| FGFR4 | FGFR | TK | 5jkg | A | | 2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanol | Human | 7089 | |
| FGFR4 | FGFR | TK | 7ybp | A | | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14500 | |
| FGFR4 | FGFR | TK | 6jpj | A | | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 11051 | |
| FGFR4 | FGFR | TK | 6nvh | A | A | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11388 | |
| FGFR4 | FGFR | TK | 6nvi | A | B | n-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamide | Human | 11389 | |
| FGFR4 | FGFR | TK | 4tyg | A | B | - | Human | 933 | |
| FGFR4 | FGFR | TK | 4xcu | A | A | n-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamide | Human | 928 | |
| FGFR4 | FGFR | TK | 7wct | A | | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | 14167 | |
| FGFR4 | FGFR | TK | 4tyi | A | | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 926 | |
| FGFR4 | FGFR | TK | 6v9c | A | A | n-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamide | Human | 12096 | |
| FGFR4 | FGFR | TK | 5nwz | A | | ~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamide | Human | 9789 | |
| FGFR4 | FGFR | TK | 7ybo | A | | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14499 | |
| FGFR4 | FGFR | TK | 6nvk | A | B | n-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamide | Human | 11390 | |
| FGFR4 | FGFR | TK | 5xff | A | | 2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanol | Human | 10375 | |
| FGFR4 | FGFR | TK | 4qqc | A | B | n-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamide | Human | 932 | |
| FGFR4 | FGFR | TK | 4qqt | A | | - | Human | 922 | |
| FGFR4 | FGFR | TK | 4qqj | A | | - | Human | 935 | |
| FGFR4 | FGFR | TK | 6jpe | A | | n-[2-[[6-[2-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]amino]pyridin-3-yl]pyrimidin-4-yl]amino]-3-methyl-phenyl]prop-2-enamide | Human | 12230 | |
| FGFR4 | FGFR | TK | 5nud | B | | 3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amine | Human | 9790 | |
| FGFR4 | FGFR | TK | 7yc3 | A | | 6-bromanyl-~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14501 | |
| FGFR4 | FGFR | TK | 4tyg | A | A | - | Human | 929 | |
| FGFR4 | FGFR | TK | 6nvj | A | | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-fluorophenyl]propanamide | Human | 11391 | |
| FGFR4 | FGFR | TK | 5nud | A | | 3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amine | Human | 9787 | |
| FGFR4 | FGFR | TK | 7vjl | A | | n-[5-(aminomethyl)-4-(2-methoxyethylamino)pyridin-2-yl]-7-[2,2,2-tris(fluoranyl)ethanoyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 14109 | |
| FGFR4 | FGFR | TK | 4qqc | A | A | n-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamide | Human | 934 | |
| FGFR4 | FGFR | TK | 6yi8 | A | B | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12811 | |
| FGFR4 | FGFR | TK | 6yi8 | B | A | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12813 | |
| FGFR4 | FGFR | TK | 6yi8 | B | B | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12814 | |
| FGFR4 | FGFR | TK | 6iup | A | B | n-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamide | Human | 11796 | |
| FGFR4 | FGFR | TK | 4r6v | A | | n-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamide | Human | 931 | |
| FGFR4 | FGFR | TK | 6nvi | A | A | n-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamide | Human | 11392 | |
| FGFR4 | FGFR | TK | 4uxq | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 930 | |
| FGFR4 | FGFR | TK | 4tye | A | | - | Human | 927 | |
| FGFR4 | FGFR | TK | 6nvk | A | A | n-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamide | Human | 11395 | |
| FGFR4 | FGFR | TK | 5nwz | B | | ~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamide | Human | 9788 | |
| FGFR4 | FGFR | TK | 4xcu | A | B | n-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamide | Human | 924 | |
| FGFR4 | FGFR | TK | 7dtz | A | | n-[2-[[5-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]methoxy]pyrimidin-2-yl]amino]-3-methyl-phenyl]-2-fluoranyl-prop-2-enamide | Human | 13506 | |
| FGFR4 | FGFR | TK | 6iuo | A | | n-({4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}methyl)prop-2-enamide | Human | 11757 | |
| FGFR4 | FGFR | TK | 7v29 | A | | n-[2-[[3-(3,5-dimethoxyphenyl)-2-oxidanylidene-1-[3-(4-propanoylpiperazin-1-yl)propyl]-4h-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]propanamide | Human | 14165 | |
| FGFR4 | FGFR | TK | 6nvg | A | | n-[3,5-dichloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)phenyl]propanamide | Human | 11394 | |
| FGFR4 | FGFR | TK | 4qrc | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 923 | |
| FGFR4 | FGFR | TK | 6v9c | A | B | n-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamide | Human | 12095 | |
| FGFR4 | FGFR | TK | 7wcw | A | | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | 14168 | |
| FGFR4 | FGFR | TK | 6yi8 | A | A | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12812 | |
| FGFR4 | FGFR | TK | 7f3m | A | | 6-[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]-2-(methylamino)-8-[3-(4-prop-2-enoylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidin-7-one | Human | 14034 | |
| FGFR4 | FGFR | TK | 7wcx | A | | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | 14166 | |
| FGFR4 | FGFR | TK | 4qq5 | A | | n-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamide | Human | 921 | |
| FGFR4 | FGFR | TK | 7ybx | A | | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14502 | |
| FGFR4 | FGFR | TK | 6iup | A | A | n-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamide | Human | 11797 | |
| FGFR4 | FGFR | TK | 8kh6 | A | | - | Human | 15287 | |
| FGFR4 | FGFR | TK | 8w5c | A | | - | Human | 15288 | |
| FGFR4 | FGFR | TK | 8kh9 | A | | - | Human | 15284 | |
| FGFR4 | FGFR | TK | 8kh7 | A | | - | Human | 15286 | |
| FGFR4 | FGFR | TK | 7yc1 | A | | ~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-propyl-pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14498 | |
| FGFR4 | FGFR | TK | 4tyj | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 925 | |
| FGFR4 | FGFR | TK | 5xfj | A | | 2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanol | Human | 10376 | |
| FGFR4 | FGFR | TK | 6nvh | A | B | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11393 | |
| FGFR4 | FGFR | TK | 8kh8 | A | | - | Human | 15285 | |