| DYRK1A | DYRK | CMGC | 6ej4 | A | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10520 | 0.44 | |
| DYRK1A | DYRK | CMGC | 6eif | A | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10534 | 0.47 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zys | A | | n-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamide | Human | 1655 | 0.66 | |
| DYRK1A | DYRK | CMGC | 6eif | B | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10544 | 0.47 | |
| PIM1 | PIM | CAMK | 5mzl | A | A | ~{n}-quinolin-5-ylpyridine-3-carboxamide | Human | 9562 | 0.48 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh6 | A | | n-phenylpyridine-3-carboxamide | Human | 5083 | 0.40 | |
| ABL1 | Abl | TK | 7cc2 | A | | [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]boronic acid | Human | 13620 | 0.41 | |
| DYRK1A | DYRK | CMGC | 6eif | C | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10525 | 0.47 | |
| DYRK1A | DYRK | CMGC | 6ej4 | D | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10545 | 0.44 | |
| AAK1 | NAK | Other | 5l4q | A | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6679 | 1.00 | |
| AAK1 | NAK | Other | 5l4q | B | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6678 | 1.00 | |
| AAK1 | NAK | Other | 5l4q | B | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6680 | 1.00 | |
| AAK1 | NAK | Other | 5l4q | A | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6677 | 1.00 | |
| DYRK1A | DYRK | CMGC | 6ej4 | B | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10523 | 0.44 | |
| DYRK1A | DYRK | CMGC | 6ej4 | C | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10519 | 0.44 | |
| DYRK1A | DYRK | CMGC | 6eif | D | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10532 | 0.47 | |
| GSK3B | GSK | CMGC | 8ff8 | A | | 2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamide | Human | 14763 | 0.42 | |
| SGK1 | SGK | AGC | 3hdm | A | | 4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 3271 | 0.44 | |
| PIM1 | PIM | CAMK | 5mzl | A | B | ~{n}-quinolin-5-ylpyridine-3-carboxamide | Human | 9563 | 0.48 | |
| MET | Met | TK | 4aoi | A | | 4-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-6-yl]benzenecarbonitrile | Human | 2958 | 0.41 | |