| DYRK1A | DYRK | CMGC | 6ej4 | A | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10520 | 0.41 | |
| DYRK1A | DYRK | CMGC | 6eif | A | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10534 | 0.41 | |
| ABL1 | Abl | TK | 8h7h | A | | 5-[3-(6-methoxyisoquinolin-7-yl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n}-methyl-~{n}-prop-2-ynyl-pyridine-3-carboxamide | Human | 14666 | 0.57 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | B | A | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9786 | 0.42 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5737 | 0.41 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5726 | 0.41 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5707 | 1.00 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5704 | 0.41 | |
| Abl1 (ABL1) | Abl | TK | 2z60 | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5735 | 1.00 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5712 | 0.41 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5718 | 0.41 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5729 | 0.41 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5725 | 0.41 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | A | B | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9783 | 0.42 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5714 | 0.41 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | B | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5716 | 1.00 | |
| JAK3 | JakA | TK | 7apf | B | B | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13132 | 0.40 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6bku | A | | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 8687 | 0.41 | |
| DYRK1A | DYRK | CMGC | 6eif | B | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10544 | 0.41 | |
| ABL1 | Abl | TK | 7dt2 | A | | [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methanoyl-5-methoxy-phenyl]boronic acid | Human | 13621 | 0.67 | |
| ABL1 | Abl | TK | 7cc2 | A | | [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]boronic acid | Human | 13620 | 0.63 | |
| DYRK1A | DYRK | CMGC | 6eif | C | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10525 | 0.41 | |
| DYRK1A | DYRK | CMGC | 6ej4 | D | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10545 | 0.41 | |
| JAK3 | JakA | TK | 7apf | B | A | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13137 | 0.40 | |
| JAK3 | JakA | TK | 7apf | A | A | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13141 | 0.40 | |
| DYRK1A | DYRK | CMGC | 6ej4 | B | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10523 | 0.41 | |
| DYRK1A | DYRK | CMGC | 6ej4 | C | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10519 | 0.41 | |
| DYRK1A | DYRK | CMGC | 6eif | D | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10532 | 0.41 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | A | A | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9784 | 0.42 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | A | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9714 | 0.41 | |
| JAK3 | JakA | TK | 7apf | A | B | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13130 | 0.40 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | B | B | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9785 | 0.42 | |
| SGK1 | SGK | AGC | 3hdm | A | | 4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 3271 | 0.47 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | A | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9716 | 0.41 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | C | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9715 | 0.41 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | B | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9713 | 0.41 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | C | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9711 | 0.41 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | B | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9709 | 0.41 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | D | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9710 | 0.41 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | D | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9708 | 0.41 | |
| ABL1 | Abl | TK | 7w7y | A | | 5-[3-(5-methanoyl-2-methoxy-4-oxidanyl-phenyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n},~{n}-dimethyl-pyridine-3-carboxamide | Human | 14195 | 0.68 | |
| ABL1 | Abl | TK | 7w7x | A | | 5-[5-(dimethylcarbamoyl)pyridin-3-yl]-3-(5-fluorosulfonyloxy-2-methoxy-phenyl)-1h-pyrrolo[2,3-b]pyridine | Human | 14196 | 0.74 | |