STE20STE4figAphosphoaminophosphonic acid-adenylate esterHuman1392
PAK4STE20STE7s48AA-Human14492
PAK4STE20STE7s48AB-Human14491
PAK4STE20STE8yhkA-Human15260
PAK4STE20STE4jdhAA-Human1371
PAK4STE20STE2cdzABn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman1374
PAK4STE20STE4o0xA1-{[1-(4-amino-1,3,5-triazin-2-yl)-2-methyl-1h-benzimidazol-6-yl]ethynyl}cyclohexanolHuman1404
PAK4STE20STE2q0nAA-Human1393
PAK4STE20STE5bmsAn~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman1389
PAK4STE20STE4o0yA4-[1-(4-amino-1,3,5-triazin-2-yl)-2-(ethylamino)-1h-benzimidazol-6-yl]-2-methylbut-3-yn-2-olHuman1388
PAK4STE20STE7cmbA1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indole-3-carboxamideHuman13818
PAK4STE20STE4jdjAA-Human1400
PAK4STE20STE5xvaA[6-chloranyl-4-[(5-methyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl]-[(3r)-3-methylpiperazin-1-yl]methanoneHuman9550
PAK4STE20STE4xbuA-Human6256
PAK4STE20STE4fieAphosphoaminophosphonic acid-adenylate esterHuman1405
PAK4STE20STE4fijA-Human1408
PAK4STE20STE5upkBphosphoaminophosphonic acid-adenylate esterHuman9435
PAK4STE20STE4jdkAA-Human1375
PAK4STE20STE4jdkAB-Human1398
PAK4STE20STE4fifABphosphoaminophosphonic acid-adenylate esterHuman1370
PAK4STE20STE5zjwAA(3z)-n-[(1s)-2-hydroxy-1-phenylethyl]-3-[(1h-imidazol-2-yl)(phenyl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamideHuman10999
PAK4STE20STE4fifBBphosphoaminophosphonic acid-adenylate esterHuman1379
PAK4STE20STE6wlxAB-Human12400
PAK4STE20STE7s47AAphosphoaminophosphonic acid-adenylate esterHuman14493
PAK4STE20STE4appABn-[6,6-dimethyl-5-[(2s)-4-methyl-2-(phenylmethyl)piperazin-1-yl]carbonyl-2,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-phenoxy-benzamideHuman1390
PAK4STE20STE2cdzAAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman1378
PAK4STE20STE4fieBphosphoaminophosphonic acid-adenylate esterHuman1372
PAK4STE20STE7cp3A[(3r)-3-azanylpiperidin-1-yl]-[1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]methanoneHuman13849
PAK4STE20STE4jdjAB-Human1397
PAK4STE20STE4o0vA1-({1-(2-aminopyrimidin-4-yl)-2-[(2-methoxyethyl)amino]-1h-benzimidazol-6-yl}ethynyl)cyclohexanolHuman1386
PAK4STE20STE2q0nAB-Human1401
PAK4STE20STE8ahgAB~{n}-methyl-3-propan-2-yl-1~{h}-pyrazolo[3,4-c]pyridine-4-carboxamideHuman14368
PAK4STE20STE5i0bA6-bromo-2-[1-methyl-3-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridineHuman7315
PAK4STE20STE8ahiA~{n}-methyl-1,3-benzothiazole-6-carboxamideHuman14369
PAK4STE20STE4jdiABphosphoaminophosphonic acid-adenylate esterHuman1380
PAK4STE20STE4fiiAB-Human1396
PAK4STE20STE6wlyAB-Human12396
PAK4STE20STE4appAAn-[6,6-dimethyl-5-[(2s)-4-methyl-2-(phenylmethyl)piperazin-1-yl]carbonyl-2,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-phenoxy-benzamideHuman1385
PAK4STE20STE4fiiAA-Human1383
PAK4STE20STE6wlyAA-Human12397
PAK4STE20STE5veeA6-(2,4-dichlorophenyl)-8-ethyl-2-{[3-fluoro-4-(piperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman8572
PAK4STE20STE8ahgAA~{n}-methyl-3-propan-2-yl-1~{h}-pyrazolo[3,4-c]pyridine-4-carboxamideHuman14370
PAK4STE20STE5vefAB5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman8571
PAK4STE20STE4jdhAB-Human1406
PAK4STE20STE2bvaA-Human1394
PAK4STE20STE5uplA-Human9436
PAK4STE20STE2bvaB-Human1407
PAK4STE20STE5xvfA2-(4-azanylpiperidin-1-yl)-6-chloranyl-n-(1-methylimidazol-4-yl)quinazolin-4-amineHuman9549
PAK4STE20STE4figBphosphoaminophosphonic acid-adenylate esterHuman1373
PAK4STE20STE5zjwAB(3z)-n-[(1s)-2-hydroxy-1-phenylethyl]-3-[(1h-imidazol-2-yl)(phenyl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamideHuman11000
PAK4STE20STE6wlyAC-Human12398
PAK4STE20STE2j0iAB-Human1377
PAK4STE20STE4fihAA-Human1399
PAK4STE20STE5xvgA[6-chloranyl-4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl]-[(3r)-3-methylpiperazin-1-yl]methanoneHuman9551
PAK4STE20STE2x4zApf-3758309Human1387
PAK4STE20STE4xbrAadenosine-5'-triphosphateHuman6257
PAK4STE20STE6wlxAA-Human12399
PAK4STE20STE5vefAA5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman8569
PAK4STE20STE7cp4A[1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]-[(3s)-3-methylpiperazin-1-yl]methanoneHuman13850
PAK4STE20STE5vedAstaurosporineHuman8570
PAK4STE20STE8ahhAB5-cyano-~{n}-methyl-pyrazolo[1,5-a]pyridine-3-carboxamideHuman14371
PAK4STE20STE4njdABn-(1h-indazol-5-yl)-n'-[2-(1h-indol-3-yl)ethyl]-6-methoxy-1,3,5-triazine-2,4-diamineHuman1384
PAK4STE20STE4jdiAAphosphoaminophosphonic acid-adenylate esterHuman1403
PAK4STE20STE4fifAAphosphoaminophosphonic acid-adenylate esterHuman1395
PAK4STE20STE7s47ABphosphoaminophosphonic acid-adenylate esterHuman14494
PAK4STE20STE4fihAB-Human1402
PAK4STE20STE7s46Aphosphoaminophosphonic acid-adenylate esterHuman14495
PAK4STE20STE8ahhAA5-cyano-~{n}-methyl-pyrazolo[1,5-a]pyridine-3-carboxamideHuman14372
PAK4STE20STE2j0iAA-Human1391
PAK4STE20STE4fifBAphosphoaminophosphonic acid-adenylate esterHuman1381