Search results (20 entries covering 10 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsSimilarity (MFP)File
DYRK1ADYRKCMGC6ej4A3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman105200.44
DYRK1ADYRKCMGC6eifA4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman105340.47
CHEK1 (CHK1)CAMKLCAMK1zysAn-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamideHuman16550.66
DYRK1ADYRKCMGC6eifB4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman105440.47
PIM1PIMCAMK5mzlAA~{n}-quinolin-5-ylpyridine-3-carboxamideHuman95620.48
MAPK14 (p38a)MAPKCMGC4eh6An-phenylpyridine-3-carboxamideHuman50830.40
ABL1AblTK7cc2A[4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]boronic acidHuman136200.41
DYRK1ADYRKCMGC6eifC4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman105250.47
DYRK1ADYRKCMGC6ej4D3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman105450.44
AAK1NAKOther5l4qAA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman66791.00
AAK1NAKOther5l4qBB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman66781.00
AAK1NAKOther5l4qBA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman66801.00
AAK1NAKOther5l4qAB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman66771.00
DYRK1ADYRKCMGC6ej4B3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman105230.44
DYRK1ADYRKCMGC6ej4C3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman105190.44
DYRK1ADYRKCMGC6eifD4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman105320.47
GSK3BGSKCMGC8ff8A2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamideHuman147630.42
SGK1SGKAGC3hdmA4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman32710.44
PIM1PIMCAMK5mzlAB~{n}-quinolin-5-ylpyridine-3-carboxamideHuman95630.48
METMetTK4aoiA4-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-6-yl]benzenecarbonitrileHuman29580.41